CN102036967B - 作为5-ht6拮抗剂的芳基磺酰基吡唑啉甲脒衍生物 - Google Patents

作为5-ht6拮抗剂的芳基磺酰基吡唑啉甲脒衍生物 Download PDF

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CN102036967B
CN102036967B CN200980108113.0A CN200980108113A CN102036967B CN 102036967 B CN102036967 B CN 102036967B CN 200980108113 A CN200980108113 A CN 200980108113A CN 102036967 B CN102036967 B CN 102036967B
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compound
mixture
dihydro
dcm
ethylamino
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Expired - Fee Related
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CN102036967A (zh
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A·梵洛维金
W·I·伊维玛巴克
A·斯托伊特
A·A·M·仁辛克
J·雯霍斯特
M·A·W·范德纽特
M·德汉
C·G·克鲁斯
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Abbott Healthcare Products BV
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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  • Health & Medical Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Psychology (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Nutrition Science (AREA)
  • Emergency Medicine (AREA)
  • Anesthesiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
CN200980108113.0A 2008-03-18 2009-03-17 作为5-ht6拮抗剂的芳基磺酰基吡唑啉甲脒衍生物 Expired - Fee Related CN102036967B (zh)

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Application Number Priority Date Filing Date Title
EP08152873 2008-03-18
EP08152873.9 2008-03-18
PCT/EP2009/053133 WO2009115515A1 (en) 2008-03-18 2009-03-17 Arylsulfonyl pyrazoline carboxamidine derivatives as 5-ht6 antagonists

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CN102036967A CN102036967A (zh) 2011-04-27
CN102036967B true CN102036967B (zh) 2014-10-15

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CN201410233817.3A Pending CN104003937A (zh) 2008-03-18 2009-03-17 作为5-ht6拮抗剂的芳基磺酰基吡唑啉甲脒衍生物

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AR079935A1 (es) * 2010-01-29 2012-02-29 Abbott Healthcare Products Bv Sintesis de derivados de pirazolin carboxamidina sustituida
AU2012296639B2 (en) * 2011-08-15 2016-06-09 University Of Utah Research Foundation Substituted (E)-N'-(1-phenylethylidene) benzohydrazide analogs as histone demethylase inhibitors
CN104903296A (zh) 2012-11-16 2015-09-09 百时美施贵宝公司 二氢吡唑gpr40调节剂
AR104762A1 (es) 2012-11-16 2017-08-16 Bristol Myers Squibb Co Moduladores de dihidropirazol gpr40
UY35143A (es) * 2012-11-16 2014-05-30 Bristol Myers Squibb Co Derivados de dihidropirazol como moduladores del receptor acoplado a la proteína gpr40 g
WO2015172059A1 (en) * 2014-05-09 2015-11-12 The United States Of America, As Represented By The Secretary, Department Of Health & Human Services Pyrazole derivatives and their use as cannabinoid receptor mediators
CA2957566C (en) 2014-08-12 2023-08-01 Daniel Paul Becker Indoline sulfonamide inhibitors of dape and ndm-1 and use of the same
EP3109237A1 (en) * 2015-06-22 2016-12-28 AnaMar AB Novel 5-ht2 antagonists
CN107460160A (zh) * 2017-08-23 2017-12-12 世贸天阶制药（江苏）有限责任公司 一种cho细胞无血清培养基
US10879709B2 (en) 2018-05-31 2020-12-29 National Taipei University Of Technology Power management system and operating method thereof
CN117567338A (zh) 2019-10-09 2024-02-20 拜耳公司 作为农药的新的杂芳基三唑化合物
CA3185968A1 (en) 2020-07-13 2022-01-20 Tony Lahoutte Antibody fragment against folr1
WO2023203135A1 (en) 2022-04-22 2023-10-26 Precirix N.V. Improved radiolabelled antibody
AU2023264245A1 (en) 2022-05-02 2024-12-19 Precirix N.V. Pre-targeting

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