PT1720867E - Processo para a preparação de ziprasidona - Google Patents
Processo para a preparação de ziprasidona Download PDFInfo
- Publication number
- PT1720867E PT1720867E PT05708625T PT05708625T PT1720867E PT 1720867 E PT1720867 E PT 1720867E PT 05708625 T PT05708625 T PT 05708625T PT 05708625 T PT05708625 T PT 05708625T PT 1720867 E PT1720867 E PT 1720867E
- Authority
- PT
- Portugal
- Prior art keywords
- ziprasidone
- preparation
- relates
- substantially pure
- hydrochloride
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Psychiatry (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Cephalosporin Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN307DE2004 | 2004-02-27 | ||
IN1395DE2004 | 2004-07-28 |
Publications (1)
Publication Number | Publication Date |
---|---|
PT1720867E true PT1720867E (pt) | 2010-01-28 |
Family
ID=34921521
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT05708625T PT1720867E (pt) | 2004-02-27 | 2005-02-28 | Processo para a preparação de ziprasidona |
Country Status (7)
Country | Link |
---|---|
US (2) | US20080312254A1 (pt) |
EP (1) | EP1720867B1 (pt) |
AT (1) | ATE451367T1 (pt) |
DE (1) | DE602005018171D1 (pt) |
ES (1) | ES2334800T3 (pt) |
PT (1) | PT1720867E (pt) |
WO (1) | WO2005085240A2 (pt) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2250000B1 (es) * | 2004-09-29 | 2007-06-01 | Medichem, S.A. | Procedimiento para la preparacion de ziprasidona. |
HU230479B1 (hu) * | 2006-05-02 | 2016-07-28 | Richter Gedeon Nyrt. | Eljárás 5-{2-[4-(1,2-benzizotiazol-3-il)-1-piperazinil]-etil}-6-klór-1,3-dihidro-2H-indol-2-on (Ziprasidon) előállítására |
WO2010010566A1 (en) * | 2008-07-25 | 2010-01-28 | Lupin Limited | Improved process for the manufacture of ziprasidone |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4831031A (en) * | 1988-01-22 | 1989-05-16 | Pfizer Inc. | Aryl piperazinyl-(C2 or C4) alkylene heterocyclic compounds having neuroleptic activity |
US5338846A (en) * | 1992-08-26 | 1994-08-16 | Pfizer Inc. | Process for preparing aryl piperazinyl-heterocyclic compounds with a piperazine salt |
US5206366A (en) * | 1992-08-26 | 1993-04-27 | Pfizer Inc. | Process for preparing aryl piperazinyl-heterocyclic compounds |
US5312925A (en) * | 1992-09-01 | 1994-05-17 | Pfizer Inc. | Monohydrate of 5-(2-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)-ethyl)-6-chloro-1,3-dihydro-2H-indol-2-one-hydrochloride |
JP3102896B2 (ja) * | 1996-05-07 | 2000-10-23 | ファイザー インク. | 5―(2―(4―(1,2―ベンズイソチアゾール―3―イル)―1―ピペラジニル)エチル)―6―クロロ―1,3―ジヒドロ―2(1h)―インドール―2―オン(=ジプラシドン)のメシレート三水和物、その調製法およびドーパミンd2アンタゴニストとしてのその使用 |
US6150366A (en) * | 1998-06-15 | 2000-11-21 | Pfizer Inc. | Ziprasidone formulations |
UY27668A1 (es) * | 2002-02-20 | 2003-10-31 | Pfizer Prod Inc | Composición de ziprasidona y controles sintéticos |
WO2004050655A1 (en) * | 2002-12-04 | 2004-06-17 | Dr. Reddy's Laboratories Limited | Polymorphic forms of ziprasidone and its hydrochloride |
AU2003245027A1 (en) * | 2003-04-11 | 2004-11-01 | Hetero Drugs Limited | Novel crystalline forms of ziprasidone hydrochloride |
EP1546146A1 (en) * | 2003-06-03 | 2005-06-29 | Teva Pharmaceutical Industries Limited | POLYMORPHIC FORMS OF ZIPRASIDONE HCl AND PROCESSES FOR THEIR PREPARATION |
US20050049295A1 (en) * | 2003-06-12 | 2005-03-03 | Dr. Reddy's Laboratories Limited | Process for the preparation of 5-(2-(4-(1,2-benzisothiazol-3-yl)-1piperazinyl) ethyl)-6-chloro-1, 3-dihydro-2h-indol-2-one hydrochloride (ziprasidone hydrochloride) and its intermediate |
CA2543805A1 (en) * | 2003-10-24 | 2005-05-06 | Gideon Pilarsky | Processes for preparation of ziprasidone |
-
2005
- 2005-02-28 US US10/598,370 patent/US20080312254A1/en not_active Abandoned
- 2005-02-28 PT PT05708625T patent/PT1720867E/pt unknown
- 2005-02-28 DE DE602005018171T patent/DE602005018171D1/de active Active
- 2005-02-28 EP EP05708625A patent/EP1720867B1/en active Active
- 2005-02-28 ES ES05708625T patent/ES2334800T3/es active Active
- 2005-02-28 AT AT05708625T patent/ATE451367T1/de not_active IP Right Cessation
- 2005-02-28 WO PCT/IB2005/000512 patent/WO2005085240A2/en active Application Filing
-
2011
- 2011-05-04 US US13/100,833 patent/US8178674B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
EP1720867A2 (en) | 2006-11-15 |
ES2334800T3 (es) | 2010-03-16 |
US20110207933A1 (en) | 2011-08-25 |
WO2005085240A3 (en) | 2005-12-01 |
DE602005018171D1 (de) | 2010-01-21 |
US20080312254A1 (en) | 2008-12-18 |
ATE451367T1 (de) | 2009-12-15 |
US8178674B2 (en) | 2012-05-15 |
WO2005085240A2 (en) | 2005-09-15 |
EP1720867B1 (en) | 2009-12-09 |
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