CN1714091A - 中位取代卟啉 - Google Patents

中位取代卟啉 Download PDF

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Publication number
CN1714091A
CN1714091A CNA2003801017372A CN200380101737A CN1714091A CN 1714091 A CN1714091 A CN 1714091A CN A2003801017372 A CNA2003801017372 A CN A2003801017372A CN 200380101737 A CN200380101737 A CN 200380101737A CN 1714091 A CN1714091 A CN 1714091A
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phenyl
porphyrin
oxygen
group
last
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Pending
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Chinese (zh)
Inventor
加布里奥·龙库奇
多娜塔·代
弗兰切斯卡·琼蒂尼
贾科莫·基蒂
达尼埃莱·尼斯特里
莉娅·凡泰蒂
瓦伦丁娜·帕斯凯塔
安纳利萨·科基
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DEI FRATELLI ALITTI DI ESERCIZIO SpA Soc
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DEI FRATELLI ALITTI DI ESERCIZIO SpA Soc
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Application filed by DEI FRATELLI ALITTI DI ESERCIZIO SpA Soc filed Critical DEI FRATELLI ALITTI DI ESERCIZIO SpA Soc
Publication of CN1714091A publication Critical patent/CN1714091A/zh
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/22Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains four or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K41/00Medicinal preparations obtained by treating materials with wave energy or particle radiation ; Therapies using these preparations
    • A61K41/0057Photodynamic therapy with a photosensitizer, i.e. agent able to produce reactive oxygen species upon exposure to light or radiation, e.g. UV or visible light; photocleavage of nucleic acids with an agent
    • A61K41/0071PDT with porphyrins having exactly 20 ring atoms, i.e. based on the non-expanded tetrapyrrolic ring system, e.g. bacteriochlorin, chlorin-e6, or phthalocyanines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02EREDUCTION OF GREENHOUSE GAS [GHG] EMISSIONS, RELATED TO ENERGY GENERATION, TRANSMISSION OR DISTRIBUTION
    • Y02E50/00Technologies for the production of fuel of non-fossil origin
    • Y02E50/10Biofuels, e.g. bio-diesel
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02EREDUCTION OF GREENHOUSE GAS [GHG] EMISSIONS, RELATED TO ENERGY GENERATION, TRANSMISSION OR DISTRIBUTION
    • Y02E50/00Technologies for the production of fuel of non-fossil origin
    • Y02E50/30Fuel from waste, e.g. synthetic alcohol or diesel

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Dermatology (AREA)
  • Epidemiology (AREA)
  • Molecular Biology (AREA)
  • Urology & Nephrology (AREA)
  • Biochemistry (AREA)
  • Vascular Medicine (AREA)
  • Virology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicinal Preparation (AREA)
  • Radiation-Therapy Devices (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
CNA2003801017372A 2002-10-21 2003-10-21 中位取代卟啉 Pending CN1714091A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ITFI2002A000200 2002-10-21
IT000200A ITFI20020200A1 (it) 2002-10-21 2002-10-21 Porfirine meso-sostituite.

Publications (1)

Publication Number Publication Date
CN1714091A true CN1714091A (zh) 2005-12-28

Family

ID=32104761

Family Applications (1)

Application Number Title Priority Date Filing Date
CNA2003801017372A Pending CN1714091A (zh) 2002-10-21 2003-10-21 中位取代卟啉

Country Status (17)

Country Link
US (2) US7947674B2 (enExample)
EP (1) EP1558616B2 (enExample)
JP (1) JP4751068B2 (enExample)
CN (1) CN1714091A (enExample)
AT (1) ATE387450T1 (enExample)
AU (1) AU2003278118B8 (enExample)
CA (1) CA2503223C (enExample)
CY (1) CY1107963T1 (enExample)
DE (1) DE60319406T3 (enExample)
DK (1) DK1558616T4 (enExample)
ES (1) ES2301840T5 (enExample)
IL (1) IL168104A0 (enExample)
IT (1) ITFI20020200A1 (enExample)
PT (1) PT1558616E (enExample)
SI (1) SI1558616T2 (enExample)
WO (1) WO2004035590A2 (enExample)
ZA (1) ZA200504102B (enExample)

Cited By (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102159569A (zh) * 2008-09-18 2011-08-17 塞拉莫普泰克工业公司 用于pdt的不对称内消旋取代的卟啉和二氢卟酚的新方法及其应用
CN102180881A (zh) * 2011-03-25 2011-09-14 西北农林科技大学 3,8,13-三碘-5,10,15-三烷基三聚吲哚的制备方法
CN102499924A (zh) * 2011-11-23 2012-06-20 中国医学科学院生物医学工程研究所 二乙撑三胺五乙酸或乙二胺四乙酸或胺三乙酸修饰卟啉的用途
CN104725388A (zh) * 2015-03-25 2015-06-24 南京林业大学 一种meso位芳胺基单取代卟啉衍生物及其制备方法
CN105924448A (zh) * 2016-06-27 2016-09-07 桂林理工大学 苯并菲己烷氧基桥连十二烷氧基苯基卟啉金属Ni配合物的合成方法
CN105949208A (zh) * 2016-06-27 2016-09-21 桂林理工大学 苯并菲己烷氧基桥连十二烷氧基苯基卟啉金属Zn配合物的合成方法
CN106046010A (zh) * 2016-06-27 2016-10-26 桂林理工大学 5‑对苯甲酸基‑10, 15, 20‑三对异辛烷氧基苯基卟啉的合成方法
CN106047369A (zh) * 2016-06-27 2016-10-26 桂林理工大学 苯并菲己烷氧基桥连十二烷氧基苯基卟啉二元化合物盘状液晶材料的合成方法
CN106117227A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲癸烷氧基桥连十二烷氧基苯基卟啉二元化合物盘状液晶材料的合成方法
CN106117222A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲十二烷氧基桥连异辛烷氧基苯基卟啉二元化合物盘状液晶材料合成方法
CN106118688A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲癸烷氧基桥连异辛烷氧基苯基卟啉二元化合物盘状液晶材料的合成方法
CN106117228A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲癸烷氧基桥连异辛烷氧基苯基卟啉金属Ni配合物的合成方法
CN106117221A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲己烷氧基桥连异辛烷氧基苯基卟啉金属Ni配合物的合成方法
CN106117224A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲十二烷氧基桥连十二烷氧基苯基卟啉二元化合物盘状液晶材料的合成方法
CN106117225A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲癸烷氧基桥连异辛烷氧基苯基卟啉金属Zn配合物的合成方法
CN106117223A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲十二烷氧基桥连异辛烷氧基苯基卟啉金属Ni配合物的合成方法
CN106117220A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲十二烷氧基桥连异辛烷氧基苯基卟啉金属Zn配合物的合成方法
CN106118689A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲己烷氧基桥连异辛烷氧基苯基卟啉二元化合物盘状液晶材料的合成方法
CN106146523A (zh) * 2016-06-27 2016-11-23 桂林理工大学 苯并菲十二烷氧基桥连十二烷氧基苯基卟啉金属Ni配合物的合成方法
CN106146522A (zh) * 2016-06-27 2016-11-23 桂林理工大学 苯并菲癸烷氧基桥连十二烷氧基苯基卟啉金属Ni配合物的合成方法
CN106588941A (zh) * 2016-12-08 2017-04-26 桂林理工大学 苯并菲十二烷氧基桥连四苯基卟啉三元化合物盘状液晶材料的合成方法
CN106588942A (zh) * 2016-12-08 2017-04-26 桂林理工大学 并菲癸氧基桥连四苯基卟啉三元化合物盘状液晶材料的合成方法
CN106588940A (zh) * 2016-12-08 2017-04-26 桂林理工大学 苯并菲癸氧基桥连异辛烷氧基苯基卟啉三元化合物盘状液晶材料的合成方法
CN106749285A (zh) * 2016-12-08 2017-05-31 桂林理工大学 苯并菲己氧基桥连异辛烷氧基苯基卟啉三元化合物盘状液晶材料的合成方法
CN106749284A (zh) * 2016-12-08 2017-05-31 桂林理工大学 苯并菲十二烷氧基桥连异辛烷氧基苯基卟啉三元化合物盘状液晶材料的合成方法
CN106905334A (zh) * 2017-04-22 2017-06-30 桂林理工大学 苯并菲十二烷氧基桥连甲氧羰基苯基卟啉金属Zn配合物的合成方法
CN106967075A (zh) * 2017-04-22 2017-07-21 桂林理工大学 苯并菲癸烷氧基桥连甲氧羰基苯基卟啉金属Zn配合物的合成方法
CN107011349A (zh) * 2017-04-22 2017-08-04 桂林理工大学 苯并菲癸烷氧基桥连异辛烷氧基苯基卟啉金属Zn配合物的合成方法
CN107043381A (zh) * 2017-04-22 2017-08-15 桂林理工大学 苯并菲十二烷氧基桥连异辛烷氧基苯基卟啉金属Zn配合物的合成方法
CN107089987A (zh) * 2017-04-22 2017-08-25 桂林理工大学 苯并菲己烷氧基桥连异辛烷氧基苯基卟啉金属Zn配合物的合成方法
CN110354770A (zh) * 2019-07-23 2019-10-22 中国石油大学(华东) 一种人工光合微反应器及制备方法

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EP1356813B1 (en) * 2002-04-25 2005-07-20 L. MOLTENI & C. DEI FRATELLI ALITTI SOCIETA' DI ESERCIZIO SOCIETA' PER AZIONI Antibacterial compositions comprising metal phthalocyanine analogues
ITFI20020200A1 (it) * 2002-10-21 2004-04-22 Molteni & C Dei Flii Alitti S P A Societa L Porfirine meso-sostituite.
GB2397067B (en) * 2002-12-23 2005-05-11 Destiny Pharma Ltd Porphin & azaporphin derivatives with at least one cationic-nitrogen-containing meso-substituent for use in photodynamic therapy & in vitro sterilisation
CA2528347A1 (en) * 2003-06-06 2005-01-06 Eukarion, Inc. Orally bioavailable low molecular weight metalloporphyrins as antioxidants
GB2415372A (en) * 2004-06-23 2005-12-28 Destiny Pharma Ltd Non photodynamical or sonodynamical antimicrobial use of porphyrins and azaporphyrins containing at least one cationic-nitrogen-containing substituent
GB2415373A (en) * 2004-06-23 2005-12-28 Destiny Pharma Ltd Porphyrins for sonodynamic therapy
GB0526474D0 (en) * 2005-12-24 2006-02-08 Destiny Pharma Ltd Novel process
WO2008108937A1 (en) 2007-03-05 2008-09-12 North Carolina State University Method of making porphyrins
EP2759546B1 (en) * 2011-09-21 2018-03-21 National University Corporation Okayama University Metalloporphyrin complex, manufacturing process therefor and its use as carbon dioxide fixation catalyst, as well as process for manufacturing cyclic carbonate
US9364537B2 (en) * 2014-08-22 2016-06-14 University Of Dayton Transition metal porphyrin complexes and methods of treatment using same
KR20180100570A (ko) * 2016-01-13 2018-09-11 제이에스알 가부시끼가이샤 감방사선성 수지 조성물, 레지스트 패턴 형성 방법, 산 확산 제어제 및 화합물
US10722582B2 (en) * 2018-04-12 2020-07-28 Purdue Research Foundation Targeted antimicrobial photodynamic therapy

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GB2397067B (en) 2002-12-23 2005-05-11 Destiny Pharma Ltd Porphin & azaporphin derivatives with at least one cationic-nitrogen-containing meso-substituent for use in photodynamic therapy & in vitro sterilisation

Cited By (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102159569A (zh) * 2008-09-18 2011-08-17 塞拉莫普泰克工业公司 用于pdt的不对称内消旋取代的卟啉和二氢卟酚的新方法及其应用
CN102159569B (zh) * 2008-09-18 2016-02-03 拜莱泰克制药市场有限公司 用于pdt的不对称内消旋取代的卟啉和二氢卟酚及其应用
CN102180881A (zh) * 2011-03-25 2011-09-14 西北农林科技大学 3,8,13-三碘-5,10,15-三烷基三聚吲哚的制备方法
CN102499924A (zh) * 2011-11-23 2012-06-20 中国医学科学院生物医学工程研究所 二乙撑三胺五乙酸或乙二胺四乙酸或胺三乙酸修饰卟啉的用途
CN104725388A (zh) * 2015-03-25 2015-06-24 南京林业大学 一种meso位芳胺基单取代卟啉衍生物及其制备方法
CN104725388B (zh) * 2015-03-25 2017-03-15 南京林业大学 一种meso位芳胺基单取代卟啉衍生物及其制备方法
CN106117223A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲十二烷氧基桥连异辛烷氧基苯基卟啉金属Ni配合物的合成方法
CN106146523A (zh) * 2016-06-27 2016-11-23 桂林理工大学 苯并菲十二烷氧基桥连十二烷氧基苯基卟啉金属Ni配合物的合成方法
CN106047369A (zh) * 2016-06-27 2016-10-26 桂林理工大学 苯并菲己烷氧基桥连十二烷氧基苯基卟啉二元化合物盘状液晶材料的合成方法
CN106117227A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲癸烷氧基桥连十二烷氧基苯基卟啉二元化合物盘状液晶材料的合成方法
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