SI1558616T1 - Meso-substituirani porfirini - Google Patents

Meso-substituirani porfirini

Info

Publication number
SI1558616T1
SI1558616T1 SI200331212T SI200331212T SI1558616T1 SI 1558616 T1 SI1558616 T1 SI 1558616T1 SI 200331212 T SI200331212 T SI 200331212T SI 200331212 T SI200331212 T SI 200331212T SI 1558616 T1 SI1558616 T1 SI 1558616T1
Authority
SI
Slovenia
Prior art keywords
meso
substituted porphyrins
porphyrins
substituted
general formula
Prior art date
Application number
SI200331212T
Other languages
English (en)
Other versions
SI1558616T2 (sl
Inventor
Gabrio Roncucci
Donata Dei
Francesca Giuntini
Giacomo Chiti
Daniele Nistri
Lia Fantetti
Valentina Paschetta
Annalisa Cocchi
Original Assignee
Molteni & C
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32104761&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI1558616(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Molteni & C filed Critical Molteni & C
Publication of SI1558616T1 publication Critical patent/SI1558616T1/sl
Publication of SI1558616T2 publication Critical patent/SI1558616T2/sl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/22Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains four or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K41/00Medicinal preparations obtained by treating materials with wave energy or particle radiation ; Therapies using these preparations
    • A61K41/0057Photodynamic therapy with a photosensitizer, i.e. agent able to produce reactive oxygen species upon exposure to light or radiation, e.g. UV or visible light; photocleavage of nucleic acids with an agent
    • A61K41/0071PDT with porphyrins having exactly 20 ring atoms, i.e. based on the non-expanded tetrapyrrolic ring system, e.g. bacteriochlorin, chlorin-e6, or phthalocyanines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02EREDUCTION OF GREENHOUSE GAS [GHG] EMISSIONS, RELATED TO ENERGY GENERATION, TRANSMISSION OR DISTRIBUTION
    • Y02E50/00Technologies for the production of fuel of non-fossil origin
    • Y02E50/10Biofuels, e.g. bio-diesel
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02EREDUCTION OF GREENHOUSE GAS [GHG] EMISSIONS, RELATED TO ENERGY GENERATION, TRANSMISSION OR DISTRIBUTION
    • Y02E50/00Technologies for the production of fuel of non-fossil origin
    • Y02E50/30Fuel from waste, e.g. synthetic alcohol or diesel

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Dermatology (AREA)
  • Biochemistry (AREA)
  • Epidemiology (AREA)
  • Urology & Nephrology (AREA)
  • Molecular Biology (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Diabetes (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicinal Preparation (AREA)
  • Radiation-Therapy Devices (AREA)
SI200331212T 2002-10-21 2003-10-21 Meso-substituirani porfirini SI1558616T2 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IT000200A ITFI20020200A1 (it) 2002-10-21 2002-10-21 Porfirine meso-sostituite.
EP03769429A EP1558616B2 (en) 2002-10-21 2003-10-21 Meso-substituted porphyrins
PCT/EP2003/011642 WO2004035590A2 (en) 2002-10-21 2003-10-21 Meso-substituted porphyrins

Publications (2)

Publication Number Publication Date
SI1558616T1 true SI1558616T1 (sl) 2008-08-31
SI1558616T2 SI1558616T2 (sl) 2011-12-30

Family

ID=32104761

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200331212T SI1558616T2 (sl) 2002-10-21 2003-10-21 Meso-substituirani porfirini

Country Status (17)

Country Link
US (2) US7947674B2 (sl)
EP (1) EP1558616B2 (sl)
JP (1) JP4751068B2 (sl)
CN (1) CN1714091A (sl)
AT (1) ATE387450T1 (sl)
AU (1) AU2003278118B8 (sl)
CA (1) CA2503223C (sl)
CY (1) CY1107963T1 (sl)
DE (1) DE60319406T3 (sl)
DK (1) DK1558616T4 (sl)
ES (1) ES2301840T5 (sl)
IL (1) IL168104A0 (sl)
IT (1) ITFI20020200A1 (sl)
PT (1) PT1558616E (sl)
SI (1) SI1558616T2 (sl)
WO (1) WO2004035590A2 (sl)
ZA (1) ZA200504102B (sl)

Families Citing this family (43)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK1356813T3 (da) * 2002-04-25 2005-12-05 Molteni & C Antibakterielle præparater der omfatter metal-phthalocyaninanaloger
ITFI20020200A1 (it) * 2002-10-21 2004-04-22 Molteni & C Dei Flii Alitti S P A Societa L Porfirine meso-sostituite.
GB2397067B (en) 2002-12-23 2005-05-11 Destiny Pharma Ltd Porphin & azaporphin derivatives with at least one cationic-nitrogen-containing meso-substituent for use in photodynamic therapy & in vitro sterilisation
AU2004252078A1 (en) * 2003-06-06 2005-01-06 Eukarion, Inc. Orally bioavailable low molecular weight metalloporphyrins as antioxidants
GB2415372A (en) * 2004-06-23 2005-12-28 Destiny Pharma Ltd Non photodynamical or sonodynamical antimicrobial use of porphyrins and azaporphyrins containing at least one cationic-nitrogen-containing substituent
GB2415373A (en) * 2004-06-23 2005-12-28 Destiny Pharma Ltd Porphyrins for sonodynamic therapy
GB0526474D0 (en) * 2005-12-24 2006-02-08 Destiny Pharma Ltd Novel process
WO2008108937A1 (en) 2007-03-05 2008-09-12 North Carolina State University Method of making porphyrins
ES2932287T3 (es) * 2008-09-18 2023-01-17 Biolitec Unternehmensberatungs Ii Ag Método y aplicación novedosos de porfirinas y clorinas meso-sustituidas asimétricamente para TFD
CN102180881A (zh) * 2011-03-25 2011-09-14 西北农林科技大学 3,8,13-三碘-5,10,15-三烷基三聚吲哚的制备方法
CN103987714B (zh) * 2011-09-21 2016-03-16 国立大学法人冈山大学 金属卟啉配位化合物、其制造方法及由其构成的二氧化碳固定化催化剂、以及环状碳酸酯的制造方法
CN102499924B (zh) * 2011-11-23 2013-07-24 中国医学科学院生物医学工程研究所 二乙撑三胺五乙酸或乙二胺四乙酸或胺三乙酸修饰卟啉的用途
US9364537B2 (en) * 2014-08-22 2016-06-14 University Of Dayton Transition metal porphyrin complexes and methods of treatment using same
CN104725388B (zh) * 2015-03-25 2017-03-15 南京林业大学 一种meso位芳胺基单取代卟啉衍生物及其制备方法
WO2017122697A1 (ja) * 2016-01-13 2017-07-20 Jsr株式会社 感放射線性樹脂組成物、レジストパターン形成方法、酸拡散制御剤及び化合物
CN105949208A (zh) * 2016-06-27 2016-09-21 桂林理工大学 苯并菲己烷氧基桥连十二烷氧基苯基卟啉金属Zn配合物的合成方法
CN106117227A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲癸烷氧基桥连十二烷氧基苯基卟啉二元化合物盘状液晶材料的合成方法
CN106118688A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲癸烷氧基桥连异辛烷氧基苯基卟啉二元化合物盘状液晶材料的合成方法
CN106117223A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲十二烷氧基桥连异辛烷氧基苯基卟啉金属Ni配合物的合成方法
CN106117222A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲十二烷氧基桥连异辛烷氧基苯基卟啉二元化合物盘状液晶材料合成方法
CN106146523A (zh) * 2016-06-27 2016-11-23 桂林理工大学 苯并菲十二烷氧基桥连十二烷氧基苯基卟啉金属Ni配合物的合成方法
CN106117220A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲十二烷氧基桥连异辛烷氧基苯基卟啉金属Zn配合物的合成方法
CN106117228A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲癸烷氧基桥连异辛烷氧基苯基卟啉金属Ni配合物的合成方法
CN106118689A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲己烷氧基桥连异辛烷氧基苯基卟啉二元化合物盘状液晶材料的合成方法
CN106046010A (zh) * 2016-06-27 2016-10-26 桂林理工大学 5‑对苯甲酸基‑10, 15, 20‑三对异辛烷氧基苯基卟啉的合成方法
CN106117221A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲己烷氧基桥连异辛烷氧基苯基卟啉金属Ni配合物的合成方法
CN105924448A (zh) * 2016-06-27 2016-09-07 桂林理工大学 苯并菲己烷氧基桥连十二烷氧基苯基卟啉金属Ni配合物的合成方法
CN106117225A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲癸烷氧基桥连异辛烷氧基苯基卟啉金属Zn配合物的合成方法
CN106117224A (zh) * 2016-06-27 2016-11-16 桂林理工大学 苯并菲十二烷氧基桥连十二烷氧基苯基卟啉二元化合物盘状液晶材料的合成方法
CN106146522A (zh) * 2016-06-27 2016-11-23 桂林理工大学 苯并菲癸烷氧基桥连十二烷氧基苯基卟啉金属Ni配合物的合成方法
CN106047369A (zh) * 2016-06-27 2016-10-26 桂林理工大学 苯并菲己烷氧基桥连十二烷氧基苯基卟啉二元化合物盘状液晶材料的合成方法
CN106749284A (zh) * 2016-12-08 2017-05-31 桂林理工大学 苯并菲十二烷氧基桥连异辛烷氧基苯基卟啉三元化合物盘状液晶材料的合成方法
CN106588942A (zh) * 2016-12-08 2017-04-26 桂林理工大学 并菲癸氧基桥连四苯基卟啉三元化合物盘状液晶材料的合成方法
CN106749285A (zh) * 2016-12-08 2017-05-31 桂林理工大学 苯并菲己氧基桥连异辛烷氧基苯基卟啉三元化合物盘状液晶材料的合成方法
CN106588940A (zh) * 2016-12-08 2017-04-26 桂林理工大学 苯并菲癸氧基桥连异辛烷氧基苯基卟啉三元化合物盘状液晶材料的合成方法
CN106588941A (zh) * 2016-12-08 2017-04-26 桂林理工大学 苯并菲十二烷氧基桥连四苯基卟啉三元化合物盘状液晶材料的合成方法
CN106967075A (zh) * 2017-04-22 2017-07-21 桂林理工大学 苯并菲癸烷氧基桥连甲氧羰基苯基卟啉金属Zn配合物的合成方法
CN106905334A (zh) * 2017-04-22 2017-06-30 桂林理工大学 苯并菲十二烷氧基桥连甲氧羰基苯基卟啉金属Zn配合物的合成方法
CN107089987A (zh) * 2017-04-22 2017-08-25 桂林理工大学 苯并菲己烷氧基桥连异辛烷氧基苯基卟啉金属Zn配合物的合成方法
CN107043381A (zh) * 2017-04-22 2017-08-15 桂林理工大学 苯并菲十二烷氧基桥连异辛烷氧基苯基卟啉金属Zn配合物的合成方法
CN107011349A (zh) * 2017-04-22 2017-08-04 桂林理工大学 苯并菲癸烷氧基桥连异辛烷氧基苯基卟啉金属Zn配合物的合成方法
US10722582B2 (en) * 2018-04-12 2020-07-28 Purdue Research Foundation Targeted antimicrobial photodynamic therapy
CN110354770B (zh) * 2019-07-23 2022-10-04 中国石油大学(华东) 一种人工光合微反应器及制备方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8805849D0 (en) * 1988-03-11 1988-04-13 Efamol Holdings Porphyrins & cancer treatment
FR2632187B1 (fr) * 1988-06-02 1990-09-14 Centre Nat Rech Scient Derives de metalloporphyrines, leur preparation, leur application en therapeutique et leur utilisation pour la preparation de molecules hybrides
ATE306936T1 (de) * 1995-06-07 2005-11-15 Univ Duke Faenger fuer oxidantien
WO1998033503A1 (en) * 1997-02-05 1998-08-06 Board Of Regents, The University Of Texas System Porphyrin compounds as telomerase inhibitors
IT1294325B1 (it) 1997-08-14 1999-03-24 Molteni L E C Dei Fratelli Ali Zinco-ftalocianine e relativi coniugati, preparazione e uso nella terapia fotodinamica e come diagnostici
CA2341507C (en) * 1998-08-28 2011-05-24 William Guy Love Porphyrin derivatives, their use in photodynamic therapy and medical devices containing them
DE60008354T2 (de) * 2000-06-15 2004-12-09 L. Molteni & C. dei Fratelli Alitti Società di Esercizio S.p.A. Substituierte Metallphthalocyaninen, ihre Herstellung und Verwendung
FR2812637B1 (fr) * 2000-08-01 2002-10-25 Anulm Ass Nantaise Pour L Util Nouveaux composes derives de dihydroporphyrine et leurs applications
ES2244793T3 (es) 2001-03-21 2005-12-16 L. MOLTENI & C. DEI FRATELLI ALITTI SOCIETA' DI ESERCIZIO SOCIETA' PER AZIONI Analogos no centrosimetricos de ftalocianina sustituidos por metales, su preparacion y su utilizacion en terapia fotodinamica y diagnostico in vivo.
ITFI20020200A1 (it) * 2002-10-21 2004-04-22 Molteni & C Dei Flii Alitti S P A Societa L Porfirine meso-sostituite.
GB2397067B (en) * 2002-12-23 2005-05-11 Destiny Pharma Ltd Porphin & azaporphin derivatives with at least one cationic-nitrogen-containing meso-substituent for use in photodynamic therapy & in vitro sterilisation

Also Published As

Publication number Publication date
CA2503223C (en) 2010-11-23
DK1558616T3 (da) 2008-06-23
EP1558616A2 (en) 2005-08-03
IT1333697B (sl) 2006-05-09
ATE387450T1 (de) 2008-03-15
CA2503223A1 (en) 2004-04-29
JP4751068B2 (ja) 2011-08-17
WO2004035590A3 (en) 2004-07-29
ES2301840T5 (es) 2012-01-13
IL168104A0 (en) 2009-02-11
EP1558616B2 (en) 2011-08-24
ZA200504102B (en) 2006-07-26
JP2006512301A (ja) 2006-04-13
AU2003278118A1 (en) 2004-05-04
CY1107963T1 (el) 2013-09-04
ITFI20020200A1 (it) 2004-04-22
CN1714091A (zh) 2005-12-28
DE60319406T3 (de) 2012-02-23
DE60319406T2 (de) 2009-03-19
DE60319406D1 (de) 2008-04-10
DK1558616T4 (da) 2011-12-12
US8288528B2 (en) 2012-10-16
EP1558616B1 (en) 2008-02-27
US20060040914A1 (en) 2006-02-23
AU2003278118B2 (en) 2009-05-21
WO2004035590A2 (en) 2004-04-29
US20110112464A1 (en) 2011-05-12
SI1558616T2 (sl) 2011-12-30
AU2003278118B8 (en) 2009-09-17
US7947674B2 (en) 2011-05-24
ES2301840T3 (es) 2008-07-01
PT1558616E (pt) 2008-05-12

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