CN106177958A - 包含dpp‑4抑制剂(利拉列汀)任选地组合其它抗糖尿病药的抗糖尿病药物 - Google Patents
包含dpp‑4抑制剂(利拉列汀)任选地组合其它抗糖尿病药的抗糖尿病药物 Download PDFInfo
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- CN106177958A CN106177958A CN201610580276.0A CN201610580276A CN106177958A CN 106177958 A CN106177958 A CN 106177958A CN 201610580276 A CN201610580276 A CN 201610580276A CN 106177958 A CN106177958 A CN 106177958A
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- antidiabetic drug
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| CN2010800161446A CN102387795A (zh) | 2009-02-13 | 2010-02-12 | 包含dpp-4抑制剂(利拉列汀)任选地组合其它抗糖尿病药的抗糖尿病药物 |
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| CN202310997781.5A Pending CN117547538A (zh) | 2009-02-13 | 2010-02-12 | 包含dpp-4抑制剂(利格列汀)任选地组合其它抗糖尿病药的抗糖尿病药物 |
| CN2010800161446A Pending CN102387795A (zh) | 2009-02-13 | 2010-02-12 | 包含dpp-4抑制剂(利拉列汀)任选地组合其它抗糖尿病药的抗糖尿病药物 |
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| CN2010800161446A Pending CN102387795A (zh) | 2009-02-13 | 2010-02-12 | 包含dpp-4抑制剂(利拉列汀)任选地组合其它抗糖尿病药的抗糖尿病药物 |
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Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN110652498A (zh) * | 2019-11-22 | 2020-01-07 | 河南合智医药科技有限公司 | 一种用于治疗2型糖尿病的药物剂型及其制备方法 |
| CN112423761A (zh) * | 2018-07-17 | 2021-02-26 | 勃林格殷格翰国际有限公司 | 心脏安全的抗糖尿病疗法 |
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| US7407955B2 (en) | 2002-08-21 | 2008-08-05 | Boehringer Ingelheim Pharma Gmbh & Co., Kg | 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions |
| US7501426B2 (en) | 2004-02-18 | 2009-03-10 | Boehringer Ingelheim International Gmbh | 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions |
| DE102004054054A1 (de) | 2004-11-05 | 2006-05-11 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine |
| US7772191B2 (en) | 2005-05-10 | 2010-08-10 | Boehringer Ingelheim International Gmbh | Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein |
| DE102005035891A1 (de) | 2005-07-30 | 2007-02-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel |
| EP1852108A1 (en) | 2006-05-04 | 2007-11-07 | Boehringer Ingelheim Pharma GmbH & Co.KG | DPP IV inhibitor formulations |
| SG174054A1 (en) | 2006-05-04 | 2011-09-29 | Boehringer Ingelheim Int | Polymorphs |
| PE20110235A1 (es) | 2006-05-04 | 2011-04-14 | Boehringer Ingelheim Int | Combinaciones farmaceuticas que comprenden linagliptina y metmorfina |
| CL2008002427A1 (es) | 2007-08-16 | 2009-09-11 | Boehringer Ingelheim Int | Composicion farmaceutica que comprende 1-cloro-4-(b-d-glucopiranos-1-il)-2-[4-((s)-tetrahidrofurano-3-iloxi)bencil]-benceno combinado con 1-[(4-metilquinazolin-2-il)metil]-3-metil-7-(2-butin-1-il)-8-(3-(r)-aminopiperidin-1-il)xantina; y su uso para tratar diabetes mellitus tipo 2. |
| PE20140960A1 (es) | 2008-04-03 | 2014-08-15 | Boehringer Ingelheim Int | Formulaciones que comprenden un inhibidor de dpp4 |
| EP2146210A1 (en) | 2008-04-07 | 2010-01-20 | Arena Pharmaceuticals, Inc. | Methods of using A G protein-coupled receptor to identify peptide YY (PYY) secretagogues and compounds useful in the treatment of conditions modulated by PYY |
| UY32030A (es) | 2008-08-06 | 2010-03-26 | Boehringer Ingelheim Int | "tratamiento para diabetes en pacientes inapropiados para terapia con metformina" |
| BRPI0916997A2 (pt) | 2008-08-06 | 2020-12-15 | Boehringer Ingelheim International Gmbh | Inibidor de dpp-4 e seu uso |
| PE20110297A1 (es) * | 2008-08-15 | 2011-05-26 | Boehringer Ingelheim Int | Inhibidores de dpp-4 para la cicatrizacion de heridas |
| RU2011113823A (ru) | 2008-09-10 | 2012-10-20 | БЕРИНГЕР ИНГЕЛЬХАЙМ ИНТЕРНАЦИОНАЛЬ ГмбХ (DE) | Комбинированная терапия, предназначенная для лечения диабета и связанных с ним состояний |
| US20200155558A1 (en) | 2018-11-20 | 2020-05-21 | Boehringer Ingelheim International Gmbh | Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug |
| HUE048608T2 (hu) | 2008-10-17 | 2020-08-28 | Sanofi Aventis Deutschland | Egy inzulin és egy GLP-1 agonista kombinációja |
| EP2382216A1 (en) | 2008-12-23 | 2011-11-02 | Boehringer Ingelheim International GmbH | Salt forms of organic compound |
| AR074990A1 (es) | 2009-01-07 | 2011-03-02 | Boehringer Ingelheim Int | Tratamiento de diabetes en pacientes con un control glucemico inadecuado a pesar de la terapia con metformina |
| SG173619A1 (en) | 2009-02-13 | 2011-09-29 | Boehringer Ingelheim Int | Pharmaceutical composition comprising a sglt2 inhibitor, a dpp-iv inhibitor and optionally a further antidiabetic agent and uses thereof |
| WO2011039108A2 (en) | 2009-09-30 | 2011-04-07 | Boehringer Ingelheim International Gmbh | Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives |
| US10610489B2 (en) | 2009-10-02 | 2020-04-07 | Boehringer Ingelheim International Gmbh | Pharmaceutical composition, pharmaceutical dosage form, process for their preparation, methods for treating and uses thereof |
| BR112012011726A2 (pt) | 2009-11-13 | 2020-05-19 | Bristol-Myers Squibb Company | comprimidos de duas camadas, seu uso, e suas combinações farmacêuticas |
| RU2537239C2 (ru) | 2009-11-13 | 2014-12-27 | Санофи-Авентис Дойчланд Гмбх | Фармацевтическая композиция, включающая агонист glp-1, инсулин и метионин |
| LT2498801T (lt) | 2009-11-13 | 2018-05-10 | Sanofi-Aventis Deutschland Gmbh | Farmacinė kompozicija, apimanti despro36eksendin-4(1-39)-lys6-nh2 ir metioniną |
| EP3646859A1 (en) | 2009-11-27 | 2020-05-06 | Boehringer Ingelheim International GmbH | Treatment of genotyped diabetic patients with dpp-iv inhibitors such as linagliptin |
| NZ602921A (en) | 2010-05-05 | 2016-01-29 | Boehringer Ingelheim Int | Combination therapy comprising the administration of a glp-1 receptor agonist and a ddp-4 inhibitor |
| CA2795105A1 (en) * | 2010-05-05 | 2011-11-10 | Peter Schneider | Pharmaceutical formulations comprising pioglitazone and linagliptin |
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- 2010-02-12 US US13/148,065 patent/US20120094894A1/en not_active Abandoned
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- 2010-02-12 NZ NZ619520A patent/NZ619520A/en unknown
- 2010-02-12 KR KR1020117018784A patent/KR20110115582A/ko not_active Ceased
- 2010-02-12 CN CN201610580276.0A patent/CN106177958A/zh active Pending
- 2010-02-12 BR BRPI1013639A patent/BRPI1013639A2/pt not_active Application Discontinuation
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- 2010-02-12 EP EP10704924A patent/EP2395988A2/en active Pending
- 2010-02-12 AU AU2010212823A patent/AU2010212823B2/en active Active
- 2010-02-12 KR KR1020167034411A patent/KR20160143897A/ko not_active Ceased
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- 2010-02-12 JP JP2011549582A patent/JP2012517977A/ja not_active Withdrawn
- 2010-02-12 CN CN2010800161446A patent/CN102387795A/zh active Pending
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- 2014-12-22 US US14/578,552 patent/US20150105318A1/en not_active Abandoned
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2020
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| CN112423761A (zh) * | 2018-07-17 | 2021-02-26 | 勃林格殷格翰国际有限公司 | 心脏安全的抗糖尿病疗法 |
| CN110652498A (zh) * | 2019-11-22 | 2020-01-07 | 河南合智医药科技有限公司 | 一种用于治疗2型糖尿病的药物剂型及其制备方法 |
| CN110652498B (zh) * | 2019-11-22 | 2022-04-05 | 河南合智医药科技有限公司 | 一种用于治疗2型糖尿病的药物制剂及其制备方法 |
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| IL213716A0 (en) | 2011-07-31 |
| CL2011001853A1 (es) | 2011-11-11 |
| WO2010092163A2 (en) | 2010-08-19 |
| CN102387795A (zh) | 2012-03-21 |
| JP2015044875A (ja) | 2015-03-12 |
| AU2010212823A1 (en) | 2011-08-18 |
| NZ619520A (en) | 2015-06-26 |
| AU2010212823B2 (en) | 2016-01-28 |
| JP6556767B2 (ja) | 2019-08-07 |
| NZ594044A (en) | 2014-08-29 |
| EA201101187A1 (ru) | 2012-10-30 |
| JP2017081984A (ja) | 2017-05-18 |
| KR20160143897A (ko) | 2016-12-14 |
| MX387264B (es) | 2025-03-18 |
| JP2012517977A (ja) | 2012-08-09 |
| CN117547538A (zh) | 2024-02-13 |
| US20120094894A1 (en) | 2012-04-19 |
| US20200323861A1 (en) | 2020-10-15 |
| CA2752437C (en) | 2017-07-11 |
| US20220088023A1 (en) | 2022-03-24 |
| US20170173027A1 (en) | 2017-06-22 |
| CA2752437A1 (en) | 2010-08-19 |
| WO2010092163A3 (en) | 2010-10-21 |
| EA029759B1 (ru) | 2018-05-31 |
| MX2011008416A (es) | 2011-09-08 |
| US20180344741A1 (en) | 2018-12-06 |
| BRPI1013639A2 (pt) | 2016-04-19 |
| KR20110115582A (ko) | 2011-10-21 |
| EP2395988A2 (en) | 2011-12-21 |
| US20150105318A1 (en) | 2015-04-16 |
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