CN100418585C - 稳定的放射性药物组合物及制备方法 - Google Patents

稳定的放射性药物组合物及制备方法 Download PDF

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Publication number
CN100418585C
CN100418585C CNB2004800200430A CN200480020043A CN100418585C CN 100418585 C CN100418585 C CN 100418585C CN B2004800200430 A CNB2004800200430 A CN B2004800200430A CN 200480020043 A CN200480020043 A CN 200480020043A CN 100418585 C CN100418585 C CN 100418585C
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radiopharmaceutical composition
acid
oxidation state
water
compound containing
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CN1822861A (zh
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陈建清
K·E·林德
E·R·马里内利
E·梅特卡夫
A·纳恩
R·E·斯温森
M·特威德勒
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Bracco Imaging SpA
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/12Preparations containing radioactive substances for use in therapy or testing in vivo characterised by a special physical form, e.g. emulsion, microcapsules, liposomes, characterized by a special physical form, e.g. emulsions, dispersions, microcapsules
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • A61K51/08Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins
    • A61K51/088Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins conjugates with carriers being peptides, polyamino acids or proteins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Optics & Photonics (AREA)
  • Epidemiology (AREA)
  • Physics & Mathematics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Dispersion Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
CNB2004800200430A 2003-07-24 2004-07-23 稳定的放射性药物组合物及制备方法 Expired - Fee Related CN100418585C (zh)

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US48985003P 2003-07-24 2003-07-24
US60/489,850 2003-07-24

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CN100418585C true CN100418585C (zh) 2008-09-17

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US (3) US20070269375A1 (enExample)
EP (1) EP1654005A4 (enExample)
JP (2) JP5139678B2 (enExample)
KR (1) KR101106533B1 (enExample)
CN (1) CN100418585C (enExample)
AU (1) AU2004259028C1 (enExample)
BR (1) BRPI0412824A (enExample)
CA (2) CA2526556C (enExample)
IL (1) IL172059A0 (enExample)
RU (1) RU2006105644A (enExample)
SG (2) SG177216A1 (enExample)
WO (1) WO2005009393A2 (enExample)
ZA (1) ZA200509666B (enExample)

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