AP361A - Process for the preparation of substituted steroidal benzo esters and acids. - Google Patents

Process for the preparation of substituted steroidal benzo esters and acids. Download PDF

Info

Publication number
AP361A
AP361A APAP/P/1993/000474A AP9300474A AP361A AP 361 A AP361 A AP 361A AP 9300474 A AP9300474 A AP 9300474A AP 361 A AP361 A AP 361A
Authority
AP
ARIPO
Prior art keywords
compound
benzo
formula
reaction
steroidal
Prior art date
Application number
APAP/P/1993/000474A
Other languages
English (en)
Other versions
AP9300474A0 (en
Inventor
Neil Howard Baine
Michael Maguire
Original Assignee
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp
Publication of AP9300474A0 publication Critical patent/AP9300474A0/xx
Application granted granted Critical
Publication of AP361A publication Critical patent/AP361A/en

Links

Classifications

    • H—ELECTRICITY
    • H10—SEMICONDUCTOR DEVICES; ELECTRIC SOLID-STATE DEVICES NOT OTHERWISE PROVIDED FOR
    • H10N—ELECTRIC SOLID-STATE DEVICES NOT OTHERWISE PROVIDED FOR
    • H10N30/00—Piezoelectric or electrostrictive devices
    • H10N30/20—Piezoelectric or electrostrictive devices with electrical input and mechanical output, e.g. functioning as actuators or vibrators
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C07J3/005—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0072—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the A ring of the steroid being aromatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0094—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 containing nitrile radicals, including thiocyanide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Toxicology (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
APAP/P/1993/000474A 1992-01-06 1993-01-05 Process for the preparation of substituted steroidal benzo esters and acids. AP361A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US81718092A 1992-01-06 1992-01-06

Publications (2)

Publication Number Publication Date
AP9300474A0 AP9300474A0 (en) 1993-01-31
AP361A true AP361A (en) 1994-09-09

Family

ID=25222515

Family Applications (1)

Application Number Title Priority Date Filing Date
APAP/P/1993/000474A AP361A (en) 1992-01-06 1993-01-05 Process for the preparation of substituted steroidal benzo esters and acids.

Country Status (21)

Country Link
EP (1) EP0621866A4 (fi)
JP (1) JPH07503008A (fi)
KR (1) KR940704064A (fi)
CN (1) CN1077200A (fi)
AP (1) AP361A (fi)
AU (1) AU3434793A (fi)
BG (1) BG98888A (fi)
BR (1) BR9305707A (fi)
CA (1) CA2127274A1 (fi)
FI (1) FI943213A (fi)
HU (1) HUT67566A (fi)
IL (1) IL104303A0 (fi)
MA (1) MA22762A1 (fi)
MX (1) MX9300026A (fi)
NO (1) NO942531L (fi)
OA (1) OA09959A (fi)
RU (1) RU94037761A (fi)
SI (1) SI9300005A (fi)
SK (1) SK80194A3 (fi)
WO (1) WO1993014107A1 (fi)
ZA (1) ZA938B (fi)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ252866A (en) * 1992-04-30 1996-09-25 Smithkline Beecham Corp 17-acyl-estra-1,3,5(10)-triene-3-carboxylic acids; precursors
GB9411103D0 (en) * 1994-06-03 1994-07-27 Smithkline Beecham Corp Compounds
GB9608045D0 (en) * 1996-04-18 1996-06-19 Pharmacia Spa Process for preparing steroids having a carboxamide side-chain
JP2000309599A (ja) 1999-04-13 2000-11-07 Kyowa Hakko Kogyo Co Ltd エストラ−１，３，５（１０），１６−テトラエン誘導体
JP5793996B2 (ja) * 2011-06-29 2015-10-14 セントラル硝子株式会社 フルオロ硫酸芳香環エステル類の製造方法
ES2873962T3 (es) 2014-06-06 2021-11-04 Scripps Research Inst Compuestos de fluoruro de azufre (VI) y métodos para la preparación de los mismos

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4937237A (en) * 1988-12-23 1990-06-26 Smithkline Beckman Corporation Phosphinic acid substituted aromatic steroids as inhibitors of steroid 5-60 -reductase
US4954446A (en) * 1988-05-25 1990-09-04 Smithkline Beecham Corporation Aromatic steroid 5-α-reductase inhibitors

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4970205A (en) * 1988-12-23 1990-11-13 Smithkline Beecham Corporation Sulfonic acid substituted aromatic steroids as inhibitors of steroid 5-α-reductase

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4954446A (en) * 1988-05-25 1990-09-04 Smithkline Beecham Corporation Aromatic steroid 5-α-reductase inhibitors
US4937237A (en) * 1988-12-23 1990-06-26 Smithkline Beckman Corporation Phosphinic acid substituted aromatic steroids as inhibitors of steroid 5-60 -reductase

Also Published As

Publication number Publication date
RU94037761A (ru) 1997-05-27
WO1993014107A1 (en) 1993-07-22
NO942531D0 (no) 1994-07-05
SK80194A3 (en) 1994-12-07
MA22762A1 (fr) 1993-10-01
AU3434793A (en) 1993-08-03
FI943213A0 (fi) 1994-07-05
HU9402029D0 (en) 1994-09-28
NO942531L (no) 1994-07-05
JPH07503008A (ja) 1995-03-30
KR940704064A (ko) 1994-12-12
BG98888A (en) 1995-05-31
EP0621866A4 (en) 1996-03-20
EP0621866A1 (en) 1994-11-02
MX9300026A (es) 1993-12-01
SI9300005A (en) 1993-09-30
CN1077200A (zh) 1993-10-13
CA2127274A1 (en) 1993-07-22
ZA938B (en) 1994-06-16
AP9300474A0 (en) 1993-01-31
IL104303A0 (en) 1993-05-13
HUT67566A (en) 1995-04-28
BR9305707A (pt) 1996-12-31
OA09959A (en) 1995-12-11
FI943213A (fi) 1994-07-05

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