CA2623032A1 - Deazapurines useful as inhibitors of janus kinases - Google Patents
Deazapurines useful as inhibitors of janus kinases Download PDFInfo
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- CA2623032A1 CA2623032A1 CA002623032A CA2623032A CA2623032A1 CA 2623032 A1 CA2623032 A1 CA 2623032A1 CA 002623032 A CA002623032 A CA 002623032A CA 2623032 A CA2623032 A CA 2623032A CA 2623032 A1 CA2623032 A1 CA 2623032A1
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Classifications
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
Landscapes
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Applications Claiming Priority (3)
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| US72256105P | 2005-09-30 | 2005-09-30 | |
| US60/722,561 | 2005-09-30 | ||
| PCT/US2006/037593 WO2007041130A2 (en) | 2005-09-30 | 2006-09-28 | Deazapurines useful as inhibitors of janus kinases |
Publications (1)
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| CA2623032A1 true CA2623032A1 (en) | 2007-04-12 |
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| CA002623032A Abandoned CA2623032A1 (en) | 2005-09-30 | 2006-09-28 | Deazapurines useful as inhibitors of janus kinases |
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| IL (1) | IL190249A0 (enExample) |
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| NZ (1) | NZ567133A (enExample) |
| RU (1) | RU2008117151A (enExample) |
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| WO (1) | WO2007041130A2 (enExample) |
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| PT1730146E (pt) | 2004-03-30 | 2011-07-11 | Vertex Pharma | Azaindoles úteis como inibidores de jak e outras proteínas quinases |
| EP1881983B1 (en) * | 2005-05-20 | 2012-01-11 | Vertex Pharmaceuticals, Inc. | Pyrrolopyridines useful as inhibitors of protein kinase |
| CA2621261C (en) | 2005-09-22 | 2014-05-20 | Incyte Corporation | Azepine inhibitors of janus kinases |
| DK3184526T3 (en) | 2005-12-13 | 2019-01-14 | Incyte Holdings Corp | PYRROLO [2,3-D] PYRIMIDINE DERIVATIVES AS A JANUS-KINASE INHIBITOR |
| TW201307354A (zh) | 2005-12-29 | 2013-02-16 | Abbott Lab | 蛋白質激酶抑制劑 |
| NZ601687A (en) | 2006-01-17 | 2014-03-28 | Vertex Pharma | Azaindoles useful as inhibitors of janus kinases |
| KR20090018895A (ko) * | 2006-04-05 | 2009-02-24 | 버텍스 파마슈티칼스 인코포레이티드 | 야누스 키나제의 억제제로서 유용한 데아자푸린 |
| MX2009002046A (es) | 2006-08-24 | 2009-03-06 | Astrazeneca Ab | Derivados de morfolino pirimidina utiles en el tratamiento de trastornos proliferativos. |
| CA2673472A1 (en) | 2006-12-21 | 2008-07-03 | Vertex Pharmaceuticals Incorporated | 5-cyan0-4- (pyrrolo) [2, 3b] pyridine-3-yl) -pyrimidine derivatives useful as protein kinase inhibitors |
| EP2121692B1 (en) | 2006-12-22 | 2013-04-10 | Incyte Corporation | Substituted heterocycles as janus kinase inhibitors |
| MX2009010127A (es) * | 2007-03-22 | 2009-11-05 | Vertex Pharma | Compuestos utiles como inhibidores de janus cinasas. |
| CL2008001709A1 (es) | 2007-06-13 | 2008-11-03 | Incyte Corp | Compuestos derivados de pirrolo [2,3-b]pirimidina, moduladores de quinasas jak; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como cancer, psoriasis, artritis reumatoide, entre otras. |
| DK2740731T3 (en) | 2007-06-13 | 2016-04-11 | Incyte Holdings Corp | CRYSTALLINE SALTS OF JANUSKINASEINHIBITOREN (R) -3- (4- (7H-pyrrolo [2,3-d] pyrimidin-4-yl) -1H-pyrazol-1-yl) -3-CYCLOPENTYLPROPANNITRIL |
| ATE554075T1 (de) | 2007-07-09 | 2012-05-15 | Astrazeneca Ab | Bei mit mtor-kinase und/oder pi3k in zusammenhang stehenden krankheiten angewendete morpholinopyrimidinderivate |
| CN101932583A (zh) * | 2007-12-19 | 2010-12-29 | 沃泰克斯药物股份有限公司 | 用作JAK2抑制剂的吡唑并[1,5-a]嘧啶类 |
| DE102008005493A1 (de) * | 2008-01-22 | 2009-07-23 | Merck Patent Gmbh | 4-(Pyrrolo[2,3-c] pyridine-3-yl)-pyrimidin-2-yl-amin-derivate |
| BRPI0909040B8 (pt) | 2008-03-11 | 2021-05-25 | Incyte Holdings Corp | derivados de azetidina e ciclobutano, seus usos, e composição |
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- 2006-09-28 SG SG200902181-7A patent/SG151327A1/en unknown
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- 2006-09-28 EP EP06815526A patent/EP1931674B1/en active Active
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| EP1931674A2 (en) | 2008-06-18 |
| RU2008117151A (ru) | 2009-11-10 |
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| KR20080063809A (ko) | 2008-07-07 |
| AU2006297351A1 (en) | 2007-04-12 |
| ZA200802685B (en) | 2009-10-28 |
| US8580802B2 (en) | 2013-11-12 |
| IL190249A0 (en) | 2008-11-03 |
| EP1931674B1 (en) | 2012-12-12 |
| SG151327A1 (en) | 2009-04-30 |
| NO20082026L (no) | 2008-06-25 |
| JP2009513571A (ja) | 2009-04-02 |
| ES2401192T3 (es) | 2013-04-17 |
| WO2007041130A2 (en) | 2007-04-12 |
| ES2401192T8 (es) | 2013-05-10 |
| CN101801971A (zh) | 2010-08-11 |
| US20070207995A1 (en) | 2007-09-06 |
| WO2007041130A3 (en) | 2010-01-21 |
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