CN100506788C - 芳基烷基氨基甲酸酯衍生物的生产及其在治疗中的用途 - Google Patents
芳基烷基氨基甲酸酯衍生物的生产及其在治疗中的用途 Download PDFInfo
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- CN100506788C CN100506788C CNB2004800027704A CN200480002770A CN100506788C CN 100506788 C CN100506788 C CN 100506788C CN B2004800027704 A CNB2004800027704 A CN B2004800027704A CN 200480002770 A CN200480002770 A CN 200480002770A CN 100506788 C CN100506788 C CN 100506788C
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0300704A FR2850377B1 (fr) | 2003-01-23 | 2003-01-23 | Derives d'arylalkylcarbamates, leur preparation et leur application en therapeutique |
| FR03/00704 | 2003-01-23 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN2007100840856A Division CN101058564B (zh) | 2003-01-23 | 2004-01-22 | 芳基烷基氨基甲酸酯衍生物的生产及其在治疗中的用途 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN1741990A CN1741990A (zh) | 2006-03-01 |
| CN100506788C true CN100506788C (zh) | 2009-07-01 |
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| Application Number | Title | Priority Date | Filing Date |
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| CNB2004800027704A Expired - Fee Related CN100506788C (zh) | 2003-01-23 | 2004-01-22 | 芳基烷基氨基甲酸酯衍生物的生产及其在治疗中的用途 |
| CN2007100840856A Expired - Fee Related CN101058564B (zh) | 2003-01-23 | 2004-01-22 | 芳基烷基氨基甲酸酯衍生物的生产及其在治疗中的用途 |
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| CN2007100840856A Expired - Fee Related CN101058564B (zh) | 2003-01-23 | 2004-01-22 | 芳基烷基氨基甲酸酯衍生物的生产及其在治疗中的用途 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2864080B1 (fr) * | 2003-12-23 | 2006-02-03 | Sanofi Synthelabo | Derives de 1-piperazine-et-1-homopiperazine-carboxylates, leur preparation et leur application en therapeutique |
| FR2865205B1 (fr) | 2004-01-16 | 2006-02-24 | Sanofi Synthelabo | Derives de type aryloxyalkylcarbamates, leur preparation et leur application en therapeutique |
| FR2866886B1 (fr) * | 2004-02-26 | 2007-08-31 | Sanofi Synthelabo | Derives d'aryl-et d'heteroaryl-akylcarbamates, leur preparation et leur application en therapeutique |
| FR2866885B1 (fr) * | 2004-02-26 | 2007-08-31 | Sanofi Synthelabo | Derives de piperidinylalkylcarbamates, leur prepation et leur application en therapeutique |
| FR2866884B1 (fr) * | 2004-02-26 | 2007-08-31 | Sanofi Synthelabo | Derives d'aryl-et d'heteroaryl-piperidinecarboxylates, leur preparation et leur application en therapeutique |
| DE102004039326A1 (de) * | 2004-08-12 | 2006-02-16 | Abbott Gmbh & Co. Kg | Neue medizinische Verwendungen und Verfahren |
| ES2639621T3 (es) | 2004-12-30 | 2017-10-27 | Janssen Pharmaceutica N.V. | Derivados de fenilamida del ácido 4-(bencil)-piperazina-1-carboxílico y compuestos relacionados como moduladores de la amida hidrolasa de ácidos grasos (FAAH) para el tratamiento de la ansiedad, el dolor y otras afecciones |
| US20070155707A1 (en) * | 2005-12-29 | 2007-07-05 | Kadmus Pharmaceuticals, Inc. | Ionizable inhibitors of fatty acid amide hydrolase |
| US20080089845A1 (en) * | 2006-09-07 | 2008-04-17 | N.V. Organon | Methods for determining effective doses of fatty acid amide hydrolase inhibitors in vivo |
| WO2008042892A2 (en) * | 2006-10-02 | 2008-04-10 | N.V. Organon | Fatty acid amide hydrolase inhibitors for energy metabolism disorders |
| WO2008063714A1 (en) * | 2006-11-20 | 2008-05-29 | N.V. Organon | Metabolically-stabilized inhibitors of fatty acid amide hydrolase |
| WO2009009041A2 (en) * | 2007-07-06 | 2009-01-15 | Kinex Pharmaceuticals, Llc | Compositions and methods for modulating a kinase cascade |
| TW200948805A (en) * | 2008-03-07 | 2009-12-01 | Sigma Tau Ind Farmaceuti | Enol carbamate derivatives as modulators of fatty acid amide hydrolase |
| CN101538245B (zh) * | 2008-03-18 | 2011-02-16 | 中国科学院上海药物研究所 | 一类哒嗪酮类化合物及其制备方法和制备药物的用途 |
| UA108233C2 (uk) * | 2010-05-03 | 2015-04-10 | Модулятори активності гідролази амідів жирних кислот | |
| EP2598477B1 (en) | 2010-07-28 | 2016-03-02 | The Regents of The University of California | Peripherally restricted faah inhibitors |
| CN104203906B (zh) | 2011-08-19 | 2018-03-13 | 加利福尼亚大学董事会 | 间位取代的联苯基外周限制性faah抑制剂 |
| CN105263907B (zh) | 2012-08-30 | 2018-11-20 | 阿西纳斯公司 | 作为蛋白质酪氨酸激酶调节剂的n-(3-氟苄基)-2-(5-(4-吗啉代苯基)吡啶-2-基)乙酰胺 |
| ES2908240T3 (es) | 2014-04-07 | 2022-04-28 | Univ California | Inhibidores de la enzima amida hidrolasa de ácidos grasos (FAAH) con biodisponibilidad oral mejorada y su uso como medicamentos |
| MX2021005842A (es) * | 2018-11-20 | 2021-07-15 | Bayer Ag | Antagonistas de los adrenoreceptores a2 subtipo c (alfa-2c) para el tratamiento de la apnea del sueño. |
| CN118515624B (zh) * | 2024-04-29 | 2025-01-24 | 聊城金歌合成材料有限公司 | 一种含三氟甲基多取代恶唑烷-4-酮的合成方法及应用 |
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| US2909467A (en) * | 1958-07-09 | 1959-10-20 | Us Vitamin Pharm Corp | 3-(d-alpha-methylphenethyl)-5-methyl-1, 3-oxazolidine-2, 4-dione |
| NL265085A (enExample) * | 1960-05-24 | |||
| US3742022A (en) * | 1967-05-08 | 1973-06-26 | A Verbiscar | Carbamate esters of physiologically active ph enenthylamines |
| DE3003653A1 (de) * | 1980-02-01 | 1981-08-06 | Hoechst Ag, 6000 Frankfurt | Verfahren zur herstellung von n-substituierten oxazolindionen-(2,4) |
| JP2616989B2 (ja) * | 1989-04-03 | 1997-06-04 | 株式会社トクヤマ | 2,4―オキサゾリジンジオン化合物 |
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