TWI557110B - 作為5-ht6拮抗劑的芳基磺醯基吡唑啉羧脒衍生物 - Google Patents

作為5-ht6拮抗劑的芳基磺醯基吡唑啉羧脒衍生物 Download PDF

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TWI557110B
TWI557110B TW098108412A TW98108412A TWI557110B TW I557110 B TWI557110 B TW I557110B TW 098108412 A TW098108412 A TW 098108412A TW 98108412 A TW98108412 A TW 98108412A TW I557110 B TWI557110 B TW I557110B
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compound
alkyl
group
mixture
dihydro
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TW098108412A
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TW200942519A (en
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阿諾德 凡羅維真
屋特I 伊威馬霸克
艾克索 史托特
阿加達A M 倫辛克
珍妮佛 凡赫斯特
馬汀那A W 凡迪那特
馬汀 迪漢
克林斯G 克勞斯
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艾伯維巴哈馬有限公司
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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  • Health & Medical Sciences (AREA)
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  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Psychology (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Nutrition Science (AREA)
  • Emergency Medicine (AREA)
  • Anesthesiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
TW098108412A 2008-03-18 2009-03-16 作為5-ht6拮抗劑的芳基磺醯基吡唑啉羧脒衍生物 TWI557110B (zh)

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EP08152873 2008-03-18

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TWI557110B true TWI557110B (zh) 2016-11-11

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US (3) US8563723B2 (enExample)
EP (2) EP2265589B1 (enExample)
JP (1) JP5504252B2 (enExample)
KR (1) KR101623357B1 (enExample)
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PL (2) PL2265589T3 (enExample)
PT (1) PT2610247T (enExample)
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AR079935A1 (es) * 2010-01-29 2012-02-29 Abbott Healthcare Products Bv Sintesis de derivados de pirazolin carboxamidina sustituida
AU2012296639B2 (en) * 2011-08-15 2016-06-09 University Of Utah Research Foundation Substituted (E)-N'-(1-phenylethylidene) benzohydrazide analogs as histone demethylase inhibitors
CN104903296A (zh) 2012-11-16 2015-09-09 百时美施贵宝公司 二氢吡唑gpr40调节剂
AR104762A1 (es) 2012-11-16 2017-08-16 Bristol Myers Squibb Co Moduladores de dihidropirazol gpr40
UY35143A (es) * 2012-11-16 2014-05-30 Bristol Myers Squibb Co Derivados de dihidropirazol como moduladores del receptor acoplado a la proteína gpr40 g
WO2015172059A1 (en) * 2014-05-09 2015-11-12 The United States Of America, As Represented By The Secretary, Department Of Health & Human Services Pyrazole derivatives and their use as cannabinoid receptor mediators
CA2957566C (en) 2014-08-12 2023-08-01 Daniel Paul Becker Indoline sulfonamide inhibitors of dape and ndm-1 and use of the same
EP3109237A1 (en) * 2015-06-22 2016-12-28 AnaMar AB Novel 5-ht2 antagonists
CN107460160A (zh) * 2017-08-23 2017-12-12 世贸天阶制药(江苏)有限责任公司 一种cho细胞无血清培养基
CN117567338A (zh) 2019-10-09 2024-02-20 拜耳公司 作为农药的新的杂芳基三唑化合物
CA3185968A1 (en) 2020-07-13 2022-01-20 Tony Lahoutte Antibody fragment against folr1
WO2023203135A1 (en) 2022-04-22 2023-10-26 Precirix N.V. Improved radiolabelled antibody
AU2023264245A1 (en) 2022-05-02 2024-12-19 Precirix N.V. Pre-targeting

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