AU2004203975B2 - Method for preparing methyl 2-diphenylmethylsulfinylacetate - Google Patents

Method for preparing methyl 2-diphenylmethylsulfinylacetate Download PDF

Info

Publication number
AU2004203975B2
AU2004203975B2 AU2004203975A AU2004203975A AU2004203975B2 AU 2004203975 B2 AU2004203975 B2 AU 2004203975B2 AU 2004203975 A AU2004203975 A AU 2004203975A AU 2004203975 A AU2004203975 A AU 2004203975A AU 2004203975 B2 AU2004203975 B2 AU 2004203975B2
Authority
AU
Australia
Prior art keywords
acid
methyl
solvent
benzhydrol
diphenylmethylsulfinylacetate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU2004203975A
Other languages
English (en)
Other versions
AU2004203975A1 (en
Inventor
Dominique Klein
Sebastien Rose
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Teva Sante SAS
Original Assignee
Teva Sante SAS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teva Sante SAS filed Critical Teva Sante SAS
Publication of AU2004203975A1 publication Critical patent/AU2004203975A1/en
Assigned to CEPHALON FRANCE reassignment CEPHALON FRANCE Request for Assignment Assignors: ORGANISATION DE SYNTHESE MONDIALE ORSYMONDE
Application granted granted Critical
Publication of AU2004203975B2 publication Critical patent/AU2004203975B2/en
Assigned to TEVA SANTE reassignment TEVA SANTE Request to Amend Deed and Register Assignors: CEPHALON FRANCE
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C315/00—Preparation of sulfones; Preparation of sulfoxides
    • C07C315/02—Preparation of sulfones; Preparation of sulfoxides by formation of sulfone or sulfoxide groups by oxidation of sulfides, or by formation of sulfone groups by oxidation of sulfoxides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/14—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AU2004203975A 2003-01-13 2004-01-08 Method for preparing methyl 2-diphenylmethylsulfinylacetate Ceased AU2004203975B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP20030290082 EP1437345A1 (en) 2003-01-13 2003-01-13 Novel method for preparing methyl 2-diphenylmethylsulfinylacetate
EP03290082.1 2003-01-13
PCT/IB2004/000002 WO2004063149A1 (en) 2003-01-13 2004-01-08 Method for preparing methyl 2-diphenylmethylsulfinylacetate

Publications (2)

Publication Number Publication Date
AU2004203975A1 AU2004203975A1 (en) 2004-07-29
AU2004203975B2 true AU2004203975B2 (en) 2010-07-01

Family

ID=32479973

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2004203975A Ceased AU2004203975B2 (en) 2003-01-13 2004-01-08 Method for preparing methyl 2-diphenylmethylsulfinylacetate

Country Status (20)

Country Link
US (1) US7211684B2 (enExample)
EP (2) EP1437345A1 (enExample)
JP (1) JP4690304B2 (enExample)
KR (1) KR101062281B1 (enExample)
CN (1) CN100516035C (enExample)
AR (1) AR042842A1 (enExample)
AU (1) AU2004203975B2 (enExample)
BR (1) BRPI0406489A (enExample)
CA (1) CA2512084C (enExample)
EA (1) EA010381B1 (enExample)
IL (1) IL169517A (enExample)
IS (1) IS7958A (enExample)
MX (1) MXPA05007419A (enExample)
NO (1) NO331507B1 (enExample)
NZ (1) NZ541089A (enExample)
PL (1) PL212412B1 (enExample)
TW (1) TWI323250B (enExample)
UA (1) UA80598C2 (enExample)
WO (1) WO2004063149A1 (enExample)
ZA (1) ZA200505381B (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1437345A1 (en) 2003-01-13 2004-07-14 Organisation de Synthese Mondiale Orsymonde Novel method for preparing methyl 2-diphenylmethylsulfinylacetate
EP1516869A1 (en) 2003-09-19 2005-03-23 Cephalon France Process for enantioselective synthesis of single enantiomers of modafinil by asymmetric oxidation
US7368591B2 (en) 2003-09-19 2008-05-06 Cephalon France Process for enantioselective synthesis of single enantiomers of modafinil by asymmetric oxidation
CN100393699C (zh) * 2005-03-10 2008-06-11 浙江工业大学 2-（二苯基甲基亚硫酰基）乙酰胺的合成方法
EP1702915A1 (en) 2005-03-14 2006-09-20 Cephalon France Process for enantioselective synthesis of single enantiomers of thio-substituted arylmethanesulfinyl derivatives by asymmetric oxidation
WO2007103221A2 (en) * 2006-03-01 2007-09-13 Teva Pharmaceutical Industries Ltd. An improved process for the preparation of armodafinil
CN104059004A (zh) * 2014-06-25 2014-09-24 江苏斯威森生物医药工程研究中心有限公司 一种2-[(4,4’-二卤-二苯基甲基)巯基]乙酸酯的制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE198165C (enExample)
GB1520812A (en) * 1975-10-02 1978-08-09 Lafon Labor Benzhydrylsulphinyl derivatives
GB1584462A (en) * 1977-03-31 1981-02-11 Lafon Labor N-diaryl-malonamide and diarylmethyl-sulphinyl-acetamide derivatives and pharmaceutical compositions containing them
DE2812542A1 (de) 1978-03-22 1979-10-04 Thomae Gmbh Dr K Neue schwefelhaltige fluorenyl-und phenanthryl-derivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
FR2528038B2 (fr) * 1982-06-04 1985-08-09 Lafon Labor Derives de benzhydrylsulfinylacetamide et leur utilisation en therapeutique
FR2528041A1 (fr) * 1982-06-04 1983-12-09 Lafon Labor Acides halogenobenzhydrylsulfinylacetohydroxamiques, procede de preparation et utilisation en therapeutique
US4964893A (en) * 1986-04-17 1990-10-23 Monsanto Company Benzhydryl compounds as herbicide antidotes
JP3233806B2 (ja) * 1995-01-23 2001-12-04 ユーシービージャパン株式会社 スルフェニル酢酸誘導体の製造法
US5571825A (en) * 1995-03-31 1996-11-05 Warner-Lambert Company Method of selectively inhibiting prostaglandin G/H synthase-2
EP1437345A1 (en) 2003-01-13 2004-07-14 Organisation de Synthese Mondiale Orsymonde Novel method for preparing methyl 2-diphenylmethylsulfinylacetate

Also Published As

Publication number Publication date
ZA200505381B (enExample) 2006-04-26
CA2512084A1 (en) 2004-07-29
CA2512084C (en) 2012-03-20
IL169517A (en) 2012-06-28
JP4690304B2 (ja) 2011-06-01
KR20050091085A (ko) 2005-09-14
EP1583739A1 (en) 2005-10-12
US20060235237A1 (en) 2006-10-19
NZ541089A (en) 2008-05-30
PL377822A1 (pl) 2006-02-20
AU2004203975A1 (en) 2004-07-29
MXPA05007419A (es) 2005-09-12
CN100516035C (zh) 2009-07-22
CN1735591A (zh) 2006-02-15
EP1437345A1 (en) 2004-07-14
BRPI0406489A (pt) 2005-12-06
AR042842A1 (es) 2005-07-06
NO20053602L (no) 2005-07-22
PL212412B1 (pl) 2012-09-28
JP2006516560A (ja) 2006-07-06
NO331507B1 (no) 2012-01-16
US7211684B2 (en) 2007-05-01
IS7958A (is) 2005-07-26
WO2004063149A1 (en) 2004-07-29
TWI323250B (en) 2010-04-11
UA80598C2 (en) 2007-10-10
TW200420530A (en) 2004-10-16
EA200501125A1 (ru) 2005-12-29
KR101062281B1 (ko) 2011-09-06
EA010381B1 (ru) 2008-08-29

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PC1 Assignment before grant (sect. 113)

Owner name: CEPHALON FRANCE

Free format text: FORMER APPLICANT(S): ORGANISATION DE SYNTHESE MONDIALE ORSYMONDE

FGA Letters patent sealed or granted (standard patent)
MK14 Patent ceased section 143(a) (annual fees not paid) or expired