CA2701868C - Bicyclic heterocyclic compounds as protein tyrosine kinase inhibitors - Google Patents

Bicyclic heterocyclic compounds as protein tyrosine kinase inhibitors Download PDF

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CA2701868C
CA2701868C CA2701868A CA2701868A CA2701868C CA 2701868 C CA2701868 C CA 2701868C CA 2701868 A CA2701868 A CA 2701868A CA 2701868 A CA2701868 A CA 2701868A CA 2701868 C CA2701868 C CA 2701868C
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CA2701868A1 (en
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Gordon Saxty
Valerio Berdini
Christopher William Murray
Charlotte Mary Griffiths-Jones
Emma Vickerstaffe
Gilbert Ebai Besong
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Astex Therapeutics Ltd
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Astex Therapeutics Ltd
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
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    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
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  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Hematology (AREA)
  • Pulmonology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
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  • Hospice & Palliative Care (AREA)
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  • Ophthalmology & Optometry (AREA)
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CA2701868A 2007-10-12 2008-10-10 Bicyclic heterocyclic compounds as protein tyrosine kinase inhibitors Active CA2701868C (en)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US97958907P 2007-10-12 2007-10-12
GBGB0720038.9A GB0720038D0 (en) 2007-10-12 2007-10-12 New compounds
GB0720038.9 2007-10-12
US60/979,589 2007-10-12
US6117208P 2008-06-13 2008-06-13
US61/061,172 2008-06-13
PCT/GB2008/003439 WO2009047522A1 (en) 2007-10-12 2008-10-10 Bicyclic heterocyclic compounds as protein tyrosine kinase inhibitors

Publications (2)

Publication Number Publication Date
CA2701868A1 CA2701868A1 (en) 2009-04-16
CA2701868C true CA2701868C (en) 2016-07-19

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Family Applications (1)

Application Number Title Priority Date Filing Date
CA2701868A Active CA2701868C (en) 2007-10-12 2008-10-10 Bicyclic heterocyclic compounds as protein tyrosine kinase inhibitors

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US (2) US8071614B2 (cg-RX-API-DMAC10.html)
EP (1) EP2203449B1 (cg-RX-API-DMAC10.html)
JP (1) JP5562858B2 (cg-RX-API-DMAC10.html)
AU (1) AU2008309342C1 (cg-RX-API-DMAC10.html)
CA (1) CA2701868C (cg-RX-API-DMAC10.html)
CY (1) CY1117820T1 (cg-RX-API-DMAC10.html)
ES (1) ES2585352T3 (cg-RX-API-DMAC10.html)
GB (1) GB0720038D0 (cg-RX-API-DMAC10.html)
HR (1) HRP20160852T1 (cg-RX-API-DMAC10.html)
HU (1) HUE028999T2 (cg-RX-API-DMAC10.html)
ME (1) ME02815B (cg-RX-API-DMAC10.html)
PL (1) PL2203449T3 (cg-RX-API-DMAC10.html)
PT (1) PT2203449T (cg-RX-API-DMAC10.html)
RS (1) RS55045B1 (cg-RX-API-DMAC10.html)
SI (1) SI2203449T1 (cg-RX-API-DMAC10.html)
WO (1) WO2009047522A1 (cg-RX-API-DMAC10.html)

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