CN101855228B - 作为gsk-3抑制剂的氰基氨基喹诺酮和四唑并氨基喹诺酮 - Google Patents
作为gsk-3抑制剂的氰基氨基喹诺酮和四唑并氨基喹诺酮 Download PDFInfo
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- CN101855228B CN101855228B CN2008801155430A CN200880115543A CN101855228B CN 101855228 B CN101855228 B CN 101855228B CN 2008801155430 A CN2008801155430 A CN 2008801155430A CN 200880115543 A CN200880115543 A CN 200880115543A CN 101855228 B CN101855228 B CN 101855228B
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Abstract
Description
Claims (6)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
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US99334607P | 2007-09-11 | 2007-09-11 | |
US60/993,346 | 2007-09-11 | ||
PCT/US2008/010615 WO2009035634A2 (en) | 2007-09-11 | 2008-09-11 | Cyanoaminoquinolones and tetrazoloaminoquinolones as gsk-3 inhibitors |
Related Child Applications (1)
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CN201110205276.XA Division CN102351880B (zh) | 2007-09-11 | 2008-09-11 | 作为gsk-3 抑制剂的氰基氨基喹诺酮和四唑并氨基喹诺酮 |
Publications (2)
Publication Number | Publication Date |
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CN101855228A CN101855228A (zh) | 2010-10-06 |
CN101855228B true CN101855228B (zh) | 2012-10-24 |
Family
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CN2008801155430A Expired - Fee Related CN101855228B (zh) | 2007-09-11 | 2008-09-11 | 作为gsk-3抑制剂的氰基氨基喹诺酮和四唑并氨基喹诺酮 |
CN201110205276.XA Expired - Fee Related CN102351880B (zh) | 2007-09-11 | 2008-09-11 | 作为gsk-3 抑制剂的氰基氨基喹诺酮和四唑并氨基喹诺酮 |
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CN201110205276.XA Expired - Fee Related CN102351880B (zh) | 2007-09-11 | 2008-09-11 | 作为gsk-3 抑制剂的氰基氨基喹诺酮和四唑并氨基喹诺酮 |
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US (1) | US8389514B2 (zh) |
EP (1) | EP2203458B1 (zh) |
JP (1) | JP5426552B2 (zh) |
KR (1) | KR101563018B1 (zh) |
CN (2) | CN101855228B (zh) |
AT (1) | ATE531721T1 (zh) |
AU (1) | AU2008299903B2 (zh) |
BR (1) | BRPI0816798A2 (zh) |
CA (1) | CA2699151A1 (zh) |
ES (1) | ES2371800T3 (zh) |
HK (1) | HK1162502A1 (zh) |
MX (1) | MX2010002667A (zh) |
WO (1) | WO2009035634A2 (zh) |
Families Citing this family (11)
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WO2010088924A1 (en) | 2009-02-06 | 2010-08-12 | Telormedix Sa | Pharmaceutical compositions comprising imidazoquinolin(amines) and derivatives thereof suitable for local administration |
EP2406266B1 (en) * | 2009-03-11 | 2013-12-25 | Kyorin Pharmaceutical Co., Ltd. | 7-cycloalkylaminoquinolones as gsk-3 inhibitors |
WO2011107494A1 (de) | 2010-03-03 | 2011-09-09 | Sanofi | Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung |
US8530413B2 (en) | 2010-06-21 | 2013-09-10 | Sanofi | Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments |
TW201215387A (en) | 2010-07-05 | 2012-04-16 | Sanofi Aventis | Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament |
TW201221505A (en) | 2010-07-05 | 2012-06-01 | Sanofi Sa | Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament |
TW201215388A (en) | 2010-07-05 | 2012-04-16 | Sanofi Sa | (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments |
WO2013037390A1 (en) | 2011-09-12 | 2013-03-21 | Sanofi | 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
WO2013045413A1 (en) | 2011-09-27 | 2013-04-04 | Sanofi | 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
WO2015155738A2 (en) | 2014-04-09 | 2015-10-15 | Christopher Rudd | Use of gsk-3 inhibitors or activators which modulate pd-1 or t-bet expression to modulate t cell immunity |
US20220133740A1 (en) | 2019-02-08 | 2022-05-05 | Frequency Therapeutics, Inc. | Valproic acid compounds and wnt agonists for treating ear disorders |
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WO2002092571A1 (en) * | 2001-05-11 | 2002-11-21 | Astrazeneca Ab | Novel 4-anilinoquinoline-3-carboxamides |
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- 2008-09-11 CA CA2699151A patent/CA2699151A1/en not_active Abandoned
- 2008-09-11 JP JP2010524862A patent/JP5426552B2/ja not_active Expired - Fee Related
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- 2008-09-11 KR KR1020107007735A patent/KR101563018B1/ko active IP Right Grant
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- 2008-09-11 ES ES08830095T patent/ES2371800T3/es active Active
- 2008-09-11 WO PCT/US2008/010615 patent/WO2009035634A2/en active Application Filing
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- 2008-09-11 US US12/677,789 patent/US8389514B2/en not_active Expired - Fee Related
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- 2008-09-11 CN CN201110205276.XA patent/CN102351880B/zh not_active Expired - Fee Related
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Also Published As
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CA2699151A1 (en) | 2009-03-19 |
EP2203458B1 (en) | 2011-11-02 |
AU2008299903A1 (en) | 2009-03-19 |
MX2010002667A (es) | 2010-04-01 |
KR20100063114A (ko) | 2010-06-10 |
EP2203458A2 (en) | 2010-07-07 |
JP5426552B2 (ja) | 2014-02-26 |
WO2009035634A3 (en) | 2009-06-04 |
BRPI0816798A2 (pt) | 2016-10-11 |
US8389514B2 (en) | 2013-03-05 |
CN101855228A (zh) | 2010-10-06 |
CN102351880A (zh) | 2012-02-15 |
JP2010539164A (ja) | 2010-12-16 |
AU2008299903B2 (en) | 2013-08-29 |
ES2371800T3 (es) | 2012-01-10 |
WO2009035634A2 (en) | 2009-03-19 |
HK1162502A1 (zh) | 2012-08-31 |
CN102351880B (zh) | 2014-11-12 |
ATE531721T1 (de) | 2011-11-15 |
KR101563018B1 (ko) | 2015-10-23 |
US20110172219A1 (en) | 2011-07-14 |
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