CA3018986A1 - Substituted aminopurine compounds, compositions thereof, and methods of treatment therewith - Google Patents
Substituted aminopurine compounds, compositions thereof, and methods of treatment therewith Download PDFInfo
- Publication number
- CA3018986A1 CA3018986A1 CA3018986A CA3018986A CA3018986A1 CA 3018986 A1 CA3018986 A1 CA 3018986A1 CA 3018986 A CA3018986 A CA 3018986A CA 3018986 A CA3018986 A CA 3018986A CA 3018986 A1 CA3018986 A1 CA 3018986A1
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- Canada
- Prior art keywords
- cancer
- purin
- cyclohexanecarboxamide
- substituted
- unsubstituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A61K31/52—Purines, e.g. adenine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201662317412P | 2016-04-01 | 2016-04-01 | |
| US62/317,412 | 2016-04-01 | ||
| PCT/US2017/025252 WO2017173206A1 (en) | 2016-04-01 | 2017-03-31 | Substituted aminopurine compounds, compositions thereof, and methods of treatment therewith |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA3018986A1 true CA3018986A1 (en) | 2017-10-05 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA3018986A Abandoned CA3018986A1 (en) | 2016-04-01 | 2017-03-31 | Substituted aminopurine compounds, compositions thereof, and methods of treatment therewith |
Country Status (15)
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|---|---|
| US (1) | US10576085B2 (OSRAM) |
| EP (1) | EP3436018A4 (OSRAM) |
| JP (1) | JP7014731B2 (OSRAM) |
| KR (1) | KR102356433B1 (OSRAM) |
| CN (1) | CN109069512B (OSRAM) |
| AU (1) | AU2017241837B2 (OSRAM) |
| BR (1) | BR112018070163A2 (OSRAM) |
| CA (1) | CA3018986A1 (OSRAM) |
| CL (1) | CL2018002787A1 (OSRAM) |
| EA (1) | EA039392B1 (OSRAM) |
| IL (1) | IL262007B2 (OSRAM) |
| MX (1) | MX379513B (OSRAM) |
| NZ (1) | NZ746554A (OSRAM) |
| SG (2) | SG11201808388QA (OSRAM) |
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2017
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- 2017-03-31 JP JP2018551358A patent/JP7014731B2/ja active Active
- 2017-03-31 SG SG11201808388QA patent/SG11201808388QA/en unknown
- 2017-03-31 KR KR1020187028514A patent/KR102356433B1/ko active Active
- 2017-03-31 IL IL262007A patent/IL262007B2/en unknown
- 2017-03-31 WO PCT/US2017/025252 patent/WO2017173206A1/en not_active Ceased
- 2017-03-31 BR BR112018070163A patent/BR112018070163A2/pt not_active Application Discontinuation
- 2017-03-31 CA CA3018986A patent/CA3018986A1/en not_active Abandoned
- 2017-03-31 EA EA201892229A patent/EA039392B1/ru unknown
- 2017-03-31 NZ NZ746554A patent/NZ746554A/en unknown
- 2017-03-31 US US15/475,899 patent/US10576085B2/en active Active
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- 2017-03-31 EP EP17776735.7A patent/EP3436018A4/en not_active Withdrawn
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Also Published As
| Publication number | Publication date |
|---|---|
| BR112018070163A2 (pt) | 2019-01-29 |
| JP2019510066A (ja) | 2019-04-11 |
| IL262007A (en) | 2018-10-31 |
| KR20180126497A (ko) | 2018-11-27 |
| IL262007B2 (en) | 2023-04-01 |
| EA201892229A1 (ru) | 2019-03-29 |
| CN109069512B (zh) | 2022-06-14 |
| CN109069512A (zh) | 2018-12-21 |
| US10576085B2 (en) | 2020-03-03 |
| MX379513B (es) | 2025-03-11 |
| KR102356433B1 (ko) | 2022-01-27 |
| WO2017173206A1 (en) | 2017-10-05 |
| CL2018002787A1 (es) | 2019-01-18 |
| EP3436018A1 (en) | 2019-02-06 |
| NZ746554A (en) | 2023-03-31 |
| MX2018011992A (es) | 2019-01-24 |
| SG11201808388QA (en) | 2018-10-30 |
| EA039392B1 (ru) | 2022-01-21 |
| US20170281633A1 (en) | 2017-10-05 |
| JP7014731B2 (ja) | 2022-02-01 |
| AU2017241837A1 (en) | 2018-10-25 |
| EP3436018A4 (en) | 2019-11-13 |
| IL262007B (en) | 2022-12-01 |
| AU2017241837B2 (en) | 2021-07-22 |
| SG10202009589UA (en) | 2020-10-29 |
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