CN1339972A - 在口腔中迅速崩解的片剂 - Google Patents
在口腔中迅速崩解的片剂 Download PDFInfo
- Publication number
- CN1339972A CN1339972A CN00803628A CN00803628A CN1339972A CN 1339972 A CN1339972 A CN 1339972A CN 00803628 A CN00803628 A CN 00803628A CN 00803628 A CN00803628 A CN 00803628A CN 1339972 A CN1339972 A CN 1339972A
- Authority
- CN
- China
- Prior art keywords
- tablet
- starch
- water soluble
- soluble excipient
- mannitol
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Inorganic Chemistry (AREA)
- Zoology (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Medicinal Preparation (AREA)
- Cosmetics (AREA)
Abstract
Description
实施例1 | 实施例2 | 实施例5 | 实施例6 | 实施例8 | 对比实施例1 | 对比实施例2 | |
硬度(kg) | 4 | 3 | 4 | 5 | 3 | 3 | 2 |
崩解时间(秒) | 19 | 27 | 15 | 35 | 30 | 411 | 80 |
口中崩解时间(秒) | 20 | 21 | 17 | 33 | 14 | >240 | 100 |
感官可接受性 | ○ | ○ | ○ | ○ | ○ | X | X |
Claims (8)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP3542999 | 1999-02-15 | ||
JP35429/1999 | 1999-02-15 | ||
JP35429/99 | 1999-02-15 |
Publications (2)
Publication Number | Publication Date |
---|---|
CN1339972A true CN1339972A (zh) | 2002-03-13 |
CN1186098C CN1186098C (zh) | 2005-01-26 |
Family
ID=12441629
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CNB008036284A Expired - Fee Related CN1186098C (zh) | 1999-02-15 | 2000-02-14 | 在口腔中迅速崩解的片剂 |
Country Status (11)
Country | Link |
---|---|
EP (1) | EP1153616B1 (zh) |
JP (1) | JP4435424B2 (zh) |
KR (2) | KR20010102122A (zh) |
CN (1) | CN1186098C (zh) |
AT (1) | ATE283708T1 (zh) |
AU (1) | AU2462200A (zh) |
CA (1) | CA2360102C (zh) |
DE (1) | DE60016381T2 (zh) |
ES (1) | ES2233329T3 (zh) |
TW (1) | TWI271198B (zh) |
WO (1) | WO2000047233A1 (zh) |
Cited By (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102413819A (zh) * | 2009-04-30 | 2012-04-11 | 罗盖特公司 | 甘露醇和颗粒淀粉的可压制的并且自由流动的共凝聚体 |
CN1915233B (zh) * | 2006-08-30 | 2012-10-03 | 四川科瑞德制药有限公司 | 一种治疗焦虑症的药物组合物及其口崩制剂 |
CN101983055B (zh) * | 2008-01-31 | 2013-05-08 | 杏林制药株式会社 | 以咪达那新为有效成分的口腔内速崩片的制造方法 |
CN102119034B (zh) * | 2008-06-13 | 2013-05-22 | 大日本住友制药株式会社 | 在口腔中快速崩解的片剂和制备其的方法 |
CN102065843B (zh) * | 2008-07-04 | 2015-01-21 | 罗盖特公司 | 口腔可分散的甘露醇 |
Families Citing this family (31)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7550156B2 (en) * | 2001-11-23 | 2009-06-23 | Rohm And Haas Company | Optimised pellet formulations |
GB0210397D0 (en) | 2002-05-07 | 2002-06-12 | Ferring Bv | Pharmaceutical formulations |
JP5584509B2 (ja) * | 2003-02-28 | 2014-09-03 | 東和薬品株式会社 | 口腔内崩壊錠剤 |
JP4551627B2 (ja) * | 2003-02-28 | 2010-09-29 | 東和薬品株式会社 | 口腔内崩壊錠剤の製造方法 |
EP1530967B1 (en) | 2003-11-13 | 2006-05-03 | Ferring B.V. | Blister pack and solid dosage form comprising desmopressin |
TWI335227B (en) | 2004-02-25 | 2011-01-01 | Medical & Pharm Ind Tech & Dev | Pharmaceutical composition of taste masking and rapidly dissolving drug and method of preparing the same |
JP2006176496A (ja) * | 2004-11-24 | 2006-07-06 | Freunt Ind Co Ltd | 固形剤およびその製造方法 |
WO2006085497A1 (ja) * | 2005-02-09 | 2006-08-17 | Kissei Pharmaceutical Co., Ltd. | 口腔内崩壊錠 |
JP2006282551A (ja) * | 2005-03-31 | 2006-10-19 | Taiyo Yakuhin Kogyo Kk | 口腔内崩壊錠およびその製造方法 |
JP5219508B2 (ja) * | 2005-05-18 | 2013-06-26 | 大日本住友製薬株式会社 | ドロキシドパを含有する安定な錠剤 |
JP4439499B2 (ja) * | 2005-08-01 | 2010-03-24 | 大日本住友製薬株式会社 | アムロジピン含有粒子およびそれからなる口腔内崩壊錠 |
JP5241681B2 (ja) * | 2005-08-01 | 2013-07-17 | 大日本住友製薬株式会社 | アムロジピン含有粒子およびそれからなる口腔内崩壊錠 |
MX2009002563A (es) | 2006-09-14 | 2009-03-20 | Astellas Pharma Inc | Tableta de desintegracion oral y proceso para la produccion de la misma. |
CA2680536A1 (en) | 2007-03-13 | 2008-10-09 | Dainippon Sumitomo Pharma Co., Ltd. | Oral disintegrating tablet |
JP5291324B2 (ja) * | 2007-11-01 | 2013-09-18 | 沢井製薬株式会社 | 口腔内崩壊錠 |
JP5352474B2 (ja) | 2007-12-28 | 2013-11-27 | 沢井製薬株式会社 | 口腔内崩壊錠およびその製造方法 |
EP2246052B1 (en) * | 2008-01-31 | 2017-03-08 | Kyorin Pharmaceutical Co., Ltd. | Orally rapidly disintegrating tablet comprising imidafenacin |
US11963995B2 (en) | 2008-05-21 | 2024-04-23 | Ferring B.V. | Methods comprising desmopressin |
US20100286045A1 (en) | 2008-05-21 | 2010-11-11 | Bjarke Mirner Klein | Methods comprising desmopressin |
PT2296686E (pt) | 2008-05-21 | 2014-05-23 | Ferring Bv | Desmopressina orodispersível para aumentar o período inicial de sono não perturbado por noctúria |
JP4954961B2 (ja) * | 2008-10-06 | 2012-06-20 | 大日本住友製薬株式会社 | 光安定性の向上した組成物 |
JP5713544B2 (ja) * | 2009-07-30 | 2015-05-07 | 杏林製薬株式会社 | イミダフェナシン含有口腔内速崩錠 |
JP2012051810A (ja) * | 2010-08-31 | 2012-03-15 | Zensei Yakuhin Kogyo Kk | 口腔内崩壊錠およびその製造法 |
US8426461B2 (en) | 2011-01-17 | 2013-04-23 | Takeda Pharmaceutical Company Limited | Orally dispersible tablet |
CN103429223A (zh) | 2011-01-17 | 2013-12-04 | 武田药品工业株式会社 | 口腔分散片 |
JP5689052B2 (ja) * | 2011-12-26 | 2015-03-25 | 大日本住友製薬株式会社 | 光安定性の向上した組成物 |
CN103445090B (zh) * | 2013-04-27 | 2015-08-19 | 华中农业大学 | 一种富含γ-氨基丁酸米制品的生产方法及产品 |
JP2016033144A (ja) * | 2015-11-20 | 2016-03-10 | 大日本住友製薬株式会社 | 光安定性の向上した組成物 |
JP2017057224A (ja) * | 2016-12-27 | 2017-03-23 | 大日本住友製薬株式会社 | 光安定性の向上した組成物 |
JP2018044015A (ja) * | 2017-12-25 | 2018-03-22 | 大日本住友製薬株式会社 | 光安定性の向上した組成物 |
WO2024088560A1 (en) * | 2022-10-28 | 2024-05-02 | Roquette Freres | Compound for formulating moisture sensitive active ingredients |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ZA726026B (en) * | 1971-12-23 | 1973-05-30 | D Woodcraft | Anti-smoking preparation |
DE2347713C3 (de) * | 1972-09-25 | 1980-03-06 | Warner-Lambert Co., Morris Plains, N.J. (V.St.A.) | Acetylsalicylsäurekautablette |
JPH0739350B2 (ja) * | 1990-08-03 | 1995-05-01 | ゼリア新薬工業株式会社 | 生薬配合チュアブル錠 |
JP3069458B2 (ja) * | 1992-01-29 | 2000-07-24 | 武田薬品工業株式会社 | 口腔内崩壊型錠剤およびその製造法 |
JP3067125B2 (ja) * | 1994-11-22 | 2000-07-17 | 田辺製薬株式会社 | 易服用性の有核錠型製剤 |
JPH08208523A (ja) * | 1995-02-03 | 1996-08-13 | Gun Ei Chem Ind Co Ltd | 製剤素材 |
JP3119801B2 (ja) * | 1995-09-28 | 2000-12-25 | 武田薬品工業株式会社 | ビタミン含有組成物の安定化方法 |
JPH10298062A (ja) * | 1997-04-24 | 1998-11-10 | Pfizer Pharmaceut Co Ltd | 口腔内速溶型錠剤 |
TW527195B (en) * | 1997-10-09 | 2003-04-11 | Ssp Co Ltd | Fast-soluble solid pharmaceutical combinations |
-
2000
- 2000-02-14 WO PCT/JP2000/000806 patent/WO2000047233A1/ja active IP Right Grant
- 2000-02-14 KR KR1020017010290A patent/KR20010102122A/ko not_active Application Discontinuation
- 2000-02-14 DE DE60016381T patent/DE60016381T2/de not_active Revoked
- 2000-02-14 CA CA002360102A patent/CA2360102C/en not_active Expired - Fee Related
- 2000-02-14 CN CNB008036284A patent/CN1186098C/zh not_active Expired - Fee Related
- 2000-02-14 TW TW089102428A patent/TWI271198B/zh not_active IP Right Cessation
- 2000-02-14 KR KR1020097026434A patent/KR20100008007A/ko active IP Right Grant
- 2000-02-14 AU AU24622/00A patent/AU2462200A/en not_active Abandoned
- 2000-02-14 JP JP2000598184A patent/JP4435424B2/ja not_active Expired - Lifetime
- 2000-02-14 EP EP00902958A patent/EP1153616B1/en not_active Revoked
- 2000-02-14 ES ES00902958T patent/ES2233329T3/es not_active Expired - Lifetime
- 2000-02-14 AT AT00902958T patent/ATE283708T1/de not_active IP Right Cessation
Cited By (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1915233B (zh) * | 2006-08-30 | 2012-10-03 | 四川科瑞德制药有限公司 | 一种治疗焦虑症的药物组合物及其口崩制剂 |
CN101983055B (zh) * | 2008-01-31 | 2013-05-08 | 杏林制药株式会社 | 以咪达那新为有效成分的口腔内速崩片的制造方法 |
CN102119034B (zh) * | 2008-06-13 | 2013-05-22 | 大日本住友制药株式会社 | 在口腔中快速崩解的片剂和制备其的方法 |
CN102065843B (zh) * | 2008-07-04 | 2015-01-21 | 罗盖特公司 | 口腔可分散的甘露醇 |
CN104382868B (zh) * | 2008-07-04 | 2018-12-07 | 罗盖特公司 | 口腔可分散的甘露醇 |
CN102413819A (zh) * | 2009-04-30 | 2012-04-11 | 罗盖特公司 | 甘露醇和颗粒淀粉的可压制的并且自由流动的共凝聚体 |
Also Published As
Publication number | Publication date |
---|---|
TWI271198B (en) | 2007-01-21 |
ES2233329T3 (es) | 2005-06-16 |
CN1186098C (zh) | 2005-01-26 |
EP1153616B1 (en) | 2004-12-01 |
DE60016381D1 (de) | 2005-01-05 |
CA2360102A1 (en) | 2000-08-17 |
AU2462200A (en) | 2000-08-29 |
KR20100008007A (ko) | 2010-01-22 |
EP1153616A1 (en) | 2001-11-14 |
JP4435424B2 (ja) | 2010-03-17 |
EP1153616A4 (en) | 2003-04-02 |
WO2000047233A1 (fr) | 2000-08-17 |
DE60016381T2 (de) | 2005-12-15 |
CA2360102C (en) | 2009-05-19 |
KR20010102122A (ko) | 2001-11-15 |
ATE283708T1 (de) | 2004-12-15 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
C06 | Publication | ||
PB01 | Publication | ||
C10 | Entry into substantive examination | ||
SE01 | Entry into force of request for substantive examination | ||
C14 | Grant of patent or utility model | ||
GR01 | Patent grant | ||
C56 | Change in the name or address of the patentee |
Owner name: DAINIPPON PHARMACEUTICAL CO., LTD. Free format text: FORMER NAME OR ADDRESS: SUMITOMO PHARMACEUTICALS CO., LTD. Owner name: NIPPO SUMITOMO PHARMACEUTICALS CO., LTD. Free format text: FORMER NAME OR ADDRESS: DAINIPPON PHARMACEUTICAL CO., LTD. |
|
CP03 | Change of name, title or address |
Address after: Osaka Japan Patentee after: Dainippon Sumitomo Pharma Co.,Ltd. Address before: Osaka Japan Patentee before: DAINIPPON PHARMACEUTICAL Co.,Ltd. Address after: Osaka Japan Patentee after: DAINIPPON PHARMACEUTICAL Co.,Ltd. Address before: Osaka Japan Patentee before: SUMITOMO PHARMACEUTICALS CO.,LTD. |
|
C17 | Cessation of patent right | ||
CF01 | Termination of patent right due to non-payment of annual fee |
Granted publication date: 20050126 Termination date: 20130214 |