CN100516035C - 制备2-二苯基甲基亚硫酰基乙酸甲酯的方法 - Google Patents

制备2-二苯基甲基亚硫酰基乙酸甲酯的方法 Download PDF

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Publication number
CN100516035C
CN100516035C CNB2004800021479A CN200480002147A CN100516035C CN 100516035 C CN100516035 C CN 100516035C CN B2004800021479 A CNB2004800021479 A CN B2004800021479A CN 200480002147 A CN200480002147 A CN 200480002147A CN 100516035 C CN100516035 C CN 100516035C
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CN
China
Prior art keywords
methyl
diphenyl
acid
solvent
acetate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
CNB2004800021479A
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English (en)
Chinese (zh)
Other versions
CN1735591A (zh
Inventor
S·罗斯
D·克雷恩
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Saifulun European Co
Teva Sante SAS
Original Assignee
Cephalon France SAS
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Publication date
Application filed by Cephalon France SAS filed Critical Cephalon France SAS
Publication of CN1735591A publication Critical patent/CN1735591A/zh
Application granted granted Critical
Publication of CN100516035C publication Critical patent/CN100516035C/zh
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C315/00—Preparation of sulfones; Preparation of sulfoxides
    • C07C315/02—Preparation of sulfones; Preparation of sulfoxides by formation of sulfone or sulfoxide groups by oxidation of sulfides, or by formation of sulfone groups by oxidation of sulfoxides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/14—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
CNB2004800021479A 2003-01-13 2004-01-08 制备2-二苯基甲基亚硫酰基乙酸甲酯的方法 Expired - Fee Related CN100516035C (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP20030290082 EP1437345A1 (en) 2003-01-13 2003-01-13 Novel method for preparing methyl 2-diphenylmethylsulfinylacetate
EP03290082.1 2003-01-13

Publications (2)

Publication Number Publication Date
CN1735591A CN1735591A (zh) 2006-02-15
CN100516035C true CN100516035C (zh) 2009-07-22

Family

ID=32479973

Family Applications (1)

Application Number Title Priority Date Filing Date
CNB2004800021479A Expired - Fee Related CN100516035C (zh) 2003-01-13 2004-01-08 制备2-二苯基甲基亚硫酰基乙酸甲酯的方法

Country Status (20)

Country Link
US (1) US7211684B2 (enExample)
EP (2) EP1437345A1 (enExample)
JP (1) JP4690304B2 (enExample)
KR (1) KR101062281B1 (enExample)
CN (1) CN100516035C (enExample)
AR (1) AR042842A1 (enExample)
AU (1) AU2004203975B2 (enExample)
BR (1) BRPI0406489A (enExample)
CA (1) CA2512084C (enExample)
EA (1) EA010381B1 (enExample)
IL (1) IL169517A (enExample)
IS (1) IS7958A (enExample)
MX (1) MXPA05007419A (enExample)
NO (1) NO331507B1 (enExample)
NZ (1) NZ541089A (enExample)
PL (1) PL212412B1 (enExample)
TW (1) TWI323250B (enExample)
UA (1) UA80598C2 (enExample)
WO (1) WO2004063149A1 (enExample)
ZA (1) ZA200505381B (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1437345A1 (en) 2003-01-13 2004-07-14 Organisation de Synthese Mondiale Orsymonde Novel method for preparing methyl 2-diphenylmethylsulfinylacetate
EP1516869A1 (en) 2003-09-19 2005-03-23 Cephalon France Process for enantioselective synthesis of single enantiomers of modafinil by asymmetric oxidation
US7368591B2 (en) 2003-09-19 2008-05-06 Cephalon France Process for enantioselective synthesis of single enantiomers of modafinil by asymmetric oxidation
CN100393699C (zh) * 2005-03-10 2008-06-11 浙江工业大学 2-（二苯基甲基亚硫酰基）乙酰胺的合成方法
EP1702915A1 (en) 2005-03-14 2006-09-20 Cephalon France Process for enantioselective synthesis of single enantiomers of thio-substituted arylmethanesulfinyl derivatives by asymmetric oxidation
WO2007103221A2 (en) * 2006-03-01 2007-09-13 Teva Pharmaceutical Industries Ltd. An improved process for the preparation of armodafinil
CN104059004A (zh) * 2014-06-25 2014-09-24 江苏斯威森生物医药工程研究中心有限公司 一种2-[(4,4’-二卤-二苯基甲基)巯基]乙酸酯的制备方法

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4964893A (en) * 1986-04-17 1990-10-23 Monsanto Company Benzhydryl compounds as herbicide antidotes
US5571825A (en) * 1995-03-31 1996-11-05 Warner-Lambert Company Method of selectively inhibiting prostaglandin G/H synthase-2

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE198165C (enExample)
GB1520812A (en) * 1975-10-02 1978-08-09 Lafon Labor Benzhydrylsulphinyl derivatives
GB1584462A (en) * 1977-03-31 1981-02-11 Lafon Labor N-diaryl-malonamide and diarylmethyl-sulphinyl-acetamide derivatives and pharmaceutical compositions containing them
DE2812542A1 (de) 1978-03-22 1979-10-04 Thomae Gmbh Dr K Neue schwefelhaltige fluorenyl-und phenanthryl-derivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
FR2528038B2 (fr) * 1982-06-04 1985-08-09 Lafon Labor Derives de benzhydrylsulfinylacetamide et leur utilisation en therapeutique
FR2528041A1 (fr) * 1982-06-04 1983-12-09 Lafon Labor Acides halogenobenzhydrylsulfinylacetohydroxamiques, procede de preparation et utilisation en therapeutique
JP3233806B2 (ja) * 1995-01-23 2001-12-04 ユーシービージャパン株式会社 スルフェニル酢酸誘導体の製造法
EP1437345A1 (en) 2003-01-13 2004-07-14 Organisation de Synthese Mondiale Orsymonde Novel method for preparing methyl 2-diphenylmethylsulfinylacetate

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4964893A (en) * 1986-04-17 1990-10-23 Monsanto Company Benzhydryl compounds as herbicide antidotes
US5571825A (en) * 1995-03-31 1996-11-05 Warner-Lambert Company Method of selectively inhibiting prostaglandin G/H synthase-2

Also Published As

Publication number Publication date
ZA200505381B (enExample) 2006-04-26
CA2512084A1 (en) 2004-07-29
CA2512084C (en) 2012-03-20
IL169517A (en) 2012-06-28
JP4690304B2 (ja) 2011-06-01
KR20050091085A (ko) 2005-09-14
EP1583739A1 (en) 2005-10-12
US20060235237A1 (en) 2006-10-19
NZ541089A (en) 2008-05-30
PL377822A1 (pl) 2006-02-20
AU2004203975A1 (en) 2004-07-29
MXPA05007419A (es) 2005-09-12
CN1735591A (zh) 2006-02-15
AU2004203975B2 (en) 2010-07-01
EP1437345A1 (en) 2004-07-14
BRPI0406489A (pt) 2005-12-06
AR042842A1 (es) 2005-07-06
NO20053602L (no) 2005-07-22
PL212412B1 (pl) 2012-09-28
JP2006516560A (ja) 2006-07-06
NO331507B1 (no) 2012-01-16
US7211684B2 (en) 2007-05-01
IS7958A (is) 2005-07-26
WO2004063149A1 (en) 2004-07-29
TWI323250B (en) 2010-04-11
UA80598C2 (en) 2007-10-10
TW200420530A (en) 2004-10-16
EA200501125A1 (ru) 2005-12-29
KR101062281B1 (ko) 2011-09-06
EA010381B1 (ru) 2008-08-29

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Legal Events

Date Code Title Description
C06 Publication
PB01 Publication
C10 Entry into substantive examination
SE01 Entry into force of request for substantive examination
C14 Grant of patent or utility model
GR01 Patent grant
ASS Succession or assignment of patent right

Owner name: TEVA SANTE S. A. S.

Free format text: FORMER OWNER: CEPHALON EUROPE CORP.

Effective date: 20150804

Owner name: CEPHALON EUROPE CORP.

Free format text: FORMER OWNER: CEPHALON FRANCE

Effective date: 20150804

C41 Transfer of patent application or patent right or utility model
TR01 Transfer of patent right

Effective date of registration: 20150804

Address after: Paris France

Patentee after: Teva Sant Co.

Address before: French Maisons Alfort

Patentee before: Saifulun European Co.

Effective date of registration: 20150804

Address after: French Maisons Alfort

Patentee after: Saifulun European Co.

Address before: French Maisons Alfort

Patentee before: Cephalon France

CF01 Termination of patent right due to non-payment of annual fee
CF01 Termination of patent right due to non-payment of annual fee

Granted publication date: 20090722

Termination date: 20180108