CH609046A5 - - Google Patents

Info

Publication number
CH609046A5
CH609046A5 CH1426274A CH1426274A CH609046A5 CH 609046 A5 CH609046 A5 CH 609046A5 CH 1426274 A CH1426274 A CH 1426274A CH 1426274 A CH1426274 A CH 1426274A CH 609046 A5 CH609046 A5 CH 609046A5
Authority
CH
Switzerland
Application number
CH1426274A
Inventor
Herbert Dr Merz
Adolf Dr Langbein
Gerhard Dr Walther
Klaus Dr Stockhaus
Original Assignee
Boehringer Sohn Ingelheim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Sohn Ingelheim filed Critical Boehringer Sohn Ingelheim
Publication of CH609046A5 publication Critical patent/CH609046A5/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
CH1426274A 1973-10-27 1974-10-24 CH609046A5 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19732354002 DE2354002A1 (de) 1973-10-27 1973-10-27 Neue n-(methoxymethyl-furylmethyl)6,7-benzomorphane und -morphinane, deren saeureadditionssalze, ihre verwendung als arzneimittel und verfahren zu deren herstellung

Publications (1)

Publication Number Publication Date
CH609046A5 true CH609046A5 (fr) 1979-02-15

Family

ID=5896658

Family Applications (6)

Application Number Title Priority Date Filing Date
CH1426374A CH609047A5 (fr) 1973-10-27 1974-10-24
CH1426574A CH609340A5 (fr) 1973-10-27 1974-10-24
CH1426274A CH609046A5 (fr) 1973-10-27 1974-10-24
CH1426474A CH609048A5 (fr) 1973-10-27 1974-10-24
CH1436974A CH609685A5 (fr) 1973-10-27 1974-10-25
CH1437074A CH609686A5 (fr) 1973-10-27 1974-10-25

Family Applications Before (2)

Application Number Title Priority Date Filing Date
CH1426374A CH609047A5 (fr) 1973-10-27 1974-10-24
CH1426574A CH609340A5 (fr) 1973-10-27 1974-10-24

Family Applications After (3)

Application Number Title Priority Date Filing Date
CH1426474A CH609048A5 (fr) 1973-10-27 1974-10-24
CH1436974A CH609685A5 (fr) 1973-10-27 1974-10-25
CH1437074A CH609686A5 (fr) 1973-10-27 1974-10-25

Country Status (27)

Country Link
US (1) US3981874A (fr)
JP (1) JPS5738590B2 (fr)
AT (6) AT335631B (fr)
BE (1) BE821505A (fr)
BG (3) BG27902A3 (fr)
CA (1) CA1056377A (fr)
CH (6) CH609047A5 (fr)
CS (3) CS171194B2 (fr)
DD (1) DD115909A5 (fr)
DE (1) DE2354002A1 (fr)
DK (1) DK138325C (fr)
ES (6) ES431057A1 (fr)
FI (1) FI62079C (fr)
FR (1) FR2248838B1 (fr)
GB (1) GB1482552A (fr)
HU (1) HU176479B (fr)
IE (1) IE41528B1 (fr)
IL (1) IL45938A (fr)
NL (1) NL7413980A (fr)
NO (1) NO140859C (fr)
PH (1) PH11894A (fr)
PL (3) PL92052B1 (fr)
RO (5) RO65656A (fr)
SE (1) SE422791B (fr)
SU (6) SU510999A3 (fr)
YU (5) YU36950B (fr)
ZA (1) ZA746790B (fr)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1513961A (en) * 1975-02-25 1978-06-14 Acf Chemiefarma Nv 6,7-benzomorphans method for their preparation and intermediates
US4208523A (en) * 1978-11-30 1980-06-17 Sterling Drug Inc. 11-Lower-alkyl-, 11-phenyl-lower-alkyl- and 11-cyclo-lower-alkyl-lower-alkyl-hexahydro-2,6-methano-3-benzazocines
AR067673A1 (es) 2007-07-26 2009-10-21 Vitae Pharmaceuticals Inc Derivados de 1,3 oxazinan - 2 - ona como inhibidores ciclicos de la 11 beta -hidroxiesteroide deshidrogenasa 1. composiciones farmaceuticas.
JP5769970B2 (ja) * 2007-11-16 2015-08-26 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ベンゾモルファン及び関連骨格のアリール−及びヘテロアリールカルボニル誘導体、かかる化合物を含有する医薬及びこれらの使用
CA2708303A1 (fr) 2007-12-11 2009-06-18 Vitae Pharmaceuticals, Inc. Inhibiteurs cycliques d'uree de la 11.beta.-hydroxysteroide dehydrogenase 1
TW200934490A (en) 2008-01-07 2009-08-16 Vitae Pharmaceuticals Inc Lactam inhibitors of 11 &abgr;-hydroxysteroid dehydrogenase 1
JP5490020B2 (ja) 2008-01-24 2014-05-14 ヴァイティー ファーマシューティカルズ,インコーポレイテッド 11β−ヒドロキシステロイドデヒドロゲナーゼ1の環状カルバゼート及びセミカルバジドインヒビター
ATE531696T1 (de) * 2008-02-12 2011-11-15 Boehringer Ingelheim Int Harnstoff-derivate von benzomorphanen, entsprechende gerüste, medikamente mit solchen verbindungen und ihre verwendung
CA2715290A1 (fr) 2008-02-15 2009-08-20 Vitae Pharmaceuticals, Inc. Inhibiteurs de la 11 beta-hydroxysteroide dehydrogenase 1
CA2723034A1 (fr) 2008-05-01 2009-11-05 Vitae Pharmaceuticals, Inc. Inhibiteurs cycliques de la 11-beta-hydroxysteroide dehydrogenase 1
AR071236A1 (es) 2008-05-01 2010-06-02 Vitae Pharmaceuticals Inc Inhibidores ciclicos de la 11beta-hidroxiesteroide deshidrogenasa 1
NZ588954A (en) 2008-05-01 2012-08-31 Vitae Pharmaceuticals Inc Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
US8765780B2 (en) 2008-05-13 2014-07-01 Boehringer Ingelheim International Gmbh Alicyclic carboxylic acid derivatives of benzomorphans and related scaffolds, medicaments containing such compounds and their use
JP5777030B2 (ja) 2008-07-25 2015-09-09 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 11β−ヒドロキシステロイドデヒドロゲナーゼ1の阻害剤
CN102119160B (zh) 2008-07-25 2014-11-05 贝林格尔·英格海姆国际有限公司 11β-羟基类固醇脱氢酶1的环状抑制剂
US8680093B2 (en) 2009-04-30 2014-03-25 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
JP5656986B2 (ja) 2009-06-11 2015-01-21 ヴァイティー ファーマシューティカルズ,インコーポレイテッド 1,3−オキサジナン−2−オン構造に基づく11β−ヒドロキシステロイドデヒドロゲナーゼ1の環状阻害剤
UY33001A (es) * 2009-11-06 2011-05-31 Boehringer Ingelheim Int Derivados arilo y heteroarilcarbonilo de hexahidroindenopiridina y octahidrobenzoquinolina
EP2582698B1 (fr) 2010-06-16 2016-09-14 Vitae Pharmaceuticals, Inc. Hétérocycles à 5, 6 et 7 chaînons substitués, médicaments contenant ces composés et leur utilisation
TWI537258B (zh) 2010-11-05 2016-06-11 百靈佳殷格翰國際股份有限公司 六氫茚并吡啶及八氫苯并喹啉之芳基-及雜環芳基羰基衍生物
JP2014524438A (ja) 2011-08-17 2014-09-22 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング インデノピリジン誘導体

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3632591A (en) * 1968-07-19 1972-01-04 Sterling Drug Inc 1 2 3 4 5 6 - hexahydro-3-(cycloaliphatic or cycloaliphatic 11-dimethyl-2 alkyl)-66-methano-3-benzazocines
US3833595A (en) * 1968-12-26 1974-09-03 Sumitomo Chemical Co 2-aroylalkyl benzomorphans
CS166803B2 (fr) * 1971-02-08 1976-03-29 Boehringer Sohn Ingelheim

Also Published As

Publication number Publication date
PL92086B1 (fr) 1977-03-31
ATA828774A (de) 1976-07-15
SU511005A3 (ru) 1976-04-15
RO65659A (fr) 1980-06-15
YU285274A (en) 1982-02-25
SU510999A3 (ru) 1976-04-15
IE41528L (en) 1975-04-27
IE41528B1 (en) 1980-01-30
NO140859B (no) 1979-08-20
SU508193A3 (ru) 1976-03-25
ATA828974A (de) 1976-08-15
FI62079B (fi) 1982-07-30
NL7413980A (nl) 1975-04-29
YU36952B (en) 1984-08-31
NO743845L (fr) 1975-05-26
SU508192A3 (ru) 1976-03-25
CS171196B2 (fr) 1976-10-29
YU285174A (en) 1982-06-18
YU285474A (en) 1982-06-18
YU36951B (en) 1984-08-31
ATA828574A (de) 1976-07-15
AT336202B (de) 1977-04-25
IL45938A0 (en) 1974-12-31
ES431058A1 (es) 1976-10-16
DK559874A (fr) 1975-06-23
JPS5071679A (fr) 1975-06-13
PL92053B1 (fr) 1977-03-31
BE821505A (fr) 1975-04-25
US3981874A (en) 1976-09-21
ATA829074A (de) 1976-07-15
ES431056A1 (es) 1976-10-16
ES431057A1 (es) 1976-10-16
YU285674A (en) 1982-06-18
RO65657A (fr) 1980-06-15
CS171194B2 (fr) 1976-10-29
BG27901A3 (en) 1980-01-15
HU176479B (en) 1981-03-28
SE7413485L (fr) 1975-04-28
AT335633B (de) 1977-03-25
DE2354002A1 (de) 1975-05-07
SU512707A3 (ru) 1976-04-30
SE422791B (sv) 1982-03-29
ATA828874A (de) 1976-06-15
NO140859C (no) 1979-11-28
FR2248838A1 (fr) 1975-05-23
CA1056377A (fr) 1979-06-12
BG27903A3 (en) 1980-01-15
CH609686A5 (fr) 1979-03-15
AT335634B (de) 1977-03-25
CH609685A5 (fr) 1979-03-15
FR2248838B1 (fr) 1977-11-04
YU285374A (en) 1982-06-18
PL92052B1 (fr) 1977-03-31
BG27902A3 (en) 1980-01-15
CH609340A5 (fr) 1979-02-28
ZA746790B (en) 1976-06-30
ES431054A1 (es) 1976-10-16
RO65658A (fr) 1979-07-15
AT335631B (de) 1977-03-25
ATA828674A (de) 1976-07-15
YU36519B (en) 1984-02-29
CS171195B2 (fr) 1976-10-29
CH609048A5 (fr) 1979-02-15
ES431055A1 (es) 1976-10-16
DK138325C (da) 1979-01-22
DK138325B (da) 1978-08-14
PH11894A (en) 1978-08-29
CH609047A5 (fr) 1979-02-15
RO65656A (fr) 1980-06-15
IL45938A (en) 1977-12-30
AT335632B (de) 1977-03-25
YU36949B (en) 1984-08-31
FI314174A (fr) 1975-04-28
FI62079C (fi) 1982-11-10
RO65655A (fr) 1980-06-15
GB1482552A (en) 1977-08-10
DD115909A5 (fr) 1975-10-20
JPS5738590B2 (fr) 1982-08-16
AT335076B (de) 1977-02-25
SU578870A3 (ru) 1977-10-30
ES431059A1 (es) 1976-10-16
YU36950B (en) 1984-08-31

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Legal Events

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PL Patent ceased