CH615198A5 - Process for the preparation of daunomycin - Google Patents

Process for the preparation of daunomycin Download PDF

Info

Publication number
CH615198A5
CH615198A5 CH352975A CH352975A CH615198A5 CH 615198 A5 CH615198 A5 CH 615198A5 CH 352975 A CH352975 A CH 352975A CH 352975 A CH352975 A CH 352975A CH 615198 A5 CH615198 A5 CH 615198A5
Authority
CH
Switzerland
Prior art keywords
trideoxy
chloro
trifluoroacetoxy
trifluoroacetamido
daunomycin
Prior art date
Application number
CH352975A
Other languages
German (de)
English (en)
Inventor
Federico Arcamone
Aurelio Di Marco
Sergio Penco
Original Assignee
Farmaceutici Italia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmaceutici Italia filed Critical Farmaceutici Italia
Publication of CH615198A5 publication Critical patent/CH615198A5/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/24—Condensed ring systems having three or more rings
    • C07H15/252—Naphthacene radicals, e.g. daunomycins, adriamycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
CH352975A 1974-03-20 1975-03-19 Process for the preparation of daunomycin CH615198A5 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB1225474A GB1457559A (en) 1974-03-20 1974-03-20 Daunomycins

Publications (1)

Publication Number Publication Date
CH615198A5 true CH615198A5 (en) 1980-01-15

Family

ID=10001195

Family Applications (1)

Application Number Title Priority Date Filing Date
CH352975A CH615198A5 (en) 1974-03-20 1975-03-19 Process for the preparation of daunomycin

Country Status (13)

Country Link
JP (1) JPS5833880B2 (pt)
AT (1) AT338419B (pt)
BE (1) BE826848A (pt)
CA (1) CA1046508A (pt)
CH (1) CH615198A5 (pt)
DE (1) DE2510926C3 (pt)
DK (1) DK146541C (pt)
FR (1) FR2264554B1 (pt)
GB (1) GB1457559A (pt)
NL (1) NL176636C (pt)
SE (1) SE434843B (pt)
SU (1) SU589926A3 (pt)
ZA (1) ZA751687B (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5977082A (en) * 1985-08-02 1999-11-02 Pharmacia & Upjohn Company Injectable ready-to-use solutions containing an antitumor anthracycline glycoside
US5124317A (en) * 1985-08-02 1992-06-23 Farmitalia Carlo Erba S.P.A. Injectable ready-to-use solutions containing an antitumor anthracycline glycoside
FR2678274A1 (fr) * 1991-06-25 1992-12-31 Medgenix Group Sa N-leucyl epirubicine application a titre de medicament antitumoral et procede de preparation.

Also Published As

Publication number Publication date
GB1457559A (en) 1976-12-08
DK146541C (da) 1984-04-09
NL176636C (nl) 1985-05-17
DK146541B (da) 1983-10-31
SE7503084L (pt) 1975-09-22
NL176636B (nl) 1984-12-17
DE2510926A1 (de) 1975-09-25
AT338419B (de) 1977-08-25
SE7503084A (pt) 1975-09-22
CA1046508A (en) 1979-01-16
FR2264554A1 (pt) 1975-10-17
SE434843B (sv) 1984-08-20
BE826848A (fr) 1975-09-19
ZA751687B (en) 1976-02-25
DE2510926B2 (de) 1979-07-19
NL7503079A (nl) 1975-09-23
AU7919775A (en) 1976-09-23
JPS50126657A (pt) 1975-10-04
SU589926A3 (ru) 1978-01-25
DE2510926C3 (de) 1980-03-13
ATA202875A (de) 1976-12-15
DK109275A (pt) 1975-09-21
FR2264554B1 (pt) 1978-07-28
JPS5833880B2 (ja) 1983-07-22

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Legal Events

Date Code Title Description
PL Patent ceased