CN1714076A - 芳基脲基衍生物及其医药用途 - Google Patents

芳基脲基衍生物及其医药用途 Download PDF

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Publication number
CN1714076A
CN1714076A CNA200380103761XA CN200380103761A CN1714076A CN 1714076 A CN1714076 A CN 1714076A CN A200380103761X A CNA200380103761X A CN A200380103761XA CN 200380103761 A CN200380103761 A CN 200380103761A CN 1714076 A CN1714076 A CN 1714076A
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alkyl
cycloalkyl
halogen
phenyl
chloro
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Chinese (zh)
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J·瓦尔盖尔森
E·O·尼尔森
D·彼得斯
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NTG Nordic Transport Group AS
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Neurosearch AS
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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
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  • Engineering & Computer Science (AREA)
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  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Hospice & Palliative Care (AREA)
  • Diabetes (AREA)
  • Psychology (AREA)
  • Urology & Nephrology (AREA)
  • Immunology (AREA)
  • Vascular Medicine (AREA)
  • Obesity (AREA)
  • Child & Adolescent Psychology (AREA)
  • Addiction (AREA)
  • Ophthalmology & Optometry (AREA)
  • Otolaryngology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Indole Compounds (AREA)
CNA200380103761XA 2002-11-21 2003-11-10 芳基脲基衍生物及其医药用途 Pending CN1714076A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA200201803 2002-11-21
DKPA200201803 2002-11-21

Publications (1)

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CN1714076A true CN1714076A (zh) 2005-12-28

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US (1) US7521480B2 (enExample)
EP (1) EP1565429B1 (enExample)
JP (1) JP2006507329A (enExample)
CN (1) CN1714076A (enExample)
AT (1) ATE431335T1 (enExample)
AU (1) AU2003280308A1 (enExample)
CA (1) CA2502705A1 (enExample)
DE (1) DE60327652D1 (enExample)
ES (1) ES2327834T3 (enExample)
MX (1) MXPA05005409A (enExample)
NZ (1) NZ539499A (enExample)
PT (1) PT1565429E (enExample)
WO (1) WO2004046090A2 (enExample)

Cited By (5)

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Publication number Priority date Publication date Assignee Title
CN106008371A (zh) * 2016-06-24 2016-10-12 谢阳 1-芳基脲基环烷基-1-甲酰胺类化合物及其药物组合物和应用
CN106946786A (zh) * 2017-04-11 2017-07-14 白银澐新生物科技有限公司 一种1‑苄基‑3‑羟基‑1h‑3‑吲唑钠盐的制备方法
WO2017219935A1 (zh) * 2016-06-22 2017-12-28 复旦大学 联芳基脲类衍生物或其盐及其制备方法和用途
CN111116420A (zh) * 2019-12-31 2020-05-08 浙江工业大学 一种对称脲类化合物的制备方法
CN114539080A (zh) * 2022-03-02 2022-05-27 八叶草健康产业研究院(厦门)有限公司 一种2-(2-氨基-6-氯苯基)-乙酸钠的制备方法

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DE102004005172A1 (de) 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
US7550499B2 (en) 2004-05-12 2009-06-23 Bristol-Myers Squibb Company Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
CN101098852A (zh) * 2004-11-09 2008-01-02 史密丝克莱恩比彻姆公司 糖原磷酸化酶抑制剂化合物和其药物组合物
FR2878522B1 (fr) * 2004-12-01 2008-04-18 Merck Sante Soc Par Actions Si Nouveaux inhibiteurs specifiques de la caspas-10
CN101287456A (zh) * 2004-12-17 2008-10-15 神经研究公司 用作钾通道激活剂的二苯基脲衍生物
AU2006206611A1 (en) 2005-01-19 2006-07-27 Bristol-Myers Squibb Company 2-phenoxy-N- (1, 3 , 4-thiadizol-2-yl) pyridin-3-amine derivatives and related compounds as P2Y1 receptor inhibitors for the treatment of thromboembolic disorders
EP1899299B1 (en) 2005-06-27 2010-10-20 Bristol-Myers Squibb Company C-linked cyclic antagonists of p2y1 receptor useful in the treatment of thrombotic conditions
ES2360818T3 (es) 2005-06-27 2011-06-09 Bristol-Myers Squibb Company Miméticos de urea lineal antagonistas del receptor p2y, útiles en el tratamiento de afecciones trombóticas.
US7714002B2 (en) 2005-06-27 2010-05-11 Bristol-Myers Squibb Company Carbocycle and heterocycle antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
MX2007016501A (es) 2005-06-27 2008-03-06 Squibb Bristol Myers Co Antagonistas heterociclicos n-enlazados del receptor de p2y1, utiles en el tratamiento de condiciones tromboticas.
WO2007044724A2 (en) * 2005-10-06 2007-04-19 Exelixis, Inc. Aminopyrimidine, aminopyridine and aniline derivatives inhibitors of pim-i and/or pim-3
WO2007104719A1 (en) * 2006-03-14 2007-09-20 Neurosearch A/S Diphenylurea derivatives and their use as chloride channel blockers or bkca channel modulators
US7960569B2 (en) 2006-10-17 2011-06-14 Bristol-Myers Squibb Company Indole antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
DE102007012908A1 (de) 2007-03-19 2008-09-25 Momentive Performance Materials Gmbh Neue Polyamid-Polysiloxan-Verbindungen
AU2008309003A1 (en) * 2007-09-28 2009-04-09 Glaxosmithkline Llc Glycogen phosphorylase inhibitor compound and pharmaceutical composition thereof
US20100292283A1 (en) * 2007-11-28 2010-11-18 Antonio Nardi Novel phenyl-acetamide and phenyl-propionamide derivatives useful as potassium channel modulators
WO2011053468A1 (en) * 2009-10-30 2011-05-05 Sanofi-Aventis Amino-benzoic acid derivatives for use in the treatment of dihydrogenase-related disorders
US10899702B2 (en) * 2015-02-07 2021-01-26 University of Pittsburgh—of the Commonwealth System of Higher Education HTRPVI chemical agents

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ATE431335T1 (de) 2009-05-15
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