IL130424A - Compositions comprising ziprasidone or its hydrochloride monohydrate, their preparation and use thereof in the preparation of medicaments for treating psychosis - Google Patents

Compositions comprising ziprasidone or its hydrochloride monohydrate, their preparation and use thereof in the preparation of medicaments for treating psychosis

Info

Publication number
IL130424A
IL130424A IL13042496A IL13042499A IL130424A IL 130424 A IL130424 A IL 130424A IL 13042496 A IL13042496 A IL 13042496A IL 13042499 A IL13042499 A IL 13042499A IL 130424 A IL130424 A IL 130424A
Authority
IL
Israel
Prior art keywords
preparation
ziprasidone
medicaments
compositions
hydrochloride monohydrate
Prior art date
Application number
IL13042496A
Other languages
English (en)
Other versions
IL130424A0 (en
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22216447&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL130424(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of IL130424A0 publication Critical patent/IL130424A0/xx
Publication of IL130424A publication Critical patent/IL130424A/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682—Processes
    • A61K9/1688—Processes resulting in pure drug agglomerate optionally containing up to 5% of excipient
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Polyamides (AREA)
  • Detergent Compositions (AREA)
  • Feeding Of Articles By Means Other Than Belts Or Rollers (AREA)
IL13042496A 1998-06-15 1999-06-10 Compositions comprising ziprasidone or its hydrochloride monohydrate, their preparation and use thereof in the preparation of medicaments for treating psychosis IL130424A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US8922998P 1998-06-15 1998-06-15

Publications (2)

Publication Number Publication Date
IL130424A0 IL130424A0 (en) 2000-06-01
IL130424A true IL130424A (en) 2003-10-31

Family

ID=22216447

Family Applications (1)

Application Number Title Priority Date Filing Date
IL13042496A IL130424A (en) 1998-06-15 1999-06-10 Compositions comprising ziprasidone or its hydrochloride monohydrate, their preparation and use thereof in the preparation of medicaments for treating psychosis

Country Status (45)

Country Link
US (1) US6150366A (xx)
EP (1) EP0965343B1 (xx)
JP (2) JP3441676B2 (xx)
KR (1) KR100338915B1 (xx)
CN (1) CN1307994C (xx)
AP (1) AP1216A (xx)
AR (1) AR015553A1 (xx)
AT (1) ATE240732T1 (xx)
AU (1) AU753820B2 (xx)
BG (1) BG64691B1 (xx)
BR (1) BR9902268A (xx)
CA (1) CA2274338C (xx)
CO (1) CO5070579A1 (xx)
CY (1) CY2003002I1 (xx)
CZ (1) CZ297954B6 (xx)
DE (1) DE69908021T2 (xx)
DK (1) DK0965343T3 (xx)
EA (1) EA002223B1 (xx)
ES (1) ES2197581T3 (xx)
GT (1) GT199900080A (xx)
HK (1) HK1024184A1 (xx)
HN (1) HN1999000089A (xx)
HR (1) HRP990193B1 (xx)
HU (1) HU226487B1 (xx)
ID (1) ID23546A (xx)
IL (1) IL130424A (xx)
IS (1) IS2182B (xx)
MA (1) MA26647A1 (xx)
MY (1) MY121397A (xx)
NO (1) NO316713B1 (xx)
NZ (1) NZ336271A (xx)
OA (1) OA11064A (xx)
PA (1) PA8475601A1 (xx)
PE (1) PE20000632A1 (xx)
PL (2) PL195606B1 (xx)
PT (1) PT965343E (xx)
RS (1) RS49611B (xx)
SG (1) SG77243A1 (xx)
SI (1) SI0965343T1 (xx)
SK (1) SK286245B6 (xx)
TR (1) TR199901379A2 (xx)
TW (1) TW590774B (xx)
UA (1) UA59383C2 (xx)
UY (1) UY25649A1 (xx)
ZA (1) ZA993938B (xx)

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US10179130B2 (en) 1999-10-29 2019-01-15 Purdue Pharma L.P. Controlled release hydrocodone formulations
AU2002227383B2 (en) 2000-10-30 2004-07-08 Euro-Celtique S.A. Controlled release hydrocodone formulations
US20040048876A1 (en) * 2002-02-20 2004-03-11 Pfizer Inc. Ziprasidone composition and synthetic controls
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AU2003231788B2 (en) 2002-05-17 2008-09-11 Duke University Method for treating obesity
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AU2003300814A1 (en) * 2002-12-04 2004-06-23 Dr. Reddy's Laboratories Inc. Polymorphic forms of ziprasidone and its hydrochloride
US20050143396A1 (en) * 2003-04-11 2005-06-30 Hertero Drugs Limited Novel crystalline forms of ziprasidone hydrochloride
WO2004096201A1 (en) * 2003-04-29 2004-11-11 Orexigen Therapeutics, Inc. Compositions for affecting weight loss
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CA2471219A1 (en) * 2004-06-14 2005-12-14 Apotex Pharmachem Inc. Improved preparation of an anhydrate form of 5-[2-[4-(1,2-benzisothiazol-3-yl)-1-piperazinyl]ethyl]-6-chloro-1,3-dihydro-2h-indol-2-one hydrochloride (ziprasidone hydrochloride)
US9044503B2 (en) * 2004-08-27 2015-06-02 University Of Kentucky Research Foundation Amyloid peptide inactivating enzyme to treat alzheimer's disease peripherally
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US8410268B2 (en) * 2008-03-11 2013-04-02 Alkem Laboratories Limited Process for the preparation of ziprasidone
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DE102008045854A1 (de) 2008-09-05 2010-03-11 Tiefenbacher Pharmachemikalien Alfred E. Tiefenbacher Gmbh & Co. Kg Partikel aus Ziprasidone und einem Sprengmittel enthaltende Pharmazeutische Zusammensetzung
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Also Published As

Publication number Publication date
HUP9901960A2 (hu) 2000-08-28
JP4187423B2 (ja) 2008-11-26
CZ212799A3 (cs) 2000-09-13
CO5070579A1 (es) 2001-08-28
KR100338915B1 (ko) 2002-05-30
AP1216A (en) 2003-10-19
IL130424A0 (en) 2000-06-01
ES2197581T3 (es) 2004-01-01
BG64691B1 (bg) 2005-12-30
JP2000007566A (ja) 2000-01-11
ATE240732T1 (de) 2003-06-15
PL195606B1 (pl) 2007-10-31
AU753820B2 (en) 2002-10-31
ZA993938B (en) 2000-12-14
NO316713B1 (no) 2004-04-13
MY121397A (en) 2006-01-28
RS49611B (sr) 2007-06-04
IS5079A (is) 1999-12-16
UA59383C2 (uk) 2003-09-15
TW590774B (en) 2004-06-11
HRP990193A2 (en) 2000-02-29
HN1999000089A (es) 1999-11-03
DE69908021D1 (de) 2003-06-26
NZ336271A (en) 2000-10-27
OA11064A (en) 2002-03-13
EP0965343A2 (en) 1999-12-22
MA26647A1 (fr) 2004-12-20
EA002223B1 (ru) 2002-02-28
IS2182B (is) 2006-12-15
HUP9901960A3 (en) 2000-09-28
GT199900080A (es) 2000-11-29
ID23546A (id) 2000-05-04
PA8475601A1 (es) 2000-09-29
PT965343E (pt) 2003-08-29
JP2002003492A (ja) 2002-01-09
BG103489A (en) 2000-07-31
YU27199A (sh) 2002-12-10
EA199900467A2 (ru) 1999-12-29
CZ297954B6 (cs) 2007-05-09
CA2274338C (en) 2003-04-15
AR015553A1 (es) 2001-05-02
US6150366A (en) 2000-11-21
CN1307994C (zh) 2007-04-04
JP3441676B2 (ja) 2003-09-02
DE69908021T2 (de) 2003-11-27
NO992892L (no) 1999-12-16
SI0965343T1 (en) 2003-10-31
UY25649A1 (es) 2000-02-23
SK76999A3 (en) 2000-12-11
TR199901379A2 (xx) 2000-01-21
PE20000632A1 (es) 2000-07-26
KR20000006143A (ko) 2000-01-25
CA2274338A1 (en) 1999-12-15
EA199900467A3 (ru) 2000-04-24
AP9901579A0 (en) 1999-06-30
CN1242987A (zh) 2000-02-02
DK0965343T3 (da) 2003-08-04
EP0965343A3 (en) 2000-02-23
CY2003002I1 (el) 2009-11-04
AU3398399A (en) 1999-12-23
EP0965343B1 (en) 2003-05-21
HU226487B1 (en) 2009-03-02
SG77243A1 (en) 2000-12-19
PL195209B1 (pl) 2007-08-31
HU9901960D0 (en) 1999-08-30
HK1024184A1 (en) 2000-10-05
BR9902268A (pt) 2000-05-02
PL333737A1 (en) 1999-12-20
NO992892D0 (no) 1999-06-14
HRP990193B1 (en) 2003-08-31
SK286245B6 (sk) 2008-06-06

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