CN103827112A - 作为杀真菌剂的哌啶吡唑 - Google Patents

作为杀真菌剂的哌啶吡唑 Download PDF

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Publication number
CN103827112A
CN103827112A CN201280044843.0A CN201280044843A CN103827112A CN 103827112 A CN103827112 A CN 103827112A CN 201280044843 A CN201280044843 A CN 201280044843A CN 103827112 A CN103827112 A CN 103827112A
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CN
China
Prior art keywords
alkyl
cycloalkyl
carbonyl
group
haloalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CN201280044843.0A
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English (en)
Chinese (zh)
Inventor
S.希勒布兰
土屋知己
S.霍夫曼
P.克里斯托
P.瓦斯奈雷
T.赛茨
J.本廷
U.瓦亨多夫-诺伊曼
J.P.施密特
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer Pharma AG
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Bayer Pharma AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Pharma AG filed Critical Bayer Pharma AG
Publication of CN103827112A publication Critical patent/CN103827112A/zh
Pending legal-status Critical Current

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Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/78—1,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
CN201280044843.0A 2011-09-15 2012-09-11 作为杀真菌剂的哌啶吡唑 Pending CN103827112A (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP11181383.8 2011-09-15
EP11181383 2011-09-15
PCT/EP2012/067728 WO2013037768A1 (de) 2011-09-15 2012-09-11 Piperidinpyrazole als fungizide

Publications (1)

Publication Number Publication Date
CN103827112A true CN103827112A (zh) 2014-05-28

Family

ID=46826533

Family Applications (1)

Application Number Title Priority Date Filing Date
CN201280044843.0A Pending CN103827112A (zh) 2011-09-15 2012-09-11 作为杀真菌剂的哌啶吡唑

Country Status (12)

Country Link
US (1) US10004232B2 (enExample)
EP (1) EP2755971B1 (enExample)
JP (1) JP5959646B2 (enExample)
CN (1) CN103827112A (enExample)
BR (1) BR112014005989B1 (enExample)
CO (1) CO6890107A2 (enExample)
ES (1) ES2661849T3 (enExample)
HK (1) HK1198385A1 (enExample)
IN (1) IN2014CN01862A (enExample)
MX (1) MX355824B (enExample)
TW (1) TWI612045B (enExample)
WO (1) WO2013037768A1 (enExample)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN106687459A (zh) * 2014-08-13 2017-05-17 Sds生物技术株式会社 稠合 11 元环化合物及含有它们的农园艺用杀菌剂
CN108601353A (zh) * 2016-02-08 2018-09-28 Sds生物技术株式会社 杀菌性组合物
WO2020034992A1 (zh) * 2018-08-14 2020-02-20 华中师范大学 含稠杂环结构的化合物及其制备方法和应用以及杀菌剤
CN111848612A (zh) * 2019-07-31 2020-10-30 华中师范大学 含稠杂环结构的化合物及其制备方法和应用以及杀菌剂

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EP2921491B1 (de) * 2011-12-27 2017-08-16 Bayer Intellectual Property GmbH Zwischenverbindungen zur herstellung von heteroarylpiperidinen und -piperazinderivaten als fungizide
AU2013216354B2 (en) 2012-02-02 2017-08-31 Idorsia Pharmaceuticals Ltd 4-(benzoimidazol-2-yl)-thiazole compounds and related aza derivatives
TWI632142B (zh) 2013-06-24 2018-08-11 德商拜耳作物科學股份有限公司 作為殺真菌劑之六氫吡啶羧酸衍生物
CN105658649B (zh) 2013-07-22 2019-03-22 爱杜西亚药品有限公司 1-(哌嗪-1-基)-2-([1,2,4]三唑-1-基)-乙酮衍生物
WO2015028457A1 (en) 2013-08-28 2015-03-05 Bayer Cropscience Ag Malonic ester derivatives of heteroarylpiperidines and -piperazines as fungicides
TWI647215B (zh) 2013-11-11 2019-01-11 德商拜耳作物科學股份有限公司 自α,α－二鹵胺製備３,５－雙鹵烷基吡唑衍生物之方法
ES2681286T3 (es) 2014-03-24 2018-09-12 Bayer Cropscience Aktiengesellschaft Derivados de fenilpiperidincarboxamida como fungicidas
AR099789A1 (es) 2014-03-24 2016-08-17 Actelion Pharmaceuticals Ltd Derivados de 8-(piperazin-1-il)-1,2,3,4-tetrahidro-isoquinolina
AR103399A1 (es) 2015-01-15 2017-05-10 Actelion Pharmaceuticals Ltd Derivados de (r)-2-metil-piperazina como moduladores del receptor cxcr3
MY187614A (en) 2015-01-15 2021-10-04 Idorsia Pharmaceuticals Ltd Hydroxyalkyl-piperazine derivatives as cxcr3 receptor modulators
WO2016202761A1 (en) 2015-06-17 2016-12-22 Bayer Cropscience Aktiengesellschaft Active compound combinations
CN108602765B (zh) 2016-02-08 2022-05-03 高文有限公司 1,2-苯二甲醇化合物的制造方法
TW201838974A (zh) 2017-04-19 2018-11-01 印度商Ｐｉ工業公司 具殺菌性質之雜環化合物
WO2019048989A1 (en) 2017-09-08 2019-03-14 Pi Industries Ltd. NOVEL FUNGICIDE HETEROCYCLIC COMPOUNDS
WO2019048988A1 (en) 2017-09-08 2019-03-14 Pi Industries Ltd. Novel fungidal heterocyclic compounds
TW202236965A (zh) 2020-12-15 2022-10-01 印度商皮埃企業有限公司 包含哌啶噻唑化合物之新穎農業化學組成物
UY39763A (es) 2021-05-15 2022-11-30 Pi Industries Ltd Composición agroquímica novedosa que comprende compuestos de piperidin-tiazol

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Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN106687459A (zh) * 2014-08-13 2017-05-17 Sds生物技术株式会社 稠合 11 元环化合物及含有它们的农园艺用杀菌剂
CN106687459B (zh) * 2014-08-13 2019-07-30 Sds生物技术株式会社 稠合11元环化合物及含有它们的农园艺用杀菌剂
CN108601353A (zh) * 2016-02-08 2018-09-28 Sds生物技术株式会社 杀菌性组合物
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CN108601353B (zh) * 2016-02-08 2024-04-05 高文作物保护公司 杀菌性组合物
WO2020034992A1 (zh) * 2018-08-14 2020-02-20 华中师范大学 含稠杂环结构的化合物及其制备方法和应用以及杀菌剤
CN111848612A (zh) * 2019-07-31 2020-10-30 华中师范大学 含稠杂环结构的化合物及其制备方法和应用以及杀菌剂
CN111848612B (zh) * 2019-07-31 2021-09-14 华中师范大学 含稠杂环结构的化合物及其制备方法和应用以及杀菌剂

Also Published As

Publication number Publication date
TWI612045B (zh) 2018-01-21
JP2014527076A (ja) 2014-10-09
JP5959646B2 (ja) 2016-08-02
ES2661849T3 (es) 2018-04-04
IN2014CN01862A (enExample) 2015-05-29
US20140228404A1 (en) 2014-08-14
EP2755971B1 (de) 2017-12-20
CO6890107A2 (es) 2014-03-10
BR112014005989A2 (pt) 2017-06-13
EP2755971A1 (de) 2014-07-23
BR112014005989B1 (pt) 2019-11-05
WO2013037768A1 (de) 2013-03-21
HK1198385A1 (en) 2015-04-17
MX2014001864A (es) 2014-05-30
TW201326165A (zh) 2013-07-01
US10004232B2 (en) 2018-06-26
MX355824B (es) 2018-05-02

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