CL2011001853A1 - Uso de una combinacion farmaceutica que comprende linagliptina y un segundo agente antidiabetico seleccionado entre biguanidas, tiazolidindionas, sulfonilureas, glinidas, entre otros, y, opcionalmente, un tercer agente antidiabetico, para tratar diabetes mellitus tipo 2 y complicaciones de la diabetes, entre otras. - Google Patents

Uso de una combinacion farmaceutica que comprende linagliptina y un segundo agente antidiabetico seleccionado entre biguanidas, tiazolidindionas, sulfonilureas, glinidas, entre otros, y, opcionalmente, un tercer agente antidiabetico, para tratar diabetes mellitus tipo 2 y complicaciones de la diabetes, entre otras.

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Publication number
CL2011001853A1
CL2011001853A1 CL2011001853A CL2011001853A CL2011001853A1 CL 2011001853 A1 CL2011001853 A1 CL 2011001853A1 CL 2011001853 A CL2011001853 A CL 2011001853A CL 2011001853 A CL2011001853 A CL 2011001853A CL 2011001853 A1 CL2011001853 A1 CL 2011001853A1
Authority
CL
Chile
Prior art keywords
antidiabetic agent
optionally
thiazolidinediones
biguanides
sulfonylureas
Prior art date
Application number
CL2011001853A
Other languages
English (en)
Spanish (es)
Inventor
Mody Eva Ulrike Woerle Hans Juergen Graefe
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42174359&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2011001853(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of CL2011001853A1 publication Critical patent/CL2011001853A1/es

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
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    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
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  • Diabetes (AREA)
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  • Cardiology (AREA)
  • Molecular Biology (AREA)
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  • Dermatology (AREA)
  • Emergency Medicine (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Urology & Nephrology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Biochemistry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Oncology (AREA)
  • Physical Education & Sports Medicine (AREA)
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CL2011001853A 2009-02-13 2011-08-02 Uso de una combinacion farmaceutica que comprende linagliptina y un segundo agente antidiabetico seleccionado entre biguanidas, tiazolidindionas, sulfonilureas, glinidas, entre otros, y, opcionalmente, un tercer agente antidiabetico, para tratar diabetes mellitus tipo 2 y complicaciones de la diabetes, entre otras. CL2011001853A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP09152869 2009-02-13

Publications (1)

Publication Number Publication Date
CL2011001853A1 true CL2011001853A1 (es) 2011-11-11

Family

ID=42174359

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2011001853A CL2011001853A1 (es) 2009-02-13 2011-08-02 Uso de una combinacion farmaceutica que comprende linagliptina y un segundo agente antidiabetico seleccionado entre biguanidas, tiazolidindionas, sulfonilureas, glinidas, entre otros, y, opcionalmente, un tercer agente antidiabetico, para tratar diabetes mellitus tipo 2 y complicaciones de la diabetes, entre otras.

Country Status (14)

Country Link
US (6) US20120094894A1 (enExample)
EP (1) EP2395988A2 (enExample)
JP (3) JP2012517977A (enExample)
KR (2) KR20110115582A (enExample)
CN (3) CN106177958A (enExample)
AU (1) AU2010212823B2 (enExample)
BR (1) BRPI1013639A2 (enExample)
CA (1) CA2752437C (enExample)
CL (1) CL2011001853A1 (enExample)
EA (1) EA029759B1 (enExample)
IL (1) IL213716A0 (enExample)
MX (2) MX387264B (enExample)
NZ (2) NZ619520A (enExample)
WO (1) WO2010092163A2 (enExample)

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US7501426B2 (en) 2004-02-18 2009-03-10 Boehringer Ingelheim International Gmbh 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
US7772191B2 (en) 2005-05-10 2010-08-10 Boehringer Ingelheim International Gmbh Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein
DE102005035891A1 (de) 2005-07-30 2007-02-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
EP2540725A1 (de) 2006-05-04 2013-01-02 Boehringer Ingelheim International GmbH Polymorphe von 1-((4-Methyl-chinazolin-2-yl)methyl)-3-methyl-7-(2-butin-1-yl)-8-(3-(R)-amino-piperidin-1-yl)xanthin
PE20080251A1 (es) 2006-05-04 2008-04-25 Boehringer Ingelheim Int Usos de inhibidores de dpp iv
EP1852108A1 (en) 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG DPP IV inhibitor formulations
PE20090938A1 (es) 2007-08-16 2009-08-08 Boehringer Ingelheim Int Composicion farmaceutica que comprende un derivado de benceno sustituido con glucopiranosilo
PE20091730A1 (es) 2008-04-03 2009-12-10 Boehringer Ingelheim Int Formulaciones que comprenden un inhibidor de dpp4
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JP2012517977A (ja) 2012-08-09
IL213716A0 (en) 2011-07-31
CA2752437A1 (en) 2010-08-19
WO2010092163A2 (en) 2010-08-19
JP2017081984A (ja) 2017-05-18
AU2010212823B2 (en) 2016-01-28
US20180344741A1 (en) 2018-12-06
EA201101187A1 (ru) 2012-10-30
CA2752437C (en) 2017-07-11
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US20170173027A1 (en) 2017-06-22
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BRPI1013639A2 (pt) 2016-04-19
EP2395988A2 (en) 2011-12-21
MX2011008416A (es) 2011-09-08
CN117547538A (zh) 2024-02-13
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US20150105318A1 (en) 2015-04-16
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