BG65239B1 - Полиморфни кристалинни форми на целекоксиб - Google Patents

Полиморфни кристалинни форми на целекоксиб Download PDF

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Publication number
BG65239B1
BG65239B1 BG105808A BG10580801A BG65239B1 BG 65239 B1 BG65239 B1 BG 65239B1 BG 105808 A BG105808 A BG 105808A BG 10580801 A BG10580801 A BG 10580801A BG 65239 B1 BG65239 B1 BG 65239B1
Authority
BG
Bulgaria
Prior art keywords
celecoxib
cyclooxygenase
compositions
celecoxib form
present
Prior art date
Application number
BG105808A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG105808A (en
Inventor
Leonard Ferro
Patricia Miyake
Original Assignee
Pharmacia Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/US2000/032760 external-priority patent/WO2001042222A1/en
Priority claimed from PCT/US2000/032434 external-priority patent/WO2001041760A2/en
Application filed by Pharmacia Corporation filed Critical Pharmacia Corporation
Publication of BG105808A publication Critical patent/BG105808A/xx
Publication of BG65239B1 publication Critical patent/BG65239B1/bg

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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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BG105808A 1999-12-08 2001-08-09 Полиморфни кристалинни форми на целекоксиб BG65239B1 (bg)

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PCT/US2000/032760 WO2001042222A1 (en) 1999-12-08 2000-12-01 Polymorphic crystalline forms of celecoxib
PCT/US2000/032434 WO2001041760A2 (en) 1999-12-08 2000-12-06 Cyclooxygenase-2 inhibitor compositions having rapid onset of therapeutic effect

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US7927613B2 (en) 2002-02-15 2011-04-19 University Of South Florida Pharmaceutical co-crystal compositions
CA2477923C (en) 2002-03-01 2021-02-23 University Of South Florida Multiple-component solid phases containing at least one active pharmaceutical ingredient
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EA014443B1 (ru) * 2004-06-29 2010-12-30 Никомед Данмарк Апс Фармацевтическая композиция (варианты) и способ ее производства
GB0423103D0 (en) * 2004-10-19 2004-11-17 Boots Healthcare Int Ltd Therapeutic agents
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CN103462920A (zh) * 2012-06-06 2013-12-25 南京亿华药业有限公司 一种口服环加氧酶-2抑制剂塞来昔布的组合物
CN103524416B (zh) * 2013-10-29 2016-08-17 湖北华世通生物医药科技有限公司 一种塞来昔布新晶型a及其制备方法
CN103508958A (zh) * 2013-10-30 2014-01-15 中美华世通生物医药科技（武汉）有限公司 一种塞来昔布新晶型c及其制备方法
CN103539739B (zh) * 2013-10-30 2016-02-10 中美华世通生物医药科技（武汉）有限公司 一种塞来昔布新晶型b及其制备方法
KR101476096B1 (ko) * 2014-03-28 2014-12-24 대원제약주식회사 용해도가 향상된 쎄레콕시브의 약제학적 조성물

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US5760068A (en) * 1993-11-30 1998-06-02 G.D. Searle & Co. Substituted pyrazolyl benzenesulfonamides for the treatment of inflammation
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AR030039A1 (es) 2003-08-13
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