BRPI0908208A2 - Composto derivado de oxazolidinona, medicamento, composição farmacêutica que o contém e uso desse composto. - Google Patents
Composto derivado de oxazolidinona, medicamento, composição farmacêutica que o contém e uso desse composto.Info
- Publication number
- BRPI0908208A2 BRPI0908208A2 BRPI0908208-5A BRPI0908208A BRPI0908208A2 BR PI0908208 A2 BRPI0908208 A2 BR PI0908208A2 BR PI0908208 A BRPI0908208 A BR PI0908208A BR PI0908208 A2 BRPI0908208 A2 BR PI0908208A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- drug
- pharmaceutical composition
- composition containing
- oxazolidinone derivative
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IB2008050651 | 2008-02-22 | ||
IB2008054095 | 2008-10-07 | ||
PCT/IB2009/050702 WO2009104159A1 (en) | 2008-02-22 | 2009-02-20 | Oxazolidinone derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0908208A2 true BRPI0908208A2 (pt) | 2015-08-25 |
Family
ID=40578768
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0908208-5A BRPI0908208A2 (pt) | 2008-02-22 | 2009-02-20 | Composto derivado de oxazolidinona, medicamento, composição farmacêutica que o contém e uso desse composto. |
Country Status (14)
Country | Link |
---|---|
US (1) | US8349826B2 (pt) |
EP (1) | EP2254887B9 (pt) |
JP (1) | JP5404652B2 (pt) |
KR (1) | KR101592046B1 (pt) |
CN (1) | CN102015698B (pt) |
AR (1) | AR070458A1 (pt) |
BR (1) | BRPI0908208A2 (pt) |
CA (1) | CA2713187C (pt) |
ES (1) | ES2398939T3 (pt) |
MX (1) | MX2010008921A (pt) |
PL (1) | PL2254887T3 (pt) |
RU (1) | RU2501799C2 (pt) |
TW (1) | TWI429643B (pt) |
WO (1) | WO2009104159A1 (pt) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
RU2010138648A (ru) | 2008-02-20 | 2012-03-27 | Актелион Фармасьютиклз Лтд (Ch) | Азатрициклические соединения антибиотиков |
WO2010041194A1 (en) | 2008-10-07 | 2010-04-15 | Actelion Pharmaceuticals Ltd | Tricyclic oxazolidinone antibiotic compounds |
WO2010041219A1 (en) * | 2008-10-10 | 2010-04-15 | Actelion Pharmaceuticals Ltd | 2-benzothiophenyl-and 2-naphthyl-0xaz0lidin0nes and their azaisostere analogues as antibacterial agents |
MX2011003188A (es) * | 2008-10-10 | 2011-04-27 | Actelion Pharmaceuticals Ltd | Antibioticos de oxazolidinilo. |
AR076222A1 (es) | 2009-04-09 | 2011-05-26 | Actelion Pharmaceuticals Ltd | Derivados 2-hidroxietil-1h-quinolin-ona y sus analogos azaisotericos con actividad antibacteriana y composiciones farmaceuticas que los contienen |
EP2674430A4 (en) | 2011-02-07 | 2014-07-02 | Daiichi Sankyo Co Ltd | AMINO-GROUP-PYRROLIDINONE DERIVATIVES |
KR20140054057A (ko) * | 2011-08-11 | 2014-05-08 | 액테리온 파마슈티칼 리미티드 | 퀴나졸린-2,4-디온 유도체 |
RU2616609C2 (ru) * | 2011-11-08 | 2017-04-18 | Актелион Фармасьютиклз Лтд | Антибиотические производные 2-оксо-оксазолидин-3, 5-диила |
CN103958525A (zh) | 2011-11-30 | 2014-07-30 | 埃科特莱茵药品有限公司 | 3,7-二取代八氢-2H-吡啶并[4,3-e][1,3]噁嗪-2-酮抗生素 |
WO2014024056A1 (en) | 2012-08-06 | 2014-02-13 | Daiichi Sankyo Company, Limited | Pyrrolidine derivatives with antibacterial properties |
EP2943492A1 (en) | 2013-01-09 | 2015-11-18 | Actelion Pharmaceuticals Ltd. | Antibacterial oxadiazolone derivatives |
CA2907832A1 (en) | 2013-04-16 | 2014-10-23 | Actelion Pharmaceuticals Ltd | Antibacterial biaromatic derivatives |
CA2910177A1 (en) | 2013-05-08 | 2014-11-13 | Actelion Pharmaceuticals Ltd | Antibacterial phthalide derivatives |
AR102256A1 (es) | 2014-10-15 | 2017-02-15 | Actelion Pharmaceuticals Ltd | Derivados biaromáticos básicos antibacterianos con sustitución de aminoalcoxi |
SG11201806166WA (en) | 2016-02-08 | 2018-08-30 | Redx Pharma Plc | Heterocyclic compounds, in particular 2-oxo-4,4,5,5,6,6,7,7-octahydrobenzoxazole derivatives, and their use as antibacterial compounds |
US20210179636A1 (en) * | 2016-02-08 | 2021-06-17 | Redx Pharma Plc | Antibacterial compounds |
GB201602235D0 (en) * | 2016-02-08 | 2016-03-23 | Redx Pharma Plc | Antibacterial compounds |
TW201833120A (zh) | 2017-02-17 | 2018-09-16 | 瑞士商愛杜西亞製藥有限公司 | 芳基噁唑啶酮抗生素化合物 |
JP7148991B2 (ja) * | 2017-06-08 | 2022-10-06 | バグワークス・リサーチ・インコーポレイテッド | 抗菌剤として有用な複素環式化合物及びその生成方法 |
US11401277B2 (en) | 2017-11-29 | 2022-08-02 | Bugworks Research, Inc. | Anti-bacterial heterocyclic compounds and their synthesis |
ES2942552T3 (es) * | 2018-03-28 | 2023-06-02 | Bugworks Res Inc | Compuestos antibióticos de oxazolidinona y procedimiento de preparación |
Family Cites Families (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB2168696B (en) | 1984-12-21 | 1989-01-11 | Boehringer Biochemia Srl | Fluoro coumarins as antilymphoedema agents |
CA2012681A1 (en) * | 1989-03-31 | 1990-09-30 | Masayasu Okuhira | Quinolone derivatives, preparation processes thereof, and antibacterial agents containing the same |
DE19514313A1 (de) * | 1994-08-03 | 1996-02-08 | Bayer Ag | Benzoxazolyl- und Benzothiazolyloxazolidinone |
DE19601265A1 (de) * | 1996-01-16 | 1997-07-17 | Bayer Ag | 2-Oxo- und 2-Thio-1,2-dihydrochinolinyl-oxazolidinone |
CN1163892A (zh) * | 1996-01-16 | 1997-11-05 | 拜尔公司 | 2-氧代-和2-硫代-1,2-二氢喹啉基-噁唑烷酮类化合物 |
DE19604223A1 (de) * | 1996-02-06 | 1997-08-07 | Bayer Ag | Neue substituierte Oxazolidinone |
WO2001030782A2 (en) | 1999-10-29 | 2001-05-03 | Syngenta Participations Ag | Novel herbicides |
GB0031086D0 (en) | 2000-12-20 | 2001-01-31 | Smithkline Beecham Plc | Medicaments |
GB0101577D0 (en) | 2001-01-22 | 2001-03-07 | Smithkline Beecham Plc | Compounds |
GB0112834D0 (en) | 2001-05-25 | 2001-07-18 | Smithkline Beecham Plc | Medicaments |
FR2852954B1 (fr) | 2003-03-28 | 2006-07-14 | Aventis Pharma Sa | Derives de quinoleines-4-substituees, leurs procede et intermediaires de preparation et les compositions pharmaceutiques qui les contiennent |
WO2006024741A2 (fr) * | 2004-07-30 | 2006-03-09 | Palumed S.A. | Molecules hybrides qa ou q est une aminoquinoleine et a est un residu antibiotique, leur synthese et leurs utilisations en tant qu'agent antibacterien |
TWI320783B (en) | 2005-04-14 | 2010-02-21 | Otsuka Pharma Co Ltd | Heterocyclic compound |
MY150958A (en) | 2005-06-16 | 2014-03-31 | Astrazeneca Ab | Compounds for the treatment of multi-drug resistant bacterial infections |
EP1963324B1 (en) | 2005-12-22 | 2010-04-21 | Glaxo Group Limited | Heterocyclic compounds, their preparation and their use as antibacterials |
WO2007093904A1 (en) * | 2006-02-14 | 2007-08-23 | Pfizer Products Inc. | Benzoxazinone and benzoxazepinone oxazolidinones as antibacterial agents |
ES2476423T3 (es) | 2006-05-26 | 2014-07-14 | Toyama Chemical Co., Ltd. | Nuevo compuesto heteroc�clico o sal del mismo e intermedio del mismo |
RU2444519C2 (ru) | 2006-06-16 | 2012-03-10 | Фарма Мар, С.А. | Противоопухолевые соединения дигидропиран-2-она |
US7977352B2 (en) | 2006-12-01 | 2011-07-12 | Galapagos Nv | Triazolopyridine compounds useful for the treatment of degenerative and inflammatory diseases |
CL2008001003A1 (es) | 2007-04-11 | 2008-10-17 | Actelion Pharmaceuticals Ltd | Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana. |
CL2008001002A1 (es) | 2007-04-11 | 2008-10-17 | Actelion Pharmaceuticals Ltd | Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana. |
-
2009
- 2009-02-20 KR KR1020107020126A patent/KR101592046B1/ko active IP Right Grant
- 2009-02-20 WO PCT/IB2009/050702 patent/WO2009104159A1/en active Application Filing
- 2009-02-20 CN CN200980106053.9A patent/CN102015698B/zh not_active Expired - Fee Related
- 2009-02-20 RU RU2010138840/04A patent/RU2501799C2/ru not_active IP Right Cessation
- 2009-02-20 TW TW098105507A patent/TWI429643B/zh not_active IP Right Cessation
- 2009-02-20 EP EP09711588.5A patent/EP2254887B9/en not_active Not-in-force
- 2009-02-20 CA CA2713187A patent/CA2713187C/en not_active Expired - Fee Related
- 2009-02-20 MX MX2010008921A patent/MX2010008921A/es active IP Right Grant
- 2009-02-20 BR BRPI0908208-5A patent/BRPI0908208A2/pt not_active IP Right Cessation
- 2009-02-20 AR ARP090100598A patent/AR070458A1/es unknown
- 2009-02-20 US US12/918,779 patent/US8349826B2/en not_active Expired - Fee Related
- 2009-02-20 PL PL09711588T patent/PL2254887T3/pl unknown
- 2009-02-20 ES ES09711588T patent/ES2398939T3/es active Active
- 2009-02-20 JP JP2010547295A patent/JP5404652B2/ja not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
US8349826B2 (en) | 2013-01-08 |
JP5404652B2 (ja) | 2014-02-05 |
CN102015698A (zh) | 2011-04-13 |
KR101592046B1 (ko) | 2016-02-05 |
RU2501799C2 (ru) | 2013-12-20 |
ES2398939T9 (es) | 2013-07-24 |
AR070458A1 (es) | 2010-04-07 |
CA2713187C (en) | 2016-06-07 |
TWI429643B (zh) | 2014-03-11 |
ES2398939T3 (es) | 2013-03-22 |
CA2713187A1 (en) | 2009-08-27 |
CN102015698B (zh) | 2014-08-27 |
AU2009215247A1 (en) | 2009-08-27 |
JP2011512401A (ja) | 2011-04-21 |
KR20100124282A (ko) | 2010-11-26 |
EP2254887B1 (en) | 2012-12-19 |
EP2254887A1 (en) | 2010-12-01 |
WO2009104159A1 (en) | 2009-08-27 |
MX2010008921A (es) | 2010-09-07 |
TW200940534A (en) | 2009-10-01 |
RU2010138840A (ru) | 2012-03-27 |
US20100331308A1 (en) | 2010-12-30 |
EP2254887B9 (en) | 2013-05-29 |
PL2254887T3 (pl) | 2013-05-31 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 8A ANUIDADE. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |