BG49275A3 - Method for preparing diazobicycloalkylchinolin carbonate acids - Google Patents

Method for preparing diazobicycloalkylchinolin carbonate acids

Info

Publication number
BG49275A3
BG49275A3 BG76465A BG7646586A BG49275A3 BG 49275 A3 BG49275 A3 BG 49275A3 BG 76465 A BG76465 A BG 76465A BG 7646586 A BG7646586 A BG 7646586A BG 49275 A3 BG49275 A3 BG 49275A3
Authority
BG
Bulgaria
Prior art keywords
diazobicycloalkylchinolin
preparing
alkyl
carbon
carbonate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
BG76465A
Other languages
English (en)
Inventor
Martin R Jefson
Paul R Mcguirk
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of BG49275A3 publication Critical patent/BG49275A3/xx
Active legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Oncology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Materials For Photolithography (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BG76465A 1985-09-18 1986-09-18 Method for preparing diazobicycloalkylchinolin carbonate acids Active BG49275A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US77747185A 1985-09-18 1985-09-18

Publications (1)

Publication Number Publication Date
BG49275A3 true BG49275A3 (en) 1991-09-16

Family

ID=25110350

Family Applications (2)

Application Number Title Priority Date Filing Date
BG76465A Active BG49275A3 (en) 1985-09-18 1986-09-18 Method for preparing diazobicycloalkylchinolin carbonate acids
BG96080A BG61091B2 (bg) 1985-09-18 1992-03-17 Антибактериални заместени мостови-диазабициклоалкил хинолон карбоксилови киселини

Family Applications After (1)

Application Number Title Priority Date Filing Date
BG96080A BG61091B2 (bg) 1985-09-18 1992-03-17 Антибактериални заместени мостови-диазабициклоалкил хинолон карбоксилови киселини

Country Status (42)

Country Link
US (3) US4861779A (ja)
EP (1) EP0215650B1 (ja)
JP (1) JPH0798819B2 (ja)
KR (1) KR870000961B1 (ja)
CN (1) CN1014789B (ja)
AT (1) ATE72245T1 (ja)
AU (1) AU576302B2 (ja)
BG (2) BG49275A3 (ja)
CA (1) CA1340734C (ja)
CY (1) CY1774A (ja)
CZ (1) CZ277825B6 (ja)
DD (1) DD259190A5 (ja)
DE (2) DE3683711D1 (ja)
DK (1) DK171276B1 (ja)
EG (1) EG18184A (ja)
ES (1) ES2001428A6 (ja)
FI (1) FI87565C (ja)
GR (1) GR862363B (ja)
HK (1) HK132795A (ja)
HU (1) HU200462B (ja)
IE (1) IE58966B1 (ja)
IL (1) IL80033A (ja)
IN (1) IN166416B (ja)
LU (1) LU90356I2 (ja)
MA (1) MA20770A1 (ja)
MW (1) MW5886A1 (ja)
MX (1) MX173358B (ja)
MY (1) MY102518A (ja)
NO (1) NO170335C (ja)
NZ (1) NZ217614A (ja)
OA (1) OA08410A (ja)
PH (2) PH24048A (ja)
PL (1) PL149987B1 (ja)
PT (1) PT83388B (ja)
SG (1) SG28094G (ja)
SK (1) SK667886A3 (ja)
SU (1) SU1482531A3 (ja)
UA (1) UA6340A1 (ja)
YU (1) YU45024B (ja)
ZA (1) ZA867063B (ja)
ZM (1) ZM8586A1 (ja)
ZW (1) ZW19386A1 (ja)

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DE3601567A1 (de) * 1986-01-21 1987-07-23 Bayer Ag 7-(azabicycloalkyl)-chinoloncarbonsaeure- und -naphthyridon-carbonsaeure-derivate
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US4968799A (en) * 1987-07-31 1990-11-06 Warner-Lambert Company Antibacterial agents
US4923879A (en) * 1987-07-31 1990-05-08 Warner-Lambert Company 1,8-Naphthyridines and their use as antibacterial agents
US4933335A (en) * 1987-08-07 1990-06-12 Warner-Lambert Company Quinolones as antibacterial agents
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DE3902079A1 (de) * 1988-04-15 1989-10-26 Bayer Ag I.m. injektionsformen von gyrase-inhibitoren
US5147873A (en) * 1988-08-23 1992-09-15 Pfizer Inc. Amino-substituted bridged azabicyclic quinolone carboxylic acids and esters
WO1990002123A1 (en) * 1988-08-23 1990-03-08 Pfizer Inc. Amino-substituted bridged azabicyclic quinolone carboxylic acids and esters
US4895943A (en) * 1988-10-25 1990-01-23 Pfizer Inc. Preparation of 1,4-diazabicyclo(3.2.2)nonane
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US5214051A (en) * 1989-08-01 1993-05-25 Pfizer Inc. Thiazolyl and oxazolyl[5,4-c]piperidyl-substituted quinolone-carboxylic acid and related analogs thereof having antibacterial properties are disclosed
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US5235054A (en) * 1992-07-15 1993-08-10 Pfizer Inc. 3-carboxaldehyde substituted quinolines and naphthyridines
GB2291421A (en) * 1994-07-16 1996-01-24 Pfizer A process for preparing a quinoline carboxylic acid
ES2092963B1 (es) * 1995-04-12 1997-12-16 Sint Quimica Sa Procedimiento para la preparacion del acido 1-ciclopropil-6-fluoro-1, 4-dihidro-7-(1s,4s)-5-metil-2,5-diazabiciclo(2.2.1) hept-2-il)-4-oxo-3-quinolincarboxilico y sus sales.
US5929086A (en) 1996-05-10 1999-07-27 Pharmacia & Upjohn Company Topical administration of antimicrobial agents for the treatment of systemic bacterial diseases
US6056436A (en) * 1997-02-20 2000-05-02 University Of Maryland Simultaneous measurement of temperature and strain using optical sensors
DE60008866T2 (de) * 1999-05-04 2005-01-27 Neurosearch A/S Heteroaryl diazabicycloalkene, deren herstellung und verwendung
FR2809732B1 (fr) * 2000-05-31 2002-07-19 Sanofi Synthelabo DERIVES DE 4(-2-PHENYLTHIAZOL-5-yl)-1,4-DIAZABICYCLO-[3.2.2] NONANE, LEUR PREPARATION ET LEUR APPLICATION ENTHERAPEUTIQUE
FR2809731B1 (fr) * 2000-05-31 2002-07-19 Sanofi Synthelabo Derives de 1,4-diazabicyclo-[3.2.2] nonane-pheylisoxazole, leur preparation et leur application en therapeutique
FR2809730B1 (fr) * 2000-05-31 2002-07-19 Sanofi Synthelabo Derives de 1,4-diazabicyclo[3.2.2] nonanebenzoxazole, -benzothiazole et -benzimidazole, leur preparation et leur application therapeutique
CN1331864C (zh) * 2001-03-02 2007-08-15 神经研究公司 新型2,5-二氮杂二环[2.2.1]庚烷衍生物
BR0314201A (pt) * 2002-09-10 2005-07-12 Pfizer Prod Inc Compostos diazabicìclicos úteis no tratamento de doenças do cns e outros distúrbios
PL210065B1 (pl) 2002-09-25 2011-11-30 Memory Pharm Corp Związki indazole, benzotiazole i benzoizotiazole, kompozycje farmaceutyczne je zawierające oraz zastosowanie związków
DE10312346A1 (de) * 2003-03-20 2004-09-30 Bayer Healthcare Ag Kontrolliertes Freisetzungssystem
DE10351448A1 (de) 2003-11-04 2005-06-09 Bayer Healthcare Ag Geschmackstoffhaltige Arzneimittelformulierungen mit verbesserten pharmazeutischen Eigenschaften
JP4824578B2 (ja) * 2003-12-22 2011-11-30 メモリー・ファーマシューティカルズ・コーポレイション インドール類、1,2−ベンズイソオキサゾール類、および1,2−ベンゾイソチアゾール類、ならびにそれらの製造と使用
KR101176670B1 (ko) * 2004-03-25 2012-08-23 메모리 파마슈티칼스 코포레이션 인다졸, 벤조티아졸, 벤조이소티아졸, 벤즈이속사졸, 및그의 제조법 및 용도
EP1742944B1 (en) * 2004-04-22 2010-11-10 Memory Pharmaceuticals Corporation Indoles, 1h-indazoles, 1,2-benzisoxazoles, 1,2-benzoisothiazoles, and preparation and uses thereof
WO2005111038A2 (en) * 2004-05-07 2005-11-24 Memory Pharmaceuticals Corporation 1h-indazoles, benzothiazoles, 1,2-benzoisoxazoles, 1,2-benzoisothiazoles, and chromones and preparation and uses thereof
DE102005055385A1 (de) * 2004-12-09 2006-06-14 Bayer Healthcare Ag Arzneimittel zur hygienischen Applikation im Ohr
AU2005319248A1 (en) * 2004-12-22 2006-06-29 Memory Pharmaceuticals Corporation Nicotinic alpha-7 receptor ligands and preparation and uses thereof
US8106066B2 (en) 2005-09-23 2012-01-31 Memory Pharmaceuticals Corporation Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof
CA2641678A1 (en) 2006-02-10 2007-08-16 Neurosearch A/S 3,9-diazabicyclo[3.3.1]nonane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
AU2007213671A1 (en) 2006-02-10 2007-08-16 Neurosearch A/S 3-heteroaryl- 3,9-diazabicyclo[3.3.1]nonane derivatives as nicotinic acetylcholine receptor agonists
WO2007090887A1 (en) 2006-02-10 2007-08-16 Neurosearch A/S 3, 9-diazabicyclo [3.3. 1]nonane derivatives and their use as monoamine?neurotransmitter re-uptake inhibitors
DE102006010643A1 (de) 2006-03-08 2007-09-13 Bayer Healthcare Aktiengesellschaft Arzneimittel enthaltend Fluorchinolone
DE102006010642A1 (de) * 2006-03-08 2007-09-27 Bayer Healthcare Aktiengesellschaft Arzneimittelformulierungen, enthaltend Fluorchinolone
DE102007026550A1 (de) * 2007-06-08 2008-12-11 Bayer Healthcare Ag Extrudate mit verbesserter Geschmacksmaskierung
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Also Published As

Publication number Publication date
DK445886A (da) 1987-05-27
EP0215650B1 (en) 1992-01-29
DD259190A5 (de) 1988-08-17
PT83388A (en) 1986-10-01
OA08410A (fr) 1988-06-30
ZM8586A1 (en) 1987-03-27
US4861779A (en) 1989-08-29
UA6340A1 (uk) 1994-12-29
JPH0798819B2 (ja) 1995-10-25
MX3751A (es) 1993-09-01
AU6276886A (en) 1987-03-19
IL80033A (en) 1992-05-25
SG28094G (en) 1994-10-28
PT83388B (pt) 1989-05-12
CY1774A (en) 1995-10-20
NO170335B (no) 1992-06-29
FI87565B (fi) 1992-10-15
US5091383A (en) 1992-02-25
EG18184A (en) 1992-12-30
DE19675019I2 (de) 2004-01-29
DK171276B1 (da) 1996-08-19
KR870003106A (ko) 1987-04-15
ZA867063B (en) 1988-04-27
CN1014789B (zh) 1991-11-20
FI87565C (fi) 1993-01-25
CN86106385A (zh) 1987-06-03
MY102518A (en) 1992-07-31
GR862363B (en) 1987-01-19
SK278605B6 (en) 1997-11-05
MW5886A1 (en) 1987-12-09
CA1340734C (en) 1999-09-14
PH25338A (en) 1991-04-30
LU90356I2 (fr) 1999-04-26
HUT43070A (en) 1987-09-28
FI863756A0 (fi) 1986-09-17
US4775668A (en) 1988-10-04
SU1482531A3 (ru) 1989-05-23
IL80033A0 (en) 1986-12-31
MA20770A1 (fr) 1987-04-01
HK132795A (en) 1995-09-01
PL149987B1 (en) 1990-04-30
JPS62103083A (ja) 1987-05-13
HU200462B (en) 1990-06-28
ATE72245T1 (de) 1992-02-15
IE862479L (en) 1987-03-18
NO863718D0 (no) 1986-09-17
ZW19386A1 (en) 1986-12-10
CZ667886A3 (en) 1993-02-17
PL261410A1 (en) 1987-11-16
SK667886A3 (en) 1997-11-05
YU161786A (en) 1987-10-31
ES2001428A6 (es) 1988-05-16
FI863756A (fi) 1987-03-19
BG61091B2 (bg) 1996-10-31
PH24048A (en) 1990-03-05
DE3683711D1 (de) 1992-03-12
NO170335C (no) 1992-10-07
DK445886D0 (da) 1986-09-17
EP0215650A3 (en) 1987-12-02
AU576302B2 (en) 1988-08-18
IN166416B (ja) 1990-05-05
IE58966B1 (en) 1993-12-01
KR870000961B1 (ko) 1987-05-14
NO863718L (no) 1987-03-19
NZ217614A (en) 1989-11-28
MX173358B (es) 1994-02-23
EP0215650A2 (en) 1987-03-25
CZ277825B6 (en) 1993-06-16
YU45024B (en) 1991-06-30

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