BRPI0907052A2 - Processo para a preparação de compostos - Google Patents

Processo para a preparação de compostos

Info

Publication number
BRPI0907052A2
BRPI0907052A2 BRPI0907052-4A BRPI0907052A BRPI0907052A2 BR PI0907052 A2 BRPI0907052 A2 BR PI0907052A2 BR PI0907052 A BRPI0907052 A BR PI0907052A BR PI0907052 A2 BRPI0907052 A2 BR PI0907052A2
Authority
BR
Brazil
Prior art keywords
compounds
preparation
Prior art date
Application number
BRPI0907052-4A
Other languages
English (en)
Inventor
Matthias Helmreich
Mike Brandner
Original Assignee
Poxel Sas
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Poxel Sas filed Critical Poxel Sas
Publication of BRPI0907052A2 publication Critical patent/BRPI0907052A2/pt
Publication of BRPI0907052B1 publication Critical patent/BRPI0907052B1/pt
Publication of BRPI0907052B8 publication Critical patent/BRPI0907052B8/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D251/00Heterocyclic compounds containing 1,3,5-triazine rings
    • C07D251/02Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings
    • C07D251/10Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
BRPI0907052A 2008-02-02 2009-01-15 processo para a preparação de compostos BRPI0907052B8 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE102008007314A DE102008007314A1 (de) 2008-02-02 2008-02-02 Verfahren zur Herstellung von 3,6-Dihydro-1,3,5-triazinderivaten
DE102008007314.8 2008-02-02
PCT/EP2009/000212 WO2009095159A1 (de) 2008-02-02 2009-01-15 Verfahren zur herstellung von 3, 6-dihydro-l, 3, 5-triazinderivaten aus metformin- und paraldehydderivaten

Publications (3)

Publication Number Publication Date
BRPI0907052A2 true BRPI0907052A2 (pt) 2015-07-07
BRPI0907052B1 BRPI0907052B1 (pt) 2020-09-24
BRPI0907052B8 BRPI0907052B8 (pt) 2021-05-25

Family

ID=40459622

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0907052A BRPI0907052B8 (pt) 2008-02-02 2009-01-15 processo para a preparação de compostos

Country Status (24)

Country Link
US (1) US8461331B2 (pt)
EP (1) EP2240456B1 (pt)
JP (1) JP5542066B2 (pt)
KR (1) KR101553568B1 (pt)
CN (1) CN101932566B (pt)
AR (1) AR070329A1 (pt)
AT (1) ATE519752T1 (pt)
AU (1) AU2009210293B2 (pt)
BR (1) BRPI0907052B8 (pt)
CA (1) CA2713236C (pt)
CY (1) CY1111837T1 (pt)
DE (1) DE102008007314A1 (pt)
DK (1) DK2240456T3 (pt)
EA (1) EA017062B1 (pt)
ES (1) ES2368116T3 (pt)
HR (1) HRP20110644T1 (pt)
IL (1) IL206816A (pt)
MX (1) MX2010008282A (pt)
PL (1) PL2240456T3 (pt)
PT (1) PT2240456E (pt)
RS (1) RS51968B (pt)
SI (1) SI2240456T1 (pt)
WO (1) WO2009095159A1 (pt)
ZA (1) ZA201006211B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2816357C (en) 2010-12-01 2015-04-28 Poxel Separation of triazine derivatives enantiomers using tartaric acid
MX2020003243A (es) 2017-10-02 2020-09-18 Poxel Métodos para tratar la insuficiencia cardíaca con fracción de eyección preservada.
ES2929994T3 (es) 2018-06-06 2022-12-05 Poxel Sa Métodos de tratamiento de sujetos que padecen diabetes con enfermedad renal crónica
MX2020013567A (es) 2018-06-14 2021-05-27 Poxel Tableta recubierta con pelicula que comprende un derivado de triazina para su uso en el tratamiento de la diabetes.
CN109655544B (zh) * 2018-12-25 2022-08-12 广东华南药业集团有限公司 一种盐酸二甲双胍及其制剂的质量控制方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1537604A (fr) 1966-09-26 1968-08-23 Sandoz Sa Procédé de préparation de biguanides
GB1250531A (pt) * 1969-01-01 1971-10-20
DE2117015A1 (de) 1971-04-02 1972-10-26 Schering Ag 1,2-Biguanide
SU458538A1 (ru) * 1973-06-14 1975-01-30 Уфимский Нефтяной Институт Способ совместного получени 1,3диеновых углеводородов и гексаметилентетрамина
JPH061779A (ja) * 1992-02-06 1994-01-11 Wakamoto Pharmaceut Co Ltd ベンズオキサジノン誘導体
US5767294A (en) * 1993-02-17 1998-06-16 Hoechst Celanese Corporation Process for the production of trioxane from formaldehyde
US5627282A (en) * 1996-01-03 1997-05-06 Yukong Limited Process for the preparation of optically pure 1,2,3,4-tetrahydro-3-isoquinolinecarboxylic acid and its derivatives
FR2804113B1 (fr) * 2000-01-26 2004-06-18 Lipha Derives animes de dihydro-1,3,5-triazine et leurs applications en therapeutique
CN100551916C (zh) * 2002-12-17 2009-10-21 浜理药品工业株式会社 新的2,4-二氨基-1,3,5-三嗪衍生物
KR101027366B1 (ko) 2002-12-17 2011-04-11 하마리야꾸힝고오교가부시끼가이샤 신규한 2,4-디아미노-1,3,5-트리아진 유도체
FR2853650B1 (fr) * 2003-04-10 2006-07-07 Merck Sante Sas Procede de dedoublement d'amines utiles pour le traitement de desordres associes au syndrome d'insulino-resistance
TWI410413B (zh) * 2006-04-26 2013-10-01 Sumitomo Seika Chemicals Preparation method of methylene disulfonate compound

Also Published As

Publication number Publication date
EA017062B1 (ru) 2012-09-28
US8461331B2 (en) 2013-06-11
HRP20110644T1 (hr) 2011-10-31
KR101553568B1 (ko) 2015-09-16
ATE519752T1 (de) 2011-08-15
RS51968B (en) 2012-02-29
SI2240456T1 (sl) 2012-01-31
MX2010008282A (es) 2010-11-30
EP2240456B1 (de) 2011-08-10
CN101932566A (zh) 2010-12-29
KR20100103698A (ko) 2010-09-27
JP5542066B2 (ja) 2014-07-09
CA2713236A1 (en) 2009-08-06
IL206816A (en) 2013-02-28
PL2240456T3 (pl) 2011-11-30
AU2009210293A1 (en) 2009-08-06
IL206816A0 (en) 2010-12-30
PT2240456E (pt) 2011-09-27
JP2011510940A (ja) 2011-04-07
DE102008007314A1 (de) 2009-08-06
WO2009095159A1 (de) 2009-08-06
CN101932566B (zh) 2013-04-10
US20110118463A1 (en) 2011-05-19
AR070329A1 (es) 2010-03-31
DK2240456T3 (da) 2011-09-26
EP2240456A1 (de) 2010-10-20
ZA201006211B (en) 2011-05-25
EA201001252A1 (ru) 2010-12-30
BRPI0907052B1 (pt) 2020-09-24
BRPI0907052B8 (pt) 2021-05-25
ES2368116T3 (es) 2011-11-14
CY1111837T1 (el) 2015-10-07
CA2713236C (en) 2016-03-22
AU2009210293B2 (en) 2013-05-23

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B06T Formal requirements before examination [chapter 6.20 patent gazette]
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]

Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.

B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 24/09/2020, OBSERVADAS AS CONDICOES LEGAIS.

B16C Correction of notification of the grant [chapter 16.3 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 15/01/2009 OBSERVADAS AS CONDICOES LEGAIS. PATENTE CONCEDIDA CONFORME ADI 5.529/DF

B21F Lapse acc. art. 78, item iv - on non-payment of the annual fees in time

Free format text: REFERENTE A 15A ANUIDADE.

B24J Lapse because of non-payment of annual fees (definitively: art 78 iv lpi, resolution 113/2013 art. 12)

Free format text: EM VIRTUDE DA EXTINCAO PUBLICADA NA RPI 2757 DE 07-11-2023 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDA A EXTINCAO DA PATENTE E SEUS CERTIFICADOS, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.