AU2041201A - Solid-state form of celecoxib having enhanced bioavailability - Google Patents
Solid-state form of celecoxib having enhanced bioavailabilityInfo
- Publication number
- AU2041201A AU2041201A AU20412/01A AU2041201A AU2041201A AU 2041201 A AU2041201 A AU 2041201A AU 20412/01 A AU20412/01 A AU 20412/01A AU 2041201 A AU2041201 A AU 2041201A AU 2041201 A AU2041201 A AU 2041201A
- Authority
- AU
- Australia
- Prior art keywords
- celecoxib
- solid
- state form
- enhanced bioavailability
- bioavailability
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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- Psychiatry (AREA)
- Biophysics (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US16985699P | 1999-12-08 | 1999-12-08 | |
US60169856 | 1999-12-08 | ||
PCT/US2000/030180 WO2001041536A2 (en) | 1999-12-08 | 2000-12-04 | Solid-state form of celecoxib having enhanced bioavailability |
Publications (1)
Publication Number | Publication Date |
---|---|
AU2041201A true AU2041201A (en) | 2001-06-18 |
Family
ID=22617480
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU20412/01A Withdrawn AU2041201A (en) | 1999-12-08 | 2000-12-04 | Solid-state form of celecoxib having enhanced bioavailability |
Country Status (21)
Country | Link |
---|---|
KR (1) | KR100717570B1 (zh) |
CN (1) | CN1216869C (zh) |
AR (2) | AR027897A1 (zh) |
AU (1) | AU2041201A (zh) |
BG (1) | BG65239B1 (zh) |
CO (1) | CO5251445A1 (zh) |
CZ (1) | CZ20012875A3 (zh) |
EA (1) | EA200401397A1 (zh) |
EC (1) | ECSP003807A (zh) |
ES (1) | ES2236011T3 (zh) |
HU (1) | HUP0200580A3 (zh) |
MY (2) | MY128971A (zh) |
NZ (1) | NZ529933A (zh) |
OA (1) | OA11831A (zh) |
PE (1) | PE20010911A1 (zh) |
PT (2) | PT1150960E (zh) |
SV (1) | SV2002000235A (zh) |
TW (1) | TWI276435B (zh) |
WO (1) | WO2001041536A2 (zh) |
YU (1) | YU57801A (zh) |
ZA (2) | ZA200107146B (zh) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NZ524252A (en) * | 2000-07-20 | 2004-03-26 | Lauras As | Cox-2 inhibitors for treating HIV and AIDS |
JP2004534812A (ja) | 2001-06-22 | 2004-11-18 | ファイザー・プロダクツ・インク | 薬物および中性ポリマーの分散物の医薬組成物 |
WO2004061433A1 (en) * | 2002-12-30 | 2004-07-22 | Transform Pharmaceuticals, Inc. | Pharmaceutical compositions with improved dissolution |
US7790905B2 (en) | 2002-02-15 | 2010-09-07 | Mcneil-Ppc, Inc. | Pharmaceutical propylene glycol solvate compositions |
US7078526B2 (en) | 2002-05-31 | 2006-07-18 | Transform Pharmaceuticals, Inc. | CIS-itraconazole crystalline forms and related processes, pharmaceutical compositions and methods |
WO2004026235A2 (en) * | 2002-09-20 | 2004-04-01 | Transform Pharmaceuticals, Inc. | Pharmaceutical compositions with improved dissolution |
US7446107B2 (en) | 2002-02-15 | 2008-11-04 | Transform Pharmaceuticals, Inc. | Crystalline forms of conazoles and methods of making and using the same |
US7927613B2 (en) | 2002-02-15 | 2011-04-19 | University Of South Florida | Pharmaceutical co-crystal compositions |
CA2477923C (en) | 2002-03-01 | 2021-02-23 | University Of South Florida | Multiple-component solid phases containing at least one active pharmaceutical ingredient |
JP2006511499A (ja) * | 2002-05-13 | 2006-04-06 | ファルマシア コーポレイション | 安定な無定形セレコキシブ複合物およびその製法 |
MXPA05000232A (es) * | 2002-06-21 | 2005-06-17 | Transform Pharmaceuticals Inc | Composiciones farmaceuticas con disolucion mejorada. |
US8183290B2 (en) | 2002-12-30 | 2012-05-22 | Mcneil-Ppc, Inc. | Pharmaceutically acceptable propylene glycol solvate of naproxen |
CA2511881C (en) * | 2002-12-30 | 2013-06-25 | Transform Pharmaceuticals, Inc. | Pharmaceutical compositions comprising a sodium salt of celecoxib with improved dissolution |
EA014443B1 (ru) * | 2004-06-29 | 2010-12-30 | Никомед Данмарк Апс | Фармацевтическая композиция (варианты) и способ ее производства |
GB0423103D0 (en) * | 2004-10-19 | 2004-11-17 | Boots Healthcare Int Ltd | Therapeutic agents |
EP1865951A1 (en) * | 2005-03-14 | 2007-12-19 | Nycomed GmbH | Method for preventing cardiovascular diseases |
CN103462920A (zh) * | 2012-06-06 | 2013-12-25 | 南京亿华药业有限公司 | 一种口服环加氧酶-2抑制剂塞来昔布的组合物 |
CN103524416B (zh) * | 2013-10-29 | 2016-08-17 | 湖北华世通生物医药科技有限公司 | 一种塞来昔布新晶型a及其制备方法 |
CN103508958A (zh) * | 2013-10-30 | 2014-01-15 | 中美华世通生物医药科技(武汉)有限公司 | 一种塞来昔布新晶型c及其制备方法 |
CN103539739B (zh) * | 2013-10-30 | 2016-02-10 | 中美华世通生物医药科技(武汉)有限公司 | 一种塞来昔布新晶型b及其制备方法 |
KR101476096B1 (ko) * | 2014-03-28 | 2014-12-24 | 대원제약주식회사 | 용해도가 향상된 쎄레콕시브의 약제학적 조성물 |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5474995A (en) * | 1993-06-24 | 1995-12-12 | Merck Frosst Canada, Inc. | Phenyl heterocycles as cox-2 inhibitors |
DK0924201T3 (da) * | 1993-11-30 | 2002-05-21 | Searle & Co | Tricyclisk substitueret pyrazolylbenzensulfonamider og deres anvendelse som cyclooxygenase II-inhibitorer |
US5633272A (en) * | 1995-02-13 | 1997-05-27 | Talley; John J. | Substituted isoxazoles for the treatment of inflammation |
CN1107058C (zh) * | 1995-02-13 | 2003-04-30 | G·D·瑟尔公司 | 用于治疗类症的取代的异噁唑 |
US5756529A (en) * | 1995-09-29 | 1998-05-26 | G.D. Searle & Co. | Substituted pyrazolyl benzenesulfonamides for use in veterinary therapies |
US5981576A (en) * | 1995-10-13 | 1999-11-09 | Merck Frosst Canada, Inc. | (Methylsulfonyl)phenyl-2-(5H)-furanones as COX-2 inhibitors |
EP0863134A1 (en) * | 1997-03-07 | 1998-09-09 | Merck Frosst Canada Inc. | 2-(3,5-difluorophenyl)-3-(4-(methyl-sulfonyl)phenyl)-2-cyclopenten-1-one useful as an inhibitor of cyclooxygenase-2 |
AU3762699A (en) * | 1998-04-27 | 1999-11-16 | Pacific Northwest Cancer Foundation | (nr-cam) gene, nucleic acids and nucleic acid products for therapeutic and diagnostic uses for tumors |
-
2000
- 2000-12-01 OA OA1200100210A patent/OA11831A/en unknown
- 2000-12-01 NZ NZ529933A patent/NZ529933A/en unknown
- 2000-12-01 ES ES00983865T patent/ES2236011T3/es not_active Expired - Lifetime
- 2000-12-01 CZ CZ20012875A patent/CZ20012875A3/cs unknown
- 2000-12-01 CN CN008060835A patent/CN1216869C/zh not_active Expired - Fee Related
- 2000-12-01 PT PT00983865T patent/PT1150960E/pt unknown
- 2000-12-01 YU YU57801A patent/YU57801A/sh unknown
- 2000-12-01 HU HU0200580A patent/HUP0200580A3/hu unknown
- 2000-12-04 EC EC2000003807A patent/ECSP003807A/es unknown
- 2000-12-04 AU AU20412/01A patent/AU2041201A/en not_active Withdrawn
- 2000-12-04 WO PCT/US2000/030180 patent/WO2001041536A2/en not_active Application Discontinuation
- 2000-12-05 AR ARP000106473A patent/AR027897A1/es unknown
- 2000-12-06 EA EA200401397A patent/EA200401397A1/ru unknown
- 2000-12-06 PE PE2000001299A patent/PE20010911A1/es not_active Application Discontinuation
- 2000-12-06 AR ARP000106475A patent/AR030039A1/es unknown
- 2000-12-06 PT PT00982255T patent/PT1150959E/pt unknown
- 2000-12-06 KR KR1020017010017A patent/KR100717570B1/ko not_active IP Right Cessation
- 2000-12-06 MY MYPI20005730A patent/MY128971A/en unknown
- 2000-12-06 MY MYPI20005733A patent/MY128366A/en unknown
- 2000-12-08 SV SV2000000235A patent/SV2002000235A/es not_active Application Discontinuation
- 2000-12-11 CO CO00094077A patent/CO5251445A1/es not_active Application Discontinuation
-
2001
- 2001-05-18 TW TW089125991A patent/TWI276435B/zh not_active IP Right Cessation
- 2001-08-09 BG BG105808A patent/BG65239B1/bg unknown
- 2001-08-29 ZA ZA200107146A patent/ZA200107146B/xx unknown
- 2001-08-29 ZA ZA200107149A patent/ZA200107149B/xx unknown
Also Published As
Publication number | Publication date |
---|---|
ZA200107149B (en) | 2003-02-28 |
HUP0200580A2 (hu) | 2002-11-28 |
NZ529933A (en) | 2005-06-24 |
HUP0200580A3 (en) | 2002-12-28 |
AR030039A1 (es) | 2003-08-13 |
KR100717570B1 (ko) | 2007-05-15 |
ES2236011T3 (es) | 2005-07-16 |
MY128971A (en) | 2007-03-30 |
ZA200107146B (en) | 2002-08-29 |
OA11831A (en) | 2005-08-23 |
MY128366A (en) | 2007-01-31 |
CZ20012875A3 (cs) | 2002-02-13 |
EA200401397A1 (ru) | 2005-08-25 |
ECSP003807A (es) | 2005-07-06 |
PT1150959E (pt) | 2008-04-21 |
KR20020002386A (ko) | 2002-01-09 |
CN1216869C (zh) | 2005-08-31 |
BG105808A (en) | 2002-09-30 |
PT1150960E (pt) | 2005-06-30 |
SV2002000235A (es) | 2002-06-13 |
AR027897A1 (es) | 2003-04-16 |
TWI276435B (en) | 2007-03-21 |
YU57801A (sh) | 2005-07-19 |
WO2001041536A2 (en) | 2001-06-14 |
CN1411447A (zh) | 2003-04-16 |
BG65239B1 (bg) | 2007-09-28 |
CO5251445A1 (es) | 2003-02-28 |
PE20010911A1 (es) | 2001-09-10 |
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Legal Events
Date | Code | Title | Description |
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MK13 | Application withdrawn section 141(2)/reg 8.3(2) - pct appl. non-entering nat. phase, withdrawn by applicant |