AU2010212823B2 - Antidiabetic medications comprising a DPP-4 inhibitor (linagliptin) optionally in combination with other antidiabetics - Google Patents

Antidiabetic medications comprising a DPP-4 inhibitor (linagliptin) optionally in combination with other antidiabetics Download PDF

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Publication number
AU2010212823B2
AU2010212823B2 AU2010212823A AU2010212823A AU2010212823B2 AU 2010212823 B2 AU2010212823 B2 AU 2010212823B2 AU 2010212823 A AU2010212823 A AU 2010212823A AU 2010212823 A AU2010212823 A AU 2010212823A AU 2010212823 B2 AU2010212823 B2 AU 2010212823B2
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AU
Australia
Prior art keywords
antidiabetic agent
dpp
inhibitor
pharmaceutically acceptable
acceptable salt
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Application number
AU2010212823A
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AU2010212823A1 (en
Inventor
Eva Ulrike Graefe-Mody
Hans-Juergen Woerle
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Boehringer Ingelheim International GmbH
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Boehringer Ingelheim International GmbH
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
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  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Diabetes (AREA)
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  • Molecular Biology (AREA)
  • Endocrinology (AREA)
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  • Immunology (AREA)
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  • Dermatology (AREA)
  • Emergency Medicine (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Urology & Nephrology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Biochemistry (AREA)
  • Child & Adolescent Psychology (AREA)
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  • Communicable Diseases (AREA)
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AU2010212823A 2009-02-13 2010-02-12 Antidiabetic medications comprising a DPP-4 inhibitor (linagliptin) optionally in combination with other antidiabetics Active AU2010212823B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP09152869.5 2009-02-13
EP09152869 2009-02-13
PCT/EP2010/051817 WO2010092163A2 (en) 2009-02-13 2010-02-12 Antidiabetic medications

Publications (2)

Publication Number Publication Date
AU2010212823A1 AU2010212823A1 (en) 2011-08-18
AU2010212823B2 true AU2010212823B2 (en) 2016-01-28

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Application Number Title Priority Date Filing Date
AU2010212823A Active AU2010212823B2 (en) 2009-02-13 2010-02-12 Antidiabetic medications comprising a DPP-4 inhibitor (linagliptin) optionally in combination with other antidiabetics

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Country Link
US (6) US20120094894A1 (enExample)
EP (1) EP2395988A2 (enExample)
JP (3) JP2012517977A (enExample)
KR (2) KR20110115582A (enExample)
CN (3) CN106177958A (enExample)
AU (1) AU2010212823B2 (enExample)
BR (1) BRPI1013639A2 (enExample)
CA (1) CA2752437C (enExample)
CL (1) CL2011001853A1 (enExample)
EA (1) EA029759B1 (enExample)
IL (1) IL213716A0 (enExample)
MX (2) MX387264B (enExample)
NZ (2) NZ619520A (enExample)
WO (1) WO2010092163A2 (enExample)

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US7501426B2 (en) 2004-02-18 2009-03-10 Boehringer Ingelheim International Gmbh 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
US7772191B2 (en) 2005-05-10 2010-08-10 Boehringer Ingelheim International Gmbh Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein
DE102005035891A1 (de) 2005-07-30 2007-02-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
EP2540725A1 (de) 2006-05-04 2013-01-02 Boehringer Ingelheim International GmbH Polymorphe von 1-((4-Methyl-chinazolin-2-yl)methyl)-3-methyl-7-(2-butin-1-yl)-8-(3-(R)-amino-piperidin-1-yl)xanthin
PE20080251A1 (es) 2006-05-04 2008-04-25 Boehringer Ingelheim Int Usos de inhibidores de dpp iv
EP1852108A1 (en) 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG DPP IV inhibitor formulations
PE20090938A1 (es) 2007-08-16 2009-08-08 Boehringer Ingelheim Int Composicion farmaceutica que comprende un derivado de benceno sustituido con glucopiranosilo
PE20091730A1 (es) 2008-04-03 2009-12-10 Boehringer Ingelheim Int Formulaciones que comprenden un inhibidor de dpp4
EP2146210A1 (en) 2008-04-07 2010-01-20 Arena Pharmaceuticals, Inc. Methods of using A G protein-coupled receptor to identify peptide YY (PYY) secretagogues and compounds useful in the treatment of conditions modulated by PYY
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