CN1681557A - 治疗碳酸酐酶介导的疾病的方法 - Google Patents
治疗碳酸酐酶介导的疾病的方法 Download PDFInfo
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- CN1681557A CN1681557A CNA038218801A CN03821880A CN1681557A CN 1681557 A CN1681557 A CN 1681557A CN A038218801 A CNA038218801 A CN A038218801A CN 03821880 A CN03821880 A CN 03821880A CN 1681557 A CN1681557 A CN 1681557A
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- hydrocarbyl
- alkyl
- halo
- carbonic anhydrase
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- A61K31/18—Sulfonamides
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Diabetes (AREA)
- Neurology (AREA)
- Hematology (AREA)
- Biomedical Technology (AREA)
- Ophthalmology & Optometry (AREA)
- Neurosurgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Cardiology (AREA)
- Pain & Pain Management (AREA)
- Immunology (AREA)
- Endocrinology (AREA)
- Rheumatology (AREA)
- Dermatology (AREA)
- Pulmonology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Reproductive Health (AREA)
- Urology & Nephrology (AREA)
- Obesity (AREA)
- Hospice & Palliative Care (AREA)
- Pregnancy & Childbirth (AREA)
- Emergency Medicine (AREA)
- Psychiatry (AREA)
- Transplantation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US10/213,793 US20030100594A1 (en) | 2001-08-10 | 2002-08-07 | Carbonic anhydrase inhibitor |
| US10/213,793 | 2002-08-07 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN1681557A true CN1681557A (zh) | 2005-10-12 |
Family
ID=31714232
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNA038218801A Pending CN1681557A (zh) | 2002-08-07 | 2003-02-14 | 治疗碳酸酐酶介导的疾病的方法 |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US20030100594A1 (https=) |
| EP (2) | EP1526869A1 (https=) |
| JP (2) | JP2005539022A (https=) |
| KR (1) | KR20050056189A (https=) |
| CN (1) | CN1681557A (https=) |
| AU (2) | AU2003225571A1 (https=) |
| BR (2) | BR0313282A (https=) |
| CA (2) | CA2495516A1 (https=) |
| IL (1) | IL166685A0 (https=) |
| MX (2) | MXPA05001496A (https=) |
| PL (1) | PL374994A1 (https=) |
| WO (2) | WO2004014430A1 (https=) |
Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102351793A (zh) * | 2011-08-30 | 2012-02-15 | 江苏正大清江制药有限公司 | 4-[3-(4-甲基苯基)-5-(三氟甲基)-1-氢-吡唑-1-基]苯磺酰胺的直接合成方法 |
| CN102574782A (zh) * | 2009-10-21 | 2012-07-11 | 拜耳医药股份有限公司 | 取代的卤代苯氧基苯甲酰胺衍生物 |
| CN109557309A (zh) * | 2018-12-04 | 2019-04-02 | 九江学院附属医院 | 碳酸酐酶-2作为检测标记物在肾结石诊断方面的应用 |
| CN111233786A (zh) * | 2020-02-04 | 2020-06-05 | 中国人民解放军军事科学院军事医学研究院 | 含五元杂环的苯磺酰胺类化合物及其制备方法和用途 |
Families Citing this family (43)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10035227A1 (de) * | 2000-07-20 | 2002-01-31 | Solvay Pharm Gmbh | Verfahren zum Auffinden von Verbindungen, welche zur Behandlung und/oder Prophylaxe von Fettleibigkeit geeignet sind |
| US6946243B2 (en) * | 2000-07-20 | 2005-09-20 | Solvay Pharmaceuticals Gmbh | Method of identifying compounds suitable for treatment and/or prophylaxis of obesity |
| US20100135980A1 (en) * | 2000-10-16 | 2010-06-03 | Rodriguez Victorio C | Therapeutic and prophylactic uses of cell specific carbonic anhydrase enzymes in treating aging, disorders of aging, cancer, as growth factors, and as an alternative to stem cell therapy |
| US20030220376A1 (en) * | 2001-08-10 | 2003-11-27 | Pharmacia Corporation | Methods for treating carbonic anhydrase mediated disorders |
| PT1636236E (pt) * | 2003-05-22 | 2013-12-16 | Nerviano Medical Sciences Srl | Derivados de pirazol-quinazolina, processo para sua preparação e sua utilização como inibidores de cinase |
| WO2005079781A1 (en) * | 2004-02-25 | 2005-09-01 | La Trobe University | Therapeutic and/or prophylactic method |
| WO2005094815A1 (en) * | 2004-03-30 | 2005-10-13 | Amorepacific Corporation | Dual inhibition of cyclooxygenase-2 and carbonic anhydrase |
| US7799336B2 (en) * | 2004-04-30 | 2010-09-21 | Allergan, Inc. | Hypotensive lipid-containing biodegradable intraocular implants and related methods |
| US8722097B2 (en) | 2004-04-30 | 2014-05-13 | Allergan, Inc. | Oil-in-water method for making polymeric implants containing a hypotensive lipid |
| US8673341B2 (en) | 2004-04-30 | 2014-03-18 | Allergan, Inc. | Intraocular pressure reduction with intracameral bimatoprost implants |
| US7993634B2 (en) | 2004-04-30 | 2011-08-09 | Allergan, Inc. | Oil-in-oil emulsified polymeric implants containing a hypotensive lipid and related methods |
| US9498457B2 (en) | 2004-04-30 | 2016-11-22 | Allergan, Inc. | Hypotensive prostamide-containing biodegradable intraocular implants and related implants |
| MY147767A (en) | 2004-06-16 | 2013-01-31 | Janssen Pharmaceutica Nv | Novel sulfamate and sulfamide derivatives useful for the treatment of epilepsy and related disorders |
| JP2008545650A (ja) | 2005-05-20 | 2008-12-18 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | スルファミド誘導体の製造方法 |
| JP4872076B2 (ja) * | 2005-09-15 | 2012-02-08 | 国立大学法人 長崎大学 | 硝子体可視化剤 |
| US20070155823A1 (en) * | 2005-12-19 | 2007-07-05 | Smith-Swintosky Virginia L | Use of benzo-fused heterocycle sulfamide derivatives as neuroprotective agents |
| US8937096B2 (en) | 2005-12-19 | 2015-01-20 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocyle sulfamide derivatives for the treatment of mania and bipolar disorder |
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Cited By (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102574782A (zh) * | 2009-10-21 | 2012-07-11 | 拜耳医药股份有限公司 | 取代的卤代苯氧基苯甲酰胺衍生物 |
| CN102574782B (zh) * | 2009-10-21 | 2014-10-08 | 拜耳知识产权有限责任公司 | 取代的卤代苯氧基苯甲酰胺衍生物 |
| CN102351793A (zh) * | 2011-08-30 | 2012-02-15 | 江苏正大清江制药有限公司 | 4-[3-(4-甲基苯基)-5-(三氟甲基)-1-氢-吡唑-1-基]苯磺酰胺的直接合成方法 |
| CN102351793B (zh) * | 2011-08-30 | 2013-11-06 | 江苏正大清江制药有限公司 | 4-[3-(4-甲基苯基)-5-(三氟甲基)-1-氢-吡唑-1-基]苯磺酰胺的直接合成方法 |
| CN109557309A (zh) * | 2018-12-04 | 2019-04-02 | 九江学院附属医院 | 碳酸酐酶-2作为检测标记物在肾结石诊断方面的应用 |
| CN109557309B (zh) * | 2018-12-04 | 2021-09-10 | 九江学院附属医院 | 碳酸酐酶-2作为检测标记物在肾结石诊断方面的应用 |
| CN111233786A (zh) * | 2020-02-04 | 2020-06-05 | 中国人民解放军军事科学院军事医学研究院 | 含五元杂环的苯磺酰胺类化合物及其制备方法和用途 |
| WO2021155781A1 (zh) * | 2020-02-04 | 2021-08-12 | 中国人民解放军军事科学院军事医学研究院 | 含五元杂环的苯磺酰胺类化合物及其制备方法和用途 |
| CN111233786B (zh) * | 2020-02-04 | 2021-11-26 | 中国人民解放军军事科学院军事医学研究院 | 含五元杂环的苯磺酰胺类化合物及其制备方法和用途 |
Also Published As
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| WO2004014352A3 (en) | 2004-09-10 |
| BR0313282A (pt) | 2005-10-18 |
| PL374994A1 (en) | 2005-11-14 |
| WO2004014430A1 (en) | 2004-02-19 |
| KR20050056189A (ko) | 2005-06-14 |
| BR0313299A (pt) | 2005-06-14 |
| US20040198781A1 (en) | 2004-10-07 |
| MXPA05001497A (es) | 2005-05-27 |
| WO2004014352A2 (en) | 2004-02-19 |
| IL166685A0 (en) | 2006-01-15 |
| AU2003225571A1 (en) | 2004-02-25 |
| AU2003213062A1 (en) | 2004-02-25 |
| EP1526895A2 (en) | 2005-05-04 |
| US20030100594A1 (en) | 2003-05-29 |
| MXPA05001496A (es) | 2005-05-16 |
| CA2495516A1 (en) | 2004-02-19 |
| JP2005539023A (ja) | 2005-12-22 |
| JP2005539022A (ja) | 2005-12-22 |
| CA2495502A1 (en) | 2004-02-19 |
| EP1526869A1 (en) | 2005-05-04 |
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