BG103489A - Зипрасидонови препарати - Google Patents

Зипрасидонови препарати

Info

Publication number
BG103489A
BG103489A BG103489A BG10348999A BG103489A BG 103489 A BG103489 A BG 103489A BG 103489 A BG103489 A BG 103489A BG 10348999 A BG10348999 A BG 10348999A BG 103489 A BG103489 A BG 103489A
Authority
BG
Bulgaria
Prior art keywords
ziprasidon
preparations
crystalline
compositions
ziprosidonhydrochloride
Prior art date
Application number
BG103489A
Other languages
English (en)
Other versions
BG64691B1 (bg
Inventor
Frank BUSCH
Angela Hausberger
Bijan Rasadi
Daniel ARENSON
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22216447&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BG103489(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of BG103489A publication Critical patent/BG103489A/bg
Publication of BG64691B1 publication Critical patent/BG64691B1/bg

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682—Processes
    • A61K9/1688—Processes resulting in pure drug agglomerate optionally containing up to 5% of excipient
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Detergent Compositions (AREA)
  • Feeding Of Articles By Means Other Than Belts Or Rollers (AREA)
  • Polyamides (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Изобретението се отнася до състави, съдържащи частици на кристална свободна база на зипрасидон или на кристален зипрасидонхидрохлорид, които имат среден размер приблизително 85 m, и фармацевтично приемлив носител. Съставите са биоеквивалентни и могат да се използват за лечение на психози като шизофрения.
BG103489A 1998-06-15 1999-06-14 Зипрасидонови препарати BG64691B1 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US8922998P 1998-06-15 1998-06-15

Publications (2)

Publication Number Publication Date
BG103489A true BG103489A (bg) 2000-07-31
BG64691B1 BG64691B1 (bg) 2005-12-30

Family

ID=22216447

Family Applications (1)

Application Number Title Priority Date Filing Date
BG103489A BG64691B1 (bg) 1998-06-15 1999-06-14 Зипрасидонови препарати

Country Status (45)

Country Link
US (1) US6150366A (bg)
EP (1) EP0965343B1 (bg)
JP (2) JP3441676B2 (bg)
KR (1) KR100338915B1 (bg)
CN (1) CN1307994C (bg)
AP (1) AP1216A (bg)
AR (1) AR015553A1 (bg)
AT (1) ATE240732T1 (bg)
AU (1) AU753820B2 (bg)
BG (1) BG64691B1 (bg)
BR (1) BR9902268A (bg)
CA (1) CA2274338C (bg)
CO (1) CO5070579A1 (bg)
CY (1) CY2003002I1 (bg)
CZ (1) CZ297954B6 (bg)
DE (1) DE69908021T2 (bg)
DK (1) DK0965343T3 (bg)
EA (1) EA002223B1 (bg)
ES (1) ES2197581T3 (bg)
GT (1) GT199900080A (bg)
HK (1) HK1024184A1 (bg)
HN (1) HN1999000089A (bg)
HR (1) HRP990193B1 (bg)
HU (1) HU226487B1 (bg)
ID (1) ID23546A (bg)
IL (1) IL130424A (bg)
IS (1) IS2182B (bg)
MA (1) MA26647A1 (bg)
MY (1) MY121397A (bg)
NO (1) NO316713B1 (bg)
NZ (1) NZ336271A (bg)
OA (1) OA11064A (bg)
PA (1) PA8475601A1 (bg)
PE (1) PE20000632A1 (bg)
PL (2) PL195209B1 (bg)
PT (1) PT965343E (bg)
RS (1) RS49611B (bg)
SG (1) SG77243A1 (bg)
SI (1) SI0965343T1 (bg)
SK (1) SK286245B6 (bg)
TR (1) TR199901379A2 (bg)
TW (1) TW590774B (bg)
UA (1) UA59383C2 (bg)
UY (1) UY25649A1 (bg)
ZA (1) ZA993938B (bg)

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Also Published As

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OA11064A (en) 2002-03-13
ES2197581T3 (es) 2004-01-01
JP2000007566A (ja) 2000-01-11
HRP990193B1 (en) 2003-08-31
CZ297954B6 (cs) 2007-05-09
CA2274338C (en) 2003-04-15
HUP9901960A2 (hu) 2000-08-28
MY121397A (en) 2006-01-28
AR015553A1 (es) 2001-05-02
JP4187423B2 (ja) 2008-11-26
SK76999A3 (en) 2000-12-11
JP3441676B2 (ja) 2003-09-02
DE69908021D1 (de) 2003-06-26
HN1999000089A (es) 1999-11-03
PL195209B1 (pl) 2007-08-31
ID23546A (id) 2000-05-04
PT965343E (pt) 2003-08-29
DK0965343T3 (da) 2003-08-04
NO992892L (no) 1999-12-16
HU9901960D0 (en) 1999-08-30
HK1024184A1 (en) 2000-10-05
KR100338915B1 (ko) 2002-05-30
EP0965343A3 (en) 2000-02-23
HRP990193A2 (en) 2000-02-29
UY25649A1 (es) 2000-02-23
IL130424A (en) 2003-10-31
NZ336271A (en) 2000-10-27
CN1242987A (zh) 2000-02-02
US6150366A (en) 2000-11-21
HUP9901960A3 (en) 2000-09-28
CZ212799A3 (cs) 2000-09-13
TW590774B (en) 2004-06-11
BR9902268A (pt) 2000-05-02
AU753820B2 (en) 2002-10-31
RS49611B (sr) 2007-06-04
SK286245B6 (sk) 2008-06-06
JP2002003492A (ja) 2002-01-09
CO5070579A1 (es) 2001-08-28
CA2274338A1 (en) 1999-12-15
SI0965343T1 (en) 2003-10-31
EP0965343A2 (en) 1999-12-22
EA002223B1 (ru) 2002-02-28
PA8475601A1 (es) 2000-09-29
KR20000006143A (ko) 2000-01-25
HU226487B1 (en) 2009-03-02
IL130424A0 (en) 2000-06-01
NO316713B1 (no) 2004-04-13
CN1307994C (zh) 2007-04-04
ZA993938B (en) 2000-12-14
EA199900467A2 (ru) 1999-12-29
NO992892D0 (no) 1999-06-14
AP9901579A0 (en) 1999-06-30
CY2003002I1 (el) 2009-11-04
AU3398399A (en) 1999-12-23
TR199901379A2 (xx) 2000-01-21
SG77243A1 (en) 2000-12-19
EP0965343B1 (en) 2003-05-21
EA199900467A3 (ru) 2000-04-24
BG64691B1 (bg) 2005-12-30
PE20000632A1 (es) 2000-07-26
ATE240732T1 (de) 2003-06-15
IS2182B (is) 2006-12-15
UA59383C2 (uk) 2003-09-15
MA26647A1 (fr) 2004-12-20
YU27199A (sh) 2002-12-10
DE69908021T2 (de) 2003-11-27
PL333737A1 (en) 1999-12-20
AP1216A (en) 2003-10-19
GT199900080A (es) 2000-11-29
PL195606B1 (pl) 2007-10-31
IS5079A (is) 1999-12-16

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