CA2783314A1 - 4-oxo-1h-quinoline-3-carboxamides as modulators of atp-binding cassette transporters - Google Patents

4-oxo-1h-quinoline-3-carboxamides as modulators of atp-binding cassette transporters Download PDF

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Publication number
CA2783314A1
CA2783314A1 CA2783314A CA2783314A CA2783314A1 CA 2783314 A1 CA2783314 A1 CA 2783314A1 CA 2783314 A CA2783314 A CA 2783314A CA 2783314 A CA2783314 A CA 2783314A CA 2783314 A1 CA2783314 A1 CA 2783314A1
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Canada
Prior art keywords
oxo
carboxamide
phenyl
quinoline
trifluoromethyl
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Abandoned
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CA2783314A
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English (en)
French (fr)
Inventor
Urvi Sheth
Lev T.D. Fanning
Mehdi Numa
Hayley Binch
Dennis James Hurley
Jinglan Zhou
Sara S. Hadida Ruah
Anna R. Hazlewood
Alina Silina
Rajendran Vairagoundar
Fredrick F. Van Goor
Peter Diederik Jan Grootenhuis
Martyn C. Botfield
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Vertex Pharmaceuticals Inc
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Vertex Pharmaceuticals Inc
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Application filed by Vertex Pharmaceuticals Inc filed Critical Vertex Pharmaceuticals Inc
Publication of CA2783314A1 publication Critical patent/CA2783314A1/en
Abandoned legal-status Critical Current

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TWI439462B (zh) 2007-12-10 2014-06-01 Novartis Ag 作為ｅｎａｃ阻抑劑之螺環胍化合物
US20110257223A1 (en) * 2008-10-23 2011-10-20 Vertex Pharmaceuticals Incorporated Modulators of Cystic Fibrosis Transmembrane Conductance Regulator

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US8354427B2 (en) 2013-01-15
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RU2552353C2 (ru) 2015-06-10
BE2015C040I2 (OSRAM) 2024-10-08
US8614327B2 (en) 2013-12-24
RU2012129206A (ru) 2014-01-20
CN102652128A (zh) 2012-08-29
EP2509954A1 (en) 2012-10-17
AU2010327993A8 (en) 2012-07-19
JP2013513617A (ja) 2013-04-22
US20130165442A1 (en) 2013-06-27
IL220283A0 (en) 2012-07-31
US20100184739A1 (en) 2010-07-22
WO2011072241A1 (en) 2011-06-16
NZ600707A (en) 2014-09-26
AU2010327993A1 (en) 2012-07-12

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