JP4801728B2 - 含ハロゲンカルバマート基とアシル基を有するエチレンジアミン誘導体の製造方法 - Google Patents

含ハロゲンカルバマート基とアシル基を有するエチレンジアミン誘導体の製造方法 Download PDF

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JP4801728B2
JP4801728B2 JP2008507376A JP2008507376A JP4801728B2 JP 4801728 B2 JP4801728 B2 JP 4801728B2 JP 2008507376 A JP2008507376 A JP 2008507376A JP 2008507376 A JP2008507376 A JP 2008507376A JP 4801728 B2 JP4801728 B2 JP 4801728B2
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carbon atoms
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JPWO2007111024A1 (ja
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豪毅 梅谷
河野  敏之
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MC Crop & Life Manufacturing
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Mitsui Chemicals Agro Inc
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B53/00—Asymmetric syntheses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C269/04—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups from amines with formation of carbamate groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C269/06—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups by reactions not involving the formation of carbamate groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06—Esters of carbamic acids
    • C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/20—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by nitrogen atoms not being part of nitro or nitroso groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06—Esters of carbamic acids
    • C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/22—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • C07D207/09—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/82—Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D307/84—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D307/85—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pyrrole Compounds (AREA)
  • Furan Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP2008507376A 2006-03-29 2007-03-27 含ハロゲンカルバマート基とアシル基を有するエチレンジアミン誘導体の製造方法 Active JP4801728B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2008507376A JP4801728B2 (ja) 2006-03-29 2007-03-27 含ハロゲンカルバマート基とアシル基を有するエチレンジアミン誘導体の製造方法

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP2006090705 2006-03-29
JP2006090705 2006-03-29
JP2008507376A JP4801728B2 (ja) 2006-03-29 2007-03-27 含ハロゲンカルバマート基とアシル基を有するエチレンジアミン誘導体の製造方法
PCT/JP2007/000307 WO2007111024A1 (ja) 2006-03-29 2007-03-27 含ハロゲンカルバマート基とアシル基を有するエチレンジアミン誘導体の製造方法、及びそれらの製造中間体

Related Child Applications (1)

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JP2011141517A Division JP5417384B2 (ja) 2006-03-29 2011-06-27 含ハロゲンカルバマート基とアシル基を有するエチレンジアミン誘導体の製造方法、及びそれらの製造中間体

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JPWO2007111024A1 JPWO2007111024A1 (ja) 2009-08-06
JP4801728B2 true JP4801728B2 (ja) 2011-10-26

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JP2011141517A Active JP5417384B2 (ja) 2006-03-29 2011-06-27 含ハロゲンカルバマート基とアシル基を有するエチレンジアミン誘導体の製造方法、及びそれらの製造中間体

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Country Link
US (1) US20090281352A1 (enExample)
EP (1) EP2008997A4 (enExample)
JP (2) JP4801728B2 (enExample)
KR (1) KR101040876B1 (enExample)
CN (1) CN101405259B (enExample)
AU (1) AU2007230511A1 (enExample)
CA (1) CA2647590C (enExample)
IN (1) IN2015DN00763A (enExample)
MX (1) MX2008012388A (enExample)
RU (1) RU2404963C2 (enExample)
TW (1) TWI338680B (enExample)
WO (1) WO2007111024A1 (enExample)
ZA (1) ZA200808332B (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY159705A (en) 2009-12-22 2017-01-13 Mitsui Chemicals Agro Inc Plant disease control composition and method for controlling plant disease by applying the same
KR101492351B1 (ko) * 2010-09-22 2015-02-10 미쓰이가가쿠 아그로 가부시키가이샤 함불소 카바메이트기를 가지는 아미노산 아미드 유도체의 제조방법, 그 제조 중간체, 및 에틸렌디아민 유도체의 제조방법
KR20250116837A (ko) 2024-01-25 2025-08-04 주식회사 엘지화학 신규 라이신 디카르복실라아제를 포함하여 펜타메틸렌디아민을 생산하는 재조합 미생물 및 이를 이용한 펜타메틸렌디아민 생산방법

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6117548A (ja) * 1984-06-12 1986-01-25 ビーチヤム・グループ・ピーエルシー β‐ラクタム化合物及びその製法
WO2005042474A1 (ja) * 2003-10-31 2005-05-12 Mitsui Chemicals, Inc. ジアミン誘導体、その製造方法およびそれらを有効成分とする植物病害防除剤

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0167011A3 (en) * 1984-06-12 1986-03-19 Beecham Group Plc Beta-lactam compounds, intermediates thereof, their use in preparing beta-lactams having a diketopiperazine group
JP4596098B2 (ja) 2000-07-26 2010-12-08 三菱瓦斯化学株式会社 光学活性α−アミノ酸の製造方法
JP4533210B2 (ja) * 2005-03-31 2010-09-01 三井化学アグロ株式会社 ジアミン誘導体、その製造方法およびそれらを有効成分とする植物病害防除剤

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6117548A (ja) * 1984-06-12 1986-01-25 ビーチヤム・グループ・ピーエルシー β‐ラクタム化合物及びその製法
WO2005042474A1 (ja) * 2003-10-31 2005-05-12 Mitsui Chemicals, Inc. ジアミン誘導体、その製造方法およびそれらを有効成分とする植物病害防除剤

Also Published As

Publication number Publication date
RU2404963C2 (ru) 2010-11-27
JP5417384B2 (ja) 2014-02-12
CN101405259B (zh) 2013-06-19
US20090281352A1 (en) 2009-11-12
JPWO2007111024A1 (ja) 2009-08-06
RU2008142736A (ru) 2010-05-10
ZA200808332B (en) 2010-02-24
TW200740730A (en) 2007-11-01
JP2011184464A (ja) 2011-09-22
WO2007111024A1 (ja) 2007-10-04
CA2647590C (en) 2010-11-30
AU2007230511A1 (en) 2007-10-04
KR101040876B1 (ko) 2011-06-16
TWI338680B (en) 2011-03-11
CA2647590A1 (en) 2007-10-04
KR20090018781A (ko) 2009-02-23
IN2015DN00763A (enExample) 2015-07-10
EP2008997A1 (en) 2008-12-31
MX2008012388A (es) 2008-10-10
CN101405259A (zh) 2009-04-08
EP2008997A4 (en) 2010-11-24

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