BG64094B1 - Метод за получаване на нафтиридони и междинни съединения - Google Patents

Метод за получаване на нафтиридони и междинни съединения Download PDF

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Publication number
BG64094B1
BG64094B1 BG103087A BG10308799A BG64094B1 BG 64094 B1 BG64094 B1 BG 64094B1 BG 103087 A BG103087 A BG 103087A BG 10308799 A BG10308799 A BG 10308799A BG 64094 B1 BG64094 B1 BG 64094B1
Authority
BG
Bulgaria
Prior art keywords
formula
compound
alkyl
trifluoromethyl
give
Prior art date
Application number
BG103087A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG103087A (en
Inventor
Charles Chiu
Lewin Wint
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of BG103087A publication Critical patent/BG103087A/xx
Publication of BG64094B1 publication Critical patent/BG64094B1/bg

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Indole Compounds (AREA)
BG103087A 1998-01-16 1999-01-15 Метод за получаване на нафтиридони и междинни съединения BG64094B1 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US7160198P 1998-01-16 1998-01-16

Publications (2)

Publication Number Publication Date
BG103087A BG103087A (en) 1999-08-31
BG64094B1 true BG64094B1 (bg) 2003-12-31

Family

ID=22102373

Family Applications (1)

Application Number Title Priority Date Filing Date
BG103087A BG64094B1 (bg) 1998-01-16 1999-01-15 Метод за получаване на нафтиридони и междинни съединения

Country Status (39)

Country Link
EP (1) EP0930297B1 (hu)
JP (1) JPH11255745A (hu)
KR (1) KR19990067905A (hu)
CN (1) CN1228422A (hu)
AP (1) AP9901440A0 (hu)
AR (1) AR017228A1 (hu)
AT (1) ATE238281T1 (hu)
AU (1) AU9711598A (hu)
BG (1) BG64094B1 (hu)
BR (1) BR9900066A (hu)
CA (1) CA2258960C (hu)
DE (1) DE69907042T2 (hu)
DK (1) DK0930297T3 (hu)
EA (1) EA199900020A3 (hu)
EG (1) EG21514A (hu)
ES (1) ES2195513T3 (hu)
GT (1) GT199800199A (hu)
HR (1) HRP990013A2 (hu)
HU (1) HUP9900121A3 (hu)
ID (1) ID23612A (hu)
IL (1) IL127945A0 (hu)
IS (1) IS4943A (hu)
MA (1) MA24745A1 (hu)
NO (1) NO990185L (hu)
NZ (1) NZ333769A (hu)
OA (1) OA10955A (hu)
PA (1) PA8464701A1 (hu)
PE (1) PE20000172A1 (hu)
PL (1) PL330859A1 (hu)
PT (1) PT930297E (hu)
SA (1) SA99190971A (hu)
SG (1) SG76584A1 (hu)
SI (1) SI0930297T1 (hu)
SK (1) SK3899A3 (hu)
TN (1) TNSN99005A1 (hu)
TR (1) TR199900070A2 (hu)
TW (1) TW483890B (hu)
YU (1) YU1799A (hu)
ZA (1) ZA99277B (hu)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7019142B2 (en) * 1998-01-16 2006-03-28 Pfizer Inc. Process for preparing naphthyridones and intermediates
HN1999000141A (es) * 1998-09-03 2000-06-19 Pfizer Prod Inc Procedimiento para preparar sales de trovafloxacina de adicion de acidos.

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5164402A (en) * 1989-08-16 1992-11-17 Pfizer Inc Azabicyclo quinolone and naphthyridinone carboxylic acids
PL166381B1 (pl) * 1989-08-16 1995-05-31 Pfizer Sposób wytwarzania nowych podstawionych kwasów 7-azabicyklochinolonokarboksylowych PL PL PL PL
US5256791A (en) * 1992-03-02 1993-10-26 Pfizer Inc. Preparation of intermediates in the synthesis of quinoline antibiotics
US5475116A (en) * 1994-04-29 1995-12-12 Pfizer Inc. Aza bicyclo[3,1,0]hexane intermediates useful in the synthesis of quinolones
DE19733439A1 (de) * 1997-08-02 1999-02-04 Bayer Ag Neue 6-endo-Amino-3-azabicyclo(3.1.0)hexande, Verfahren zu deren Herstellung und deren Verwendung zur Herstellung von Chinolon- und Naphthyridincarbonsäure-Derviaten mit verbesserten Eigenschaften

Also Published As

Publication number Publication date
PL330859A1 (en) 1999-07-19
BR9900066A (pt) 2000-05-09
NO990185L (no) 1999-07-19
KR19990067905A (ko) 1999-08-25
DK0930297T3 (da) 2003-07-21
HU9900121D0 (en) 1999-03-29
TR199900070A3 (tr) 1999-10-21
PT930297E (pt) 2003-08-29
HUP9900121A3 (en) 2000-02-28
NZ333769A (en) 2000-03-27
PE20000172A1 (es) 2000-03-09
DE69907042T2 (de) 2003-10-16
AR017228A1 (es) 2001-08-22
ES2195513T3 (es) 2003-12-01
SA99190971A (ar) 2005-12-03
SG76584A1 (en) 2000-11-21
OA10955A (en) 2001-10-31
MA24745A1 (fr) 1999-10-01
IS4943A (is) 1999-07-17
IL127945A0 (en) 1999-11-30
EG21514A (en) 2001-11-28
ATE238281T1 (de) 2003-05-15
YU1799A (sh) 2000-03-21
EP0930297B1 (en) 2003-04-23
EA199900020A3 (ru) 1999-12-29
HRP990013A2 (en) 1999-10-31
TR199900070A2 (xx) 1999-10-21
EP0930297A1 (en) 1999-07-21
CA2258960C (en) 2002-09-03
SK3899A3 (en) 2000-03-13
SI0930297T1 (en) 2003-08-31
NO990185D0 (no) 1999-01-15
ZA99277B (en) 2000-07-17
TW483890B (en) 2002-04-21
ID23612A (id) 2000-05-04
CN1228422A (zh) 1999-09-15
EA199900020A2 (ru) 1999-08-26
JPH11255745A (ja) 1999-09-21
DE69907042D1 (de) 2003-05-28
BG103087A (en) 1999-08-31
TNSN99005A1 (fr) 2005-11-10
AU9711598A (en) 1999-08-05
AP9901440A0 (en) 1999-03-31
CA2258960A1 (en) 1999-07-16
GT199800199A (es) 2000-06-07
PA8464701A1 (es) 2000-09-29
HUP9900121A2 (hu) 1999-09-28

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