BG61815B1 - Фармакологично активни енантиомери - Google Patents

Фармакологично активни енантиомери Download PDF

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Publication number
BG61815B1
BG61815B1 BG100331A BG10033196A BG61815B1 BG 61815 B1 BG61815 B1 BG 61815B1 BG 100331 A BG100331 A BG 100331A BG 10033196 A BG10033196 A BG 10033196A BG 61815 B1 BG61815 B1 BG 61815B1
Authority
BG
Bulgaria
Prior art keywords
compound
formula
alkyl
alk
physiologically acceptable
Prior art date
Application number
BG100331A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG100331A (bg
Inventor
Leandro Baiocchi
Valerio Cioli
Original Assignee
Angelini Ricerche Spa Societa'consortile
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Angelini Ricerche Spa Societa'consortile filed Critical Angelini Ricerche Spa Societa'consortile
Publication of BG100331A publication Critical patent/BG100331A/bg
Publication of BG61815B1 publication Critical patent/BG61815B1/bg

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00—Anaesthetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/06—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Epoxy Compounds (AREA)
BG100331A 1993-07-01 1996-02-01 Фармакологично активни енантиомери BG61815B1 (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT93MI001418A IT1268414B1 (it) 1993-07-01 1993-07-01 Enantiomeri farmacologicamente attivi
PCT/EP1994/002061 WO1995001354A1 (en) 1993-07-01 1994-06-21 Pharmacologically active enantiomers

Publications (2)

Publication Number Publication Date
BG100331A BG100331A (bg) 1996-09-30
BG61815B1 true BG61815B1 (bg) 1998-06-30

Family

ID=11366510

Family Applications (1)

Application Number Title Priority Date Filing Date
BG100331A BG61815B1 (bg) 1993-07-01 1996-02-01 Фармакологично активни енантиомери

Country Status (30)

Country Link
US (3) US5741907A (zh)
EP (1) EP0707587B1 (zh)
JP (1) JP3096065B2 (zh)
KR (1) KR100306018B1 (zh)
CN (3) CN1046281C (zh)
AT (1) ATE158796T1 (zh)
AU (1) AU689478B2 (zh)
BG (1) BG61815B1 (zh)
BR (1) BR9406996A (zh)
CA (1) CA2166470C (zh)
CZ (1) CZ289526B6 (zh)
DE (1) DE69405999T2 (zh)
DK (1) DK0707587T3 (zh)
ES (1) ES2111309T3 (zh)
FI (1) FI111943B (zh)
GE (1) GEP19991791B (zh)
GR (1) GR3025806T3 (zh)
HK (2) HK1018777A1 (zh)
HU (1) HU221631B1 (zh)
IT (1) IT1268414B1 (zh)
LV (1) LV11546B (zh)
NO (1) NO305957B1 (zh)
NZ (1) NZ268014A (zh)
PL (1) PL181831B1 (zh)
RO (2) RO116899B1 (zh)
RU (1) RU2128180C1 (zh)
SK (1) SK281060B6 (zh)
UA (1) UA53607C2 (zh)
WO (1) WO1995001354A1 (zh)
ZA (1) ZA944570B (zh)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1268414B1 (it) * 1993-07-01 1997-02-27 Angelini Francesco Ist Ricerca Enantiomeri farmacologicamente attivi
JP2009018992A (ja) * 2007-07-10 2009-01-29 Sumitomo Chemical Co Ltd 光学活性ミルタザピンの製造方法
RU2706700C1 (ru) 2019-09-24 2019-11-20 Общество с ограниченной ответственностью "Научно-производственная компания "СКиФФ" Фармацевтическая композиция для коррекции поведения кошек и собак в стрессовых ситуациях

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3365453A (en) * 1963-10-28 1968-01-23 Sterling Drug Inc 1-phenyl-4-lower-alkyl-2-piperazinones
IT1066857B (it) * 1965-12-15 1985-03-12 Acraf Derivati della s ipiazolo 4.3 a piridina e processi per la loro preparazione
US5303837A (en) * 1991-03-05 1994-04-19 Portola Packaging, Inc. One-piece fitment and plug with tamper-evident band
GEP20001939B (en) * 1992-01-17 2000-02-05 Angelini Ricerca S P A Soc Consortile Alkyl Derivatives of Trazodone with CNS Activity
US5543563A (en) * 1992-01-17 1996-08-06 Istituto Ricerca Francesco Angelini S.P.A. Alkyl derivatives of trazodone with CNS activity
IT1268414B1 (it) * 1993-07-01 1997-02-27 Angelini Francesco Ist Ricerca Enantiomeri farmacologicamente attivi
US5399765A (en) * 1994-05-23 1995-03-21 Sepracor, Inc. Enantioselective preparation of optically pure albuterol

Also Published As

Publication number Publication date
CZ348595A3 (en) 1996-04-17
US5973150A (en) 1999-10-26
DE69405999T2 (de) 1998-04-16
KR100306018B1 (ko) 2001-11-30
AU7072994A (en) 1995-01-24
PL181831B1 (pl) 2001-09-28
DE69405999D1 (de) 1997-11-06
CA2166470C (en) 2001-12-18
FI956334A (fi) 1996-02-19
CN1046281C (zh) 1999-11-10
GEP19991791B (en) 1999-10-05
ITMI931418A1 (it) 1995-01-01
PL312419A1 (en) 1996-04-15
RO116899B1 (ro) 2001-07-30
GR3025806T3 (en) 1998-03-31
CN1215052A (zh) 1999-04-28
CZ289526B6 (cs) 2002-02-13
IT1268414B1 (it) 1997-02-27
EP0707587B1 (en) 1997-10-01
FI956334A0 (fi) 1995-12-29
NO955345L (no) 1996-02-29
NO305957B1 (no) 1999-08-23
CN1136201C (zh) 2004-01-28
ES2111309T3 (es) 1998-03-01
RO121031B1 (ro) 2006-11-30
HU9503876D0 (en) 1996-02-28
JP3096065B2 (ja) 2000-10-10
SK166495A3 (en) 1996-09-04
US5741907A (en) 1998-04-21
BG100331A (bg) 1996-09-30
DK0707587T3 (da) 1998-05-11
RU2128180C1 (ru) 1999-03-27
LV11546B (en) 1997-02-20
CN1129939A (zh) 1996-08-28
CN1136200C (zh) 2004-01-28
CN1215053A (zh) 1999-04-28
ZA944570B (en) 1995-04-11
ITMI931418A0 (it) 1993-07-01
NZ268014A (en) 1997-08-22
LV11546A (lv) 1996-10-20
HK1018777A1 (en) 2000-01-07
HK1018781A1 (en) 2000-01-07
UA53607C2 (uk) 2003-02-17
JPH08512036A (ja) 1996-12-17
BR9406996A (pt) 1996-09-10
EP0707587A1 (en) 1996-04-24
US5817815A (en) 1998-10-06
ATE158796T1 (de) 1997-10-15
WO1995001354A1 (en) 1995-01-12
SK281060B6 (sk) 2000-11-07
HUT73230A (en) 1996-07-29
NO955345D0 (no) 1995-12-29
FI111943B (fi) 2003-10-15
CA2166470A1 (en) 1995-01-12
HU221631B1 (hu) 2002-12-28
AU689478B2 (en) 1998-04-02

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