CN101405259B - 具有含卤氨基甲酸酯基和酰基的乙二胺衍生物的制备方法及它们的制备中间体 - Google Patents
具有含卤氨基甲酸酯基和酰基的乙二胺衍生物的制备方法及它们的制备中间体 Download PDFInfo
- Publication number
- CN101405259B CN101405259B CN2007800096002A CN200780009600A CN101405259B CN 101405259 B CN101405259 B CN 101405259B CN 2007800096002 A CN2007800096002 A CN 2007800096002A CN 200780009600 A CN200780009600 A CN 200780009600A CN 101405259 B CN101405259 B CN 101405259B
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- 0 CC(*)(CN)N(*)C(O*)=O Chemical compound CC(*)(CN)N(*)C(O*)=O 0.000 description 3
- FORGMRSGVSYZQR-YFKPBYRVSA-N CC(C)C[C@@H](C(N)=O)N Chemical compound CC(C)C[C@@H](C(N)=O)N FORGMRSGVSYZQR-YFKPBYRVSA-N 0.000 description 1
- YRAZPXKZQDCPGM-LURJTMIESA-N CC(C)C[C@@H](C(N)=O)NC(OCC(F)(F)F)=O Chemical compound CC(C)C[C@@H](C(N)=O)NC(OCC(F)(F)F)=O YRAZPXKZQDCPGM-LURJTMIESA-N 0.000 description 1
- JZPKHQXHWQVDLM-SSDOTTSWSA-N CC(C)[C@@H](CN)N(C)C=O Chemical compound CC(C)[C@@H](CN)N(C)C=O JZPKHQXHWQVDLM-SSDOTTSWSA-N 0.000 description 1
- OGBFVYCMSNRCLA-ZCFIWIBFSA-N CC(C)[C@@H](CN)NC(OCC(F)(F)F)=O Chemical compound CC(C)[C@@H](CN)NC(OCC(F)(F)F)=O OGBFVYCMSNRCLA-ZCFIWIBFSA-N 0.000 description 1
- WXHUIGDMKJHLQC-GFCCVEGCSA-N CC(C)[C@@H](CNC(c1cc2ccccc2[o]1)=O)NC(OCC(F)(F)F)=O Chemical compound CC(C)[C@@H](CNC(c1cc2ccccc2[o]1)=O)NC(OCC(F)(F)F)=O WXHUIGDMKJHLQC-GFCCVEGCSA-N 0.000 description 1
- PWVIASPWMOAULL-CYBMUJFWSA-N CC(C)[C@@H](CNC(c1ccc(C(F)(F)F)cc1)=O)N(C)C(OCC(F)(F)F)=O Chemical compound CC(C)[C@@H](CNC(c1ccc(C(F)(F)F)cc1)=O)N(C)C(OCC(F)(F)F)=O PWVIASPWMOAULL-CYBMUJFWSA-N 0.000 description 1
- ANGRCXGCASUEOA-LURJTMIESA-N N#C[C@H](CCC1)N1C(OCC(F)(F)F)=O Chemical compound N#C[C@H](CCC1)N1C(OCC(F)(F)F)=O ANGRCXGCASUEOA-LURJTMIESA-N 0.000 description 1
- PWDVWOLFBLJMPW-DSEUIKHZSA-N NC([C@H](CCC1)N1C(O)OCC(F)(F)F)=O Chemical compound NC([C@H](CCC1)N1C(O)OCC(F)(F)F)=O PWDVWOLFBLJMPW-DSEUIKHZSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B53/00—Asymmetric syntheses
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C269/04—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups from amines with formation of carbamate groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C269/06—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups by reactions not involving the formation of carbamate groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C271/06—Esters of carbamic acids
- C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
- C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C271/20—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by nitrogen atoms not being part of nitro or nitroso groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C271/06—Esters of carbamic acids
- C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
- C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C271/22—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
- C07D207/09—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/82—Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D307/84—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D307/85—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pyrrole Compounds (AREA)
- Furan Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP090705/2006 | 2006-03-29 | ||
| JP2006090705 | 2006-03-29 | ||
| PCT/JP2007/000307 WO2007111024A1 (ja) | 2006-03-29 | 2007-03-27 | 含ハロゲンカルバマート基とアシル基を有するエチレンジアミン誘導体の製造方法、及びそれらの製造中間体 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN101405259A CN101405259A (zh) | 2009-04-08 |
| CN101405259B true CN101405259B (zh) | 2013-06-19 |
Family
ID=38540959
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN2007800096002A Active CN101405259B (zh) | 2006-03-29 | 2007-03-27 | 具有含卤氨基甲酸酯基和酰基的乙二胺衍生物的制备方法及它们的制备中间体 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US20090281352A1 (enExample) |
| EP (1) | EP2008997A4 (enExample) |
| JP (2) | JP4801728B2 (enExample) |
| KR (1) | KR101040876B1 (enExample) |
| CN (1) | CN101405259B (enExample) |
| AU (1) | AU2007230511A1 (enExample) |
| CA (1) | CA2647590C (enExample) |
| IN (1) | IN2015DN00763A (enExample) |
| MX (1) | MX2008012388A (enExample) |
| RU (1) | RU2404963C2 (enExample) |
| TW (1) | TWI338680B (enExample) |
| WO (1) | WO2007111024A1 (enExample) |
| ZA (1) | ZA200808332B (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MY159705A (en) | 2009-12-22 | 2017-01-13 | Mitsui Chemicals Agro Inc | Plant disease control composition and method for controlling plant disease by applying the same |
| KR101492351B1 (ko) * | 2010-09-22 | 2015-02-10 | 미쓰이가가쿠 아그로 가부시키가이샤 | 함불소 카바메이트기를 가지는 아미노산 아미드 유도체의 제조방법, 그 제조 중간체, 및 에틸렌디아민 유도체의 제조방법 |
| KR20250116837A (ko) | 2024-01-25 | 2025-08-04 | 주식회사 엘지화학 | 신규 라이신 디카르복실라아제를 포함하여 펜타메틸렌디아민을 생산하는 재조합 미생물 및 이를 이용한 펜타메틸렌디아민 생산방법 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8414986D0 (en) * | 1984-06-12 | 1984-07-18 | Beecham Group Plc | Chemical process |
| EP0167011A3 (en) * | 1984-06-12 | 1986-03-19 | Beecham Group Plc | Beta-lactam compounds, intermediates thereof, their use in preparing beta-lactams having a diketopiperazine group |
| JP4596098B2 (ja) | 2000-07-26 | 2010-12-08 | 三菱瓦斯化学株式会社 | 光学活性α−アミノ酸の製造方法 |
| KR100863849B1 (ko) * | 2003-10-31 | 2008-10-15 | 미쓰이 가가쿠 가부시키가이샤 | 디아민 유도체, 그 제조방법 및 그것을 유효 성분으로 하는식물 병해 방제제 |
| JP4533210B2 (ja) * | 2005-03-31 | 2010-09-01 | 三井化学アグロ株式会社 | ジアミン誘導体、その製造方法およびそれらを有効成分とする植物病害防除剤 |
-
2007
- 2007-03-27 MX MX2008012388A patent/MX2008012388A/es not_active Application Discontinuation
- 2007-03-27 RU RU2008142736/04A patent/RU2404963C2/ru not_active IP Right Cessation
- 2007-03-27 JP JP2008507376A patent/JP4801728B2/ja active Active
- 2007-03-27 KR KR1020087025709A patent/KR101040876B1/ko active Active
- 2007-03-27 CA CA2647590A patent/CA2647590C/en not_active Expired - Fee Related
- 2007-03-27 CN CN2007800096002A patent/CN101405259B/zh active Active
- 2007-03-27 ZA ZA200808332A patent/ZA200808332B/xx unknown
- 2007-03-27 AU AU2007230511A patent/AU2007230511A1/en not_active Abandoned
- 2007-03-27 WO PCT/JP2007/000307 patent/WO2007111024A1/ja not_active Ceased
- 2007-03-27 US US12/295,167 patent/US20090281352A1/en not_active Abandoned
- 2007-03-27 EP EP07736964A patent/EP2008997A4/en not_active Withdrawn
- 2007-03-27 IN IN763DEN2015 patent/IN2015DN00763A/en unknown
- 2007-03-29 TW TW096110968A patent/TWI338680B/zh active
-
2011
- 2011-06-27 JP JP2011141517A patent/JP5417384B2/ja active Active
Non-Patent Citations (2)
| Title |
|---|
| John A.W. Kruijtzer et al..Approaches to the Synthesis of Ureapeptoid Peptidomimetics.《Tetrahedron Letters》.1997,第38卷(第30期),5335-5338. * |
| Michael North et al..SYNTHETIC STUDIES TOWARDS CYCLIC PEPTIDES.CONCISE SYNTHESIS OF THIAZOLINE AND THIAZOLE CONTAINING AMINO ACIDS.《Tetrahedron》.1990,第46卷(第24期),8267-829. * |
Also Published As
| Publication number | Publication date |
|---|---|
| RU2404963C2 (ru) | 2010-11-27 |
| JP5417384B2 (ja) | 2014-02-12 |
| US20090281352A1 (en) | 2009-11-12 |
| JPWO2007111024A1 (ja) | 2009-08-06 |
| RU2008142736A (ru) | 2010-05-10 |
| JP4801728B2 (ja) | 2011-10-26 |
| ZA200808332B (en) | 2010-02-24 |
| TW200740730A (en) | 2007-11-01 |
| JP2011184464A (ja) | 2011-09-22 |
| WO2007111024A1 (ja) | 2007-10-04 |
| CA2647590C (en) | 2010-11-30 |
| AU2007230511A1 (en) | 2007-10-04 |
| KR101040876B1 (ko) | 2011-06-16 |
| TWI338680B (en) | 2011-03-11 |
| CA2647590A1 (en) | 2007-10-04 |
| KR20090018781A (ko) | 2009-02-23 |
| IN2015DN00763A (enExample) | 2015-07-10 |
| EP2008997A1 (en) | 2008-12-31 |
| MX2008012388A (es) | 2008-10-10 |
| CN101405259A (zh) | 2009-04-08 |
| EP2008997A4 (en) | 2010-11-24 |
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| C14 | Grant of patent or utility model | ||
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