CA2127274A1 - Process for preparing 3-acylestratrienes and acylbenzenes - Google Patents

Process for preparing 3-acylestratrienes and acylbenzenes

Info

Publication number
CA2127274A1
CA2127274A1 CA002127274A CA2127274A CA2127274A1 CA 2127274 A1 CA2127274 A1 CA 2127274A1 CA 002127274 A CA002127274 A CA 002127274A CA 2127274 A CA2127274 A CA 2127274A CA 2127274 A1 CA2127274 A1 CA 2127274A1
Authority
CA
Canada
Prior art keywords
compound
benzo
formula
reaction
triene
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002127274A
Other languages
English (en)
French (fr)
Inventor
Neil Howard Baine
Michael A. Mcguire
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Corp
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2127274A1 publication Critical patent/CA2127274A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • HELECTRICITY
    • H10SEMICONDUCTOR DEVICES; ELECTRIC SOLID-STATE DEVICES NOT OTHERWISE PROVIDED FOR
    • H10NELECTRIC SOLID-STATE DEVICES NOT OTHERWISE PROVIDED FOR
    • H10N30/00Piezoelectric or electrostrictive devices
    • H10N30/20Piezoelectric or electrostrictive devices with electrical input and mechanical output, e.g. functioning as actuators or vibrators
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J51/00Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C51/00Preparation of carboxylic acids or their salts, halides or anhydrides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J3/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C07J3/005Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J31/00Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0072Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the A ring of the steroid being aromatic
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0094Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 containing nitrile radicals, including thiocyanide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Toxicology (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
CA002127274A 1992-01-06 1993-01-06 Process for preparing 3-acylestratrienes and acylbenzenes Abandoned CA2127274A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US81718092A 1992-01-06 1992-01-06
US07/817,180 1992-01-06
PCT/US1993/000078 WO1993014107A1 (en) 1992-01-06 1993-01-06 Process for preparing 3-acylestratrienes and acylbenzenes

Publications (1)

Publication Number Publication Date
CA2127274A1 true CA2127274A1 (en) 1993-07-22

Family

ID=25222515

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002127274A Abandoned CA2127274A1 (en) 1992-01-06 1993-01-06 Process for preparing 3-acylestratrienes and acylbenzenes

Country Status (21)

Country Link
EP (1) EP0621866A4 (fi)
JP (1) JPH07503008A (fi)
KR (1) KR940704064A (fi)
CN (1) CN1077200A (fi)
AP (1) AP361A (fi)
AU (1) AU3434793A (fi)
BG (1) BG98888A (fi)
BR (1) BR9305707A (fi)
CA (1) CA2127274A1 (fi)
FI (1) FI943213A (fi)
HU (1) HUT67566A (fi)
IL (1) IL104303A0 (fi)
MA (1) MA22762A1 (fi)
MX (1) MX9300026A (fi)
NO (1) NO942531D0 (fi)
OA (1) OA09959A (fi)
RU (1) RU94037761A (fi)
SI (1) SI9300005A (fi)
SK (1) SK80194A3 (fi)
WO (1) WO1993014107A1 (fi)
ZA (1) ZA938B (fi)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SK129294A3 (en) * 1992-04-30 1995-07-11 Smithkline Beecham Corp 17-alpha and 17-beta-substituted estra-1,3,5(10)-triene-3- -carboxylic acid
GB9411103D0 (en) * 1994-06-03 1994-07-27 Smithkline Beecham Corp Compounds
GB9608045D0 (en) * 1996-04-18 1996-06-19 Pharmacia Spa Process for preparing steroids having a carboxamide side-chain
JP2000309599A (ja) 1999-04-13 2000-11-07 Kyowa Hakko Kogyo Co Ltd エストラ−1,3,5(10),16−テトラエン誘導体
JP5793996B2 (ja) * 2011-06-29 2015-10-14 セントラル硝子株式会社 フルオロ硫酸芳香環エステル類の製造方法
US10117840B2 (en) * 2014-06-06 2018-11-06 The Scripps Research Institute Sulfur(VI) fluoride compounds and methods for the preparation thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4954446A (en) * 1988-05-25 1990-09-04 Smithkline Beecham Corporation Aromatic steroid 5-α-reductase inhibitors
US4970205A (en) * 1988-12-23 1990-11-13 Smithkline Beecham Corporation Sulfonic acid substituted aromatic steroids as inhibitors of steroid 5-α-reductase
US4937237A (en) * 1988-12-23 1990-06-26 Smithkline Beckman Corporation Phosphinic acid substituted aromatic steroids as inhibitors of steroid 5-60 -reductase

Also Published As

Publication number Publication date
FI943213A0 (fi) 1994-07-05
CN1077200A (zh) 1993-10-13
SI9300005A (en) 1993-09-30
SK80194A3 (en) 1994-12-07
FI943213A (fi) 1994-07-05
BR9305707A (pt) 1996-12-31
AU3434793A (en) 1993-08-03
OA09959A (en) 1995-12-11
KR940704064A (ko) 1994-12-12
AP361A (en) 1994-09-09
BG98888A (en) 1995-05-31
JPH07503008A (ja) 1995-03-30
MX9300026A (es) 1993-12-01
RU94037761A (ru) 1997-05-27
WO1993014107A1 (en) 1993-07-22
EP0621866A1 (en) 1994-11-02
HU9402029D0 (en) 1994-09-28
EP0621866A4 (en) 1996-03-20
MA22762A1 (fr) 1993-10-01
AP9300474A0 (en) 1993-01-31
IL104303A0 (en) 1993-05-13
NO942531L (no) 1994-07-05
NO942531D0 (no) 1994-07-05
ZA938B (en) 1994-06-16
HUT67566A (en) 1995-04-28

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Legal Events

Date Code Title Description
FZDE Discontinued