CN102811619B - 激酶抑制剂 - Google Patents

激酶抑制剂 Download PDF

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Publication number
CN102811619B
CN102811619B CN201080051548.9A CN201080051548A CN102811619B CN 102811619 B CN102811619 B CN 102811619B CN 201080051548 A CN201080051548 A CN 201080051548A CN 102811619 B CN102811619 B CN 102811619B
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methyl
disease
compound
heteroatoms
cancer
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CN102811619A (zh
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李宰圭
宋浩俊
高钟声
李熙圭
金泳三
金洪宇
张纯花
林顺熙
崔章植
金正皓
金世源
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Oscotec Inc
Genosco
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Oscotec Inc
Genosco
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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CN201080051548.9A 2009-11-13 2010-11-12 激酶抑制剂 Active CN102811619B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US26110009P 2009-11-13 2009-11-13
US61/261,100 2009-11-13
PCT/US2010/056583 WO2011060295A1 (en) 2009-11-13 2010-11-12 Kinase inhibitors

Publications (2)

Publication Number Publication Date
CN102811619A CN102811619A (zh) 2012-12-05
CN102811619B true CN102811619B (zh) 2015-04-22

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US (1) US8629132B2 (enExample)
EP (1) EP2498607B1 (enExample)
JP (1) JP5740409B2 (enExample)
KR (1) KR101663637B1 (enExample)
CN (1) CN102811619B (enExample)
BR (1) BR112012011287B1 (enExample)
CA (1) CA2780892C (enExample)
CL (1) CL2012001221A1 (enExample)
EA (1) EA024729B1 (enExample)
IL (1) IL219726A (enExample)
MX (1) MX2012005332A (enExample)
MY (1) MY160820A (enExample)
NZ (1) NZ599041A (enExample)
SG (1) SG10201407453TA (enExample)
WO (1) WO2011060295A1 (enExample)
ZA (1) ZA201204246B (enExample)

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