CN114026079A - 一种sglt2/dpp4抑制剂及其应用 - Google Patents
一种sglt2/dpp4抑制剂及其应用 Download PDFInfo
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- CN114026079A CN114026079A CN202080047668.5A CN202080047668A CN114026079A CN 114026079 A CN114026079 A CN 114026079A CN 202080047668 A CN202080047668 A CN 202080047668A CN 114026079 A CN114026079 A CN 114026079A
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Abstract
作为SGLT2/DPP4双抑制剂的一类化合物,以及在制备作为SGLT2/DPP4双抑制剂的药物中的应用。具体涉及式(Ⅰ)所示化合物、其异构体或其药学上可接受的盐。
Description
PCT国内申请,说明书已公开。
Claims (9)
- PCT国内申请,权利要求书已公开。
Applications Claiming Priority (7)
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CN201910683099 | 2019-07-26 | ||
CN2019106830992 | 2019-07-26 | ||
CN202010119914 | 2020-02-26 | ||
CN2020101199145 | 2020-02-26 | ||
CN2020105722264 | 2020-06-22 | ||
CN202010572226 | 2020-06-22 | ||
PCT/CN2020/104521 WO2021018044A1 (zh) | 2019-07-26 | 2020-07-24 | 一种sglt2/dpp4抑制剂及其应用 |
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KR (1) | KR102471055B1 (zh) |
CN (1) | CN114026079B (zh) |
AU (1) | AU2020320890B2 (zh) |
CA (1) | CA3145678C (zh) |
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WO2022160737A1 (zh) * | 2021-01-26 | 2022-08-04 | 东宝紫星(杭州)生物医药有限公司 | 四氢吡喃环类化合物的晶型及其制备方法 |
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TWI499414B (zh) | 2006-09-29 | 2015-09-11 | Lexicon Pharmaceuticals Inc | 鈉與葡萄糖第2型共同運輸體(co-transporter 2)的抑制物與其應用方法 |
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2020
- 2020-07-24 MX MX2022001044A patent/MX2022001044A/es unknown
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- 2020-07-24 JP JP2022505531A patent/JP7227427B2/ja active Active
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- 2020-07-24 WO PCT/CN2020/104521 patent/WO2021018044A1/zh unknown
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- 2020-07-24 US US17/629,527 patent/US20220242898A1/en active Pending
- 2020-07-24 CN CN202080047668.5A patent/CN114026079B/zh active Active
- 2020-07-24 AU AU2020320890A patent/AU2020320890B2/en active Active
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CN101343296A (zh) * | 2007-07-10 | 2009-01-14 | 莱西肯医药有限公司 | 钠-葡萄糖协同转运蛋白2的抑制剂及其用法 |
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US20220242898A1 (en) | 2022-08-04 |
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EP4006017A1 (en) | 2022-06-01 |
KR20220031735A (ko) | 2022-03-11 |
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