CN106061971B - 吡咯烷基砜衍生物及其作为RORγ调节剂的用途 - Google Patents

吡咯烷基砜衍生物及其作为RORγ调节剂的用途 Download PDF

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CN106061971B
CN106061971B CN201580011338.XA CN201580011338A CN106061971B CN 106061971 B CN106061971 B CN 106061971B CN 201580011338 A CN201580011338 A CN 201580011338A CN 106061971 B CN106061971 B CN 106061971B
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substituted
alkyl
base
phenyl
hydrogen
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CN106061971A (zh
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段敬武
T.G.M.达
江斌
陆忠辉
肖海云
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Bristol Myers Squibb Co
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CN201580011338.XA 2014-01-06 2015-01-05 吡咯烷基砜衍生物及其作为RORγ调节剂的用途 Expired - Fee Related CN106061971B (zh)

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US201461923896P 2014-01-06 2014-01-06
US61/923896 2014-01-06
PCT/US2015/010089 WO2015103509A1 (en) 2014-01-06 2015-01-05 Pyrrolidinyl sulfone derivatives and their use as ror gamma modulators

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WO2015035278A1 (en) 2013-09-09 2015-03-12 Bristol-Myers Squibb Company RORγ MODULATORS
US9725443B2 (en) 2013-09-20 2017-08-08 Bristol-Myers Squibb Company RORγ modulators
CN106132931B (zh) 2014-01-06 2019-08-02 百时美施贵宝公司 碳环砜RORγ调节剂
US9637455B2 (en) 2014-01-06 2017-05-02 Bristol-Myers Squibb Company Heterocyclic sulfone RORγ modulators
EP3092215B1 (en) 2014-01-06 2018-10-17 Bristol-Myers Squibb Company Cyclohexyl sulfone ror gamma modulators
ES2708025T3 (es) 2014-10-30 2019-04-08 Janssen Pharmaceutica Nv Tiazoles como moduladores de RORyt
JOP20200117A1 (ar) 2014-10-30 2017-06-16 Janssen Pharmaceutica Nv كحولات ثلاثي فلوروميثيل كمُعدلات للمستقبل النووي جاما تي المرتبط بحمض الريتيونَويك ROR?t
ES2767303T3 (es) 2014-10-30 2020-06-17 Janssen Pharmaceutica Nv Tiazoles sustituidos por amida como moduladores de Rorgamma T
WO2016179460A1 (en) 2015-05-07 2016-11-10 Bristol-Myers Squibb Company Tricyclic sulfones as rorϒ modulators
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