ECSP003807A - Composiciones valdecoxib - Google Patents

Composiciones valdecoxib

Info

Publication number
ECSP003807A
ECSP003807A EC2000003807A ECSP003807A ECSP003807A EC SP003807 A ECSP003807 A EC SP003807A EC 2000003807 A EC2000003807 A EC 2000003807A EC SP003807 A ECSP003807 A EC SP003807A EC SP003807 A ECSP003807 A EC SP003807A
Authority
EC
Ecuador
Prior art keywords
compositions
valdecoxib
valdecoxib compositions
cyclooxygenase
prophylaxis
Prior art date
Application number
EC2000003807A
Other languages
English (en)
Inventor
Sreekant Nadkarni
Mark J Kontny
Tugrul Kararli
Subhash Desai
Original Assignee
Pharmacia Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia Corp filed Critical Pharmacia Corp
Publication of ECSP003807A publication Critical patent/ECSP003807A/es

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Classifications

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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    • A61K9/51—Nanocapsules; Nanoparticles
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Abstract

Se proporcionan las composiciones farmacéuticas que comprenden valdecoxib particulado en una cantidad de aproximadamente 1 mg a aproximadamente 100 mg y uno o más excipientes farmacéuticamente aceptables. Las composiciones son útiles en el tratamiento o profilaxis de las condiciones o desórdenes mediados por ciclooxígenasa-2.
EC2000003807A 1999-12-08 2000-12-04 Composiciones valdecoxib ECSP003807A (es)

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CO (1) CO5251445A1 (es)
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EA (1) EA200401397A1 (es)
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BR0210518A (pt) 2001-06-22 2004-06-22 Pfizer Prod Inc Composições farmacêuticas de dispersões de drogas e polìmeros neutros
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US7927613B2 (en) 2002-02-15 2011-04-19 University Of South Florida Pharmaceutical co-crystal compositions
US20030224006A1 (en) 2002-03-01 2003-12-04 Zaworotko Michael J. Multiple-component solid phases containing at least one active pharmaceutical ingredient
US7446107B2 (en) 2002-02-15 2008-11-04 Transform Pharmaceuticals, Inc. Crystalline forms of conazoles and methods of making and using the same
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EP1515703A1 (en) * 2002-06-21 2005-03-23 Transform Pharmaceuticals, Inc. Pharmaceutical compositions with improved dissolution
AU2003267231A1 (en) * 2002-09-20 2004-04-08 Transform Pharmaceuticals, Inc. Pharmaceutical compositions with improved dissolution
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ES2450648T3 (es) * 2004-06-29 2014-03-25 Takeda Pharma A/S Fabricación de composiciones farmacéuticas con liberación rápida de fármacos insolubles en agua y composiciones farmacéuticas obtenidas mediante el procedimiento de la invención
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US20080171746A1 (en) * 2005-03-14 2008-07-17 Thomas Klein Method for Preventing Cardiovascular Diseases
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CN103524416B (zh) * 2013-10-29 2016-08-17 湖北华世通生物医药科技有限公司 一种塞来昔布新晶型a及其制备方法
CN103508958A (zh) * 2013-10-30 2014-01-15 中美华世通生物医药科技（武汉）有限公司 一种塞来昔布新晶型c及其制备方法
CN103539739B (zh) * 2013-10-30 2016-02-10 中美华世通生物医药科技（武汉）有限公司 一种塞来昔布新晶型b及其制备方法
KR101476096B1 (ko) * 2014-03-28 2014-12-24 대원제약주식회사 용해도가 향상된 쎄레콕시브의 약제학적 조성물

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CN1216869C (zh) 2005-08-31
TWI276435B (en) 2007-03-21
PT1150960E (pt) 2005-06-30
ZA200107149B (en) 2003-02-28
AU2041201A (en) 2001-06-18
CO5251445A1 (es) 2003-02-28
WO2001041536A2 (en) 2001-06-14
ZA200107146B (en) 2002-08-29
OA11831A (en) 2005-08-23
KR20020002386A (ko) 2002-01-09
AR030039A1 (es) 2003-08-13
BG105808A (en) 2002-09-30
MY128366A (en) 2007-01-31
NZ529933A (en) 2005-06-24
HUP0200580A2 (hu) 2002-11-28
KR100717570B1 (ko) 2007-05-15
AR027897A1 (es) 2003-04-16
CN1411447A (zh) 2003-04-16
PE20010911A1 (es) 2001-09-10
YU57801A (sh) 2005-07-19
CZ20012875A3 (cs) 2002-02-13
SV2002000235A (es) 2002-06-13
EA200401397A1 (ru) 2005-08-25
BG65239B1 (bg) 2007-09-28
MY128971A (en) 2007-03-30
PT1150959E (pt) 2008-04-21
ES2236011T3 (es) 2005-07-16
HUP0200580A3 (en) 2002-12-28

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