CN101495113A - Il-8受体拮抗剂 - Google Patents
Il-8受体拮抗剂 Download PDFInfo
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- CN101495113A CN101495113A CNA2007800232115A CN200780023211A CN101495113A CN 101495113 A CN101495113 A CN 101495113A CN A2007800232115 A CNA2007800232115 A CN A2007800232115A CN 200780023211 A CN200780023211 A CN 200780023211A CN 101495113 A CN101495113 A CN 101495113A
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- chloro
- phenyl
- urea
- sulfonyl
- diazabicylo
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Classifications
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-
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Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
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| US79383606P | 2006-04-21 | 2006-04-21 | |
| US60/793,836 | 2006-04-21 |
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| CN101495113A true CN101495113A (zh) | 2009-07-29 |
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| CNA2007800232115A Pending CN101495113A (zh) | 2006-04-21 | 2007-04-20 | Il-8受体拮抗剂 |
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| Country | Link |
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| EP (1) | EP2010180A4 (enExample) |
| JP (1) | JP2009534420A (enExample) |
| CN (1) | CN101495113A (enExample) |
| AU (1) | AU2007240364A1 (enExample) |
| BR (1) | BRPI0710559A2 (enExample) |
| CA (1) | CA2650007A1 (enExample) |
| IL (1) | IL194700A0 (enExample) |
| MX (1) | MX2008013599A (enExample) |
| RU (1) | RU2008145871A (enExample) |
| WO (1) | WO2007124423A2 (enExample) |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2019137484A1 (zh) * | 2018-01-11 | 2019-07-18 | 南京明德新药研发股份有限公司 | Cxcr2拮抗剂 |
| WO2021004531A1 (zh) * | 2019-07-11 | 2021-01-14 | 南京明德新药研发有限公司 | 一种cxcr2拮抗剂的晶型及其应用 |
| CN114702503A (zh) * | 2016-05-26 | 2022-07-05 | 拜耳医药股份有限公司 | 甲酮化合物 |
Families Citing this family (12)
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| EP2009992B1 (en) | 2006-04-21 | 2012-06-27 | GlaxoSmithKline LLC | Il-8 receptor antagonists |
| MX2008013599A (es) | 2006-04-21 | 2008-10-31 | Smithkline Beechman Corp | Antagonistas del receptor il-8. |
| TW201035102A (en) * | 2009-03-04 | 2010-10-01 | Gruenethal Gmbh | Sulfonylated tetrahydroazolopyrazines and their use as medicinal products |
| JO3156B1 (ar) | 2009-07-09 | 2017-09-20 | Novartis Ag | ايميدازولات مدمجة والتركيبات التي تشملها لعلاج الأمراض الطفيلية على مثال الملاريا |
| CN102781448B (zh) * | 2010-03-01 | 2015-01-21 | 诺瓦药品公司 | 用于治疗病毒性疾病的组合物和方法 |
| US8648070B2 (en) * | 2010-12-17 | 2014-02-11 | Boehringer Ingelheim International Gmbh | Bicyclic ring system substituted sulfonamide functionalised phenols as medicaments |
| US8648118B2 (en) * | 2010-12-17 | 2014-02-11 | Boehringer Ingelheim International Gmbh | Bicyclic ring system substituted amide functionalised phenols as medicaments |
| US9241930B2 (en) | 2011-08-24 | 2016-01-26 | Novadrug, Llc | Compositions and methods for treating viral diseases |
| KR20150002713A (ko) | 2012-03-28 | 2015-01-07 | 뉴로포레 테라피스, 인코포레이티드 | 단백질 응집 저해제로서의 페닐-우레아 및 페닐-카바메이트 유도체 |
| EA036824B1 (ru) * | 2016-07-11 | 2020-12-24 | Байер Фарма Акциенгезельшафт | [8-(фенилсульфонил)-3,8-диазабицикло[3.2.1]окт-3-ил](1н-1,2,3-триазол-4-ил)метаноны |
| AU2018235937A1 (en) * | 2017-03-15 | 2019-09-19 | Lunella Biotech, Inc. | Mitoriboscins: mitochondrial-based therapeutics targeting cancer cells, bacteria, and pathogenic yeast |
| EP3615030A1 (en) | 2017-04-24 | 2020-03-04 | Novartis AG | Therapeutic regimen of 2-amino-l-(2-(4-fluorophenyl)-3-(4-fluorophenylamino)-8,8-dimethyl-5,6-dihydroimidazo[1,2-a]pyrazin-7(8h)-yl)ethanone and combinations thereof |
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- 2007-04-20 US US12/297,917 patent/US8097626B2/en not_active Expired - Fee Related
- 2007-04-20 AU AU2007240364A patent/AU2007240364A1/en not_active Abandoned
- 2007-04-20 CN CNA2007800232115A patent/CN101495113A/zh active Pending
- 2007-04-20 CA CA002650007A patent/CA2650007A1/en not_active Abandoned
- 2007-04-20 WO PCT/US2007/067088 patent/WO2007124423A2/en not_active Ceased
- 2007-04-20 EP EP07761016A patent/EP2010180A4/en not_active Withdrawn
- 2007-04-20 BR BRPI0710559-2A patent/BRPI0710559A2/pt not_active IP Right Cessation
- 2007-04-20 RU RU2008145871/04A patent/RU2008145871A/ru not_active Application Discontinuation
- 2007-04-20 JP JP2009506793A patent/JP2009534420A/ja active Pending
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- 2008-10-12 IL IL194700A patent/IL194700A0/en unknown
Cited By (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN114702503A (zh) * | 2016-05-26 | 2022-07-05 | 拜耳医药股份有限公司 | 甲酮化合物 |
| CN114702503B (zh) * | 2016-05-26 | 2023-12-22 | 拜耳医药股份有限公司 | 甲酮化合物 |
| WO2019137484A1 (zh) * | 2018-01-11 | 2019-07-18 | 南京明德新药研发股份有限公司 | Cxcr2拮抗剂 |
| US11136315B2 (en) | 2018-01-11 | 2021-10-05 | Medshine Discovery Inc. | CXCR2 antagonist |
| WO2021004531A1 (zh) * | 2019-07-11 | 2021-01-14 | 南京明德新药研发有限公司 | 一种cxcr2拮抗剂的晶型及其应用 |
Also Published As
| Publication number | Publication date |
|---|---|
| JP2009534420A (ja) | 2009-09-24 |
| US8097626B2 (en) | 2012-01-17 |
| IL194700A0 (en) | 2009-08-03 |
| AU2007240364A1 (en) | 2007-11-01 |
| BRPI0710559A2 (pt) | 2011-08-16 |
| EP2010180A4 (en) | 2010-10-13 |
| WO2007124423A2 (en) | 2007-11-01 |
| RU2008145871A (ru) | 2010-05-27 |
| US20090298810A1 (en) | 2009-12-03 |
| MX2008013599A (es) | 2008-10-31 |
| WO2007124423A3 (en) | 2009-04-09 |
| CA2650007A1 (en) | 2007-11-01 |
| EP2010180A2 (en) | 2009-01-07 |
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