BR9900066A - Processo para a preparação de naftiridonas e intermediários. - Google Patents

Processo para a preparação de naftiridonas e intermediários.

Info

Publication number
BR9900066A
BR9900066A BR9900066-0A BR9900066A BR9900066A BR 9900066 A BR9900066 A BR 9900066A BR 9900066 A BR9900066 A BR 9900066A BR 9900066 A BR9900066 A BR 9900066A
Authority
BR
Brazil
Prior art keywords
preparation
intermediates
naphthyridones
naphydrides
naphthyridone
Prior art date
Application number
BR9900066-0A
Other languages
English (en)
Inventor
Charles Kwok-Fung Chiu
Lewin Theophilus Wint
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of BR9900066A publication Critical patent/BR9900066A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Indole Compounds (AREA)

Abstract

Patente de Invenção: <B>"PROCESSO PARA A PREPARAçãO DE NAFTIRIDONAS E INTERMEDIáRIOS''<D>. Um processo para a preparação de um ácido naftiridona-carboxílico e seus derivados faz uso de intermediários de cadeia lateral de fórmulas I e IV aqui incluídas.
BR9900066-0A 1998-01-16 1999-01-14 Processo para a preparação de naftiridonas e intermediários. BR9900066A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US7160198P 1998-01-16 1998-01-16

Publications (1)

Publication Number Publication Date
BR9900066A true BR9900066A (pt) 2000-05-09

Family

ID=22102373

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9900066-0A BR9900066A (pt) 1998-01-16 1999-01-14 Processo para a preparação de naftiridonas e intermediários.

Country Status (39)

Country Link
EP (1) EP0930297B1 (pt)
JP (1) JPH11255745A (pt)
KR (1) KR19990067905A (pt)
CN (1) CN1228422A (pt)
AP (1) AP9901440A0 (pt)
AR (1) AR017228A1 (pt)
AT (1) ATE238281T1 (pt)
AU (1) AU9711598A (pt)
BG (1) BG64094B1 (pt)
BR (1) BR9900066A (pt)
CA (1) CA2258960C (pt)
DE (1) DE69907042T2 (pt)
DK (1) DK0930297T3 (pt)
EA (1) EA199900020A3 (pt)
EG (1) EG21514A (pt)
ES (1) ES2195513T3 (pt)
GT (1) GT199800199A (pt)
HR (1) HRP990013A2 (pt)
HU (1) HUP9900121A3 (pt)
ID (1) ID23612A (pt)
IL (1) IL127945A0 (pt)
IS (1) IS4943A (pt)
MA (1) MA24745A1 (pt)
NO (1) NO990185L (pt)
NZ (1) NZ333769A (pt)
OA (1) OA10955A (pt)
PA (1) PA8464701A1 (pt)
PE (1) PE20000172A1 (pt)
PL (1) PL330859A1 (pt)
PT (1) PT930297E (pt)
SA (1) SA99190971A (pt)
SG (1) SG76584A1 (pt)
SI (1) SI0930297T1 (pt)
SK (1) SK3899A3 (pt)
TN (1) TNSN99005A1 (pt)
TR (1) TR199900070A2 (pt)
TW (1) TW483890B (pt)
YU (1) YU1799A (pt)
ZA (1) ZA99277B (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7019142B2 (en) * 1998-01-16 2006-03-28 Pfizer Inc. Process for preparing naphthyridones and intermediates
HN1999000141A (es) * 1998-09-03 2000-06-19 Pfizer Prod Inc Procedimiento para preparar sales de trovafloxacina de adicion de acidos.

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5164402A (en) * 1989-08-16 1992-11-17 Pfizer Inc Azabicyclo quinolone and naphthyridinone carboxylic acids
IE66202B1 (en) * 1989-08-16 1995-12-13 Pfizer Azabicyclo quinolone carboxylic acids
US5256791A (en) * 1992-03-02 1993-10-26 Pfizer Inc. Preparation of intermediates in the synthesis of quinoline antibiotics
US5475116A (en) * 1994-04-29 1995-12-12 Pfizer Inc. Aza bicyclo[3,1,0]hexane intermediates useful in the synthesis of quinolones
DE19733439A1 (de) * 1997-08-02 1999-02-04 Bayer Ag Neue 6-endo-Amino-3-azabicyclo(3.1.0)hexande, Verfahren zu deren Herstellung und deren Verwendung zur Herstellung von Chinolon- und Naphthyridincarbonsäure-Derviaten mit verbesserten Eigenschaften

Also Published As

Publication number Publication date
AP9901440A0 (en) 1999-03-31
TR199900070A3 (tr) 1999-10-21
JPH11255745A (ja) 1999-09-21
DE69907042D1 (de) 2003-05-28
TW483890B (en) 2002-04-21
AR017228A1 (es) 2001-08-22
KR19990067905A (ko) 1999-08-25
ID23612A (id) 2000-05-04
ES2195513T3 (es) 2003-12-01
TR199900070A2 (xx) 1999-10-21
NO990185L (no) 1999-07-19
HUP9900121A2 (hu) 1999-09-28
PE20000172A1 (es) 2000-03-09
DK0930297T3 (da) 2003-07-21
NZ333769A (en) 2000-03-27
OA10955A (en) 2001-10-31
HU9900121D0 (en) 1999-03-29
CA2258960A1 (en) 1999-07-16
GT199800199A (es) 2000-06-07
ZA99277B (en) 2000-07-17
AU9711598A (en) 1999-08-05
SG76584A1 (en) 2000-11-21
BG103087A (en) 1999-08-31
BG64094B1 (bg) 2003-12-31
PT930297E (pt) 2003-08-29
EP0930297B1 (en) 2003-04-23
IL127945A0 (en) 1999-11-30
CN1228422A (zh) 1999-09-15
EA199900020A2 (ru) 1999-08-26
TNSN99005A1 (fr) 2005-11-10
EG21514A (en) 2001-11-28
SI0930297T1 (en) 2003-08-31
DE69907042T2 (de) 2003-10-16
YU1799A (sh) 2000-03-21
SK3899A3 (en) 2000-03-13
NO990185D0 (no) 1999-01-15
IS4943A (is) 1999-07-17
ATE238281T1 (de) 2003-05-15
SA99190971A (ar) 2005-12-03
EP0930297A1 (en) 1999-07-21
HRP990013A2 (en) 1999-10-31
PA8464701A1 (es) 2000-09-29
CA2258960C (en) 2002-09-03
EA199900020A3 (ru) 1999-12-29
HUP9900121A3 (en) 2000-02-28
PL330859A1 (en) 1999-07-19
MA24745A1 (fr) 1999-10-01

Similar Documents

Publication Publication Date Title
BR9912109B1 (pt) compostos derivados de quinolina, composições farmacêuticas, processo para a manufatura de um composto, e, uso de um composto.
DK0804421T3 (da) 2-((Dihydro)pyrazolyl-3&#39;-oxymethylen)-anilider som skadedyrsbekæmpelsesmidler og fungicider
BR9714787A (pt) Compostos de 4- fenilpiperidina e processo para sua preparação
BR9809745A (pt) Sal cristalino de amina de cefdinir
CY1109593T1 (el) Παραγωγα 12,13-κυκλοπροπανο εποθιλονης
NO932873L (no) 9-(substituerte glycyl)amido)-6- dementyl-6-deoksotetrasykliner
ES2070660B1 (es) Un procedimiento para la preparacion de 2,5-damino-3-hidroxihexanos sustituidos, utiles como inhibidores de proteasas retrovirales.
BR9803755A (pt) Processo aperfeiçoado para obtenção de precursores de insulina tendo pontes de cistina corretamente ligadas.
BR9712100A (pt) Intermediários e processo para preparar olanzapina.
BR9812837A (pt) Processo para fazer um composto, e, composto
BR9912104B1 (pt) compostos derivados de quinolina, composições farmacêuticas, e, processo para a manufatura de um composto.
FI902555A0 (fi) Diarylstyrylkinolindisyror.
FI963169A (fi) Enkefalinaasin ja ACE:n inhibittoreina käyttökelpoisia uusia merkaptoasetyyliamido-1,3,4,5-tetrahydrobents/c/-atsepin-3-onidisulfidijohdannaisia
BR9909739A (pt) Benzotiadiazóis e derivados
PT1169337E (pt) Nitratos esteroides para o tratamento de lesoes oxidativas e disfuncoes endoteliais
BR0011700A (pt) Dinitrilas de ácido arilmalÈnico substituìdo como intermediários para a preparação de herbicidas
ZA200005161B (en) Anti-inflammatory, antibacterial benzyl phenol agents.
BR0115501A (pt) Processo quìmico e novos intermediários
BR0101230A (pt) Processo para a preparação de11-amino-3-cloro-6,11-diidro-5-5-dioxo-6-metil-dibenzo[c,f][1,2]tiazepina e aplicação para a sìntese detianeptina
DK0882726T3 (da) Carbazolcarboxamider som 5-HT1F-agonister
BR9916615A (pt) Método para a preparação de éteres de arila
MX11866A (es) Nuevas cicloalquilamidas y procedimiento para su preparacion.
BR9900066A (pt) Processo para a preparação de naftiridonas e intermediários.
BR9814495A (pt) Composto, processo para prepará-lo, uso do mesmo, composição farmacêutica, e, processo
BR9712307A (pt) Pirazolinonas para o tratamento de potência enfraquecida

Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 4, 5,6,7 E 8A ANUIDADES

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1910 DE 14/08/2007.