BE836528A - Nouveaux derives d'acide 3-amino- indazolecarboxylique - Google Patents

Nouveaux derives d'acide 3-amino- indazolecarboxylique

Info

Publication number
BE836528A
BE836528A BE162651A BE162651A BE836528A BE 836528 A BE836528 A BE 836528A BE 162651 A BE162651 A BE 162651A BE 162651 A BE162651 A BE 162651A BE 836528 A BE836528 A BE 836528A
Authority
BE
Belgium
Prior art keywords
amino
new derivatives
indazolecarboxylic acid
indazolecarboxylic
acid
Prior art date
Application number
BE162651A
Other languages
English (en)
French (fr)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE836528A publication Critical patent/BE836528A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
BE162651A 1974-12-13 1975-12-11 Nouveaux derives d'acide 3-amino- indazolecarboxylique BE836528A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2458965A DE2458965C3 (de) 1974-12-13 1974-12-13 3-Amino-indazol-N-carbonsäure-Derivate, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
BE836528A true BE836528A (fr) 1976-06-11

Family

ID=5933305

Family Applications (1)

Application Number Title Priority Date Filing Date
BE162651A BE836528A (fr) 1974-12-13 1975-12-11 Nouveaux derives d'acide 3-amino- indazolecarboxylique

Country Status (27)

Country Link
US (1) US4051252A (sv)
JP (1) JPS5182266A (sv)
AT (1) AT343653B (sv)
BE (1) BE836528A (sv)
CA (1) CA1059523A (sv)
CH (1) CH622250A5 (sv)
CS (1) CS189731B2 (sv)
DD (1) DD125484A5 (sv)
DE (1) DE2458965C3 (sv)
DK (1) DK137082C (sv)
ES (1) ES443429A1 (sv)
FI (1) FI753493A (sv)
FR (1) FR2293928A1 (sv)
GB (1) GB1490306A (sv)
HK (1) HK52580A (sv)
HU (1) HU173557B (sv)
IE (1) IE42208B1 (sv)
IL (1) IL48642A (sv)
KE (1) KE3078A (sv)
LU (1) LU73993A1 (sv)
NL (1) NL7514521A (sv)
NO (1) NO145382C (sv)
PL (1) PL99858B1 (sv)
SE (1) SE419645B (sv)
SU (1) SU604487A3 (sv)
YU (1) YU315275A (sv)
ZA (1) ZA757777B (sv)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431657A (en) * 1982-05-24 1984-02-14 Ayerst, Mckenna & Harrison Inc. Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives
KR20010086657A (ko) * 2000-03-02 2001-09-15 성재갑 아미노인다졸 유도체 및 이를 함유하는 싸이클린 의존키나아제 저해제 조성물
CN1926132B (zh) * 2000-09-15 2010-12-29 沃泰克斯药物股份有限公司 可用作蛋白激酶抑制剂的吡唑化合物
US6660731B2 (en) 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
AU2001291013A1 (en) * 2000-09-15 2002-03-26 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
SI1318997T1 (sl) * 2000-09-15 2006-12-31 Vertex Pharma Pirazolne spojine, uporabne kot inhibitorji protein-kinaze
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
HUP0400908A3 (en) 2000-12-21 2010-03-29 Vertex Pharma Pyrazole compounds useful as protein kinase inhibitors, their use and pharmaceutical compositions containing them
KR100406634B1 (ko) * 2001-03-12 2003-11-20 주식회사 엘지생명과학 3,5-디아미노인다졸 유도체, 그의 제조방법 및 사이클린의존성 키나아제 저해제로서의 그의 용도
JP4542338B2 (ja) 2001-09-26 2010-09-15 ファイザー イタリア ソシエタ ア レスポンサビリタ リミタータ キナーゼ阻害因子として活性なアミノインダゾール誘導体、それらの製造方法及びそれらを含有する医薬組成物
JP4656838B2 (ja) * 2002-02-06 2011-03-23 バーテックス ファーマシューティカルズ インコーポレイテッド Gsk−3の阻害剤として有用なヘテロアリール化合物
FR2836915B1 (fr) * 2002-03-11 2008-01-11 Aventis Pharma Sa Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
EP1485380B1 (en) 2002-03-15 2010-05-19 Vertex Pharmaceuticals Incorporated Azolylaminoazines as inhibitors of protein kinases
BR0311291A (pt) 2002-05-17 2005-03-29 Pharmacia Italia Spa Derivados de aminoindazol ativos como inibidores da cinase, processo para sua preparação e composições farmacêuticas compreendendo os mesmos
MY141867A (en) 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
ES2273043T3 (es) 2002-08-02 2007-05-01 Vertex Pharmaceuticals Incorporated Composiciones de pirazol utiles como inhibidores de gsk-3.
EP1556053A4 (en) * 2002-10-31 2006-04-19 Amgen Inc ANTI-INFLAMMATORY AGENTS
WO2004072029A2 (en) 2003-02-06 2004-08-26 Vertex Pharmaceuticals Incorporated Pyrazolopyridazines useful as inhibitors of protein kinases
JP2007513184A (ja) * 2003-12-04 2007-05-24 バーテックス ファーマシューティカルズ インコーポレイテッド プロテインキナーゼのインヒビターとして有用なキノキサリン
DE102004005172A1 (de) * 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
AU2006279376B2 (en) 2005-08-18 2011-04-14 Vertex Pharmaceuticals Incoporated Pyrazine kinase inhibitors
US7528142B2 (en) * 2005-11-03 2009-05-05 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
WO2007121339A2 (en) * 2006-04-14 2007-10-25 Abbott Laboratories Process for the preparation of indazolyl ureas that inhibit vanilloid subtype 1 (vr1) receptors
AU2007317435A1 (en) 2006-11-02 2008-05-15 Vertex Pharmaceuticals Incorporated Aminopyridines and aminopyrimidines useful as inhibitors of protein kinases
NZ577768A (en) 2006-12-19 2012-01-12 Vertex Pharma Aminopyrimidines useful as inhibitors of protein kinases
JP5393489B2 (ja) 2007-03-09 2014-01-22 バーテックス ファーマシューティカルズ インコーポレイテッド 蛋白キナーゼの阻害剤として有用なアミノピリミジン
JP2010520887A (ja) 2007-03-09 2010-06-17 バーテックス ファーマシューティカルズ インコーポレイテッド 蛋白キナーゼの阻害剤として有用なアミノピリジン
ES2435997T3 (es) 2007-03-09 2013-12-26 Vertex Pharmaceuticals, Inc. Aminopirimidinas útiles como inhibidores de las proteínas cinasas
CN101679386A (zh) 2007-04-13 2010-03-24 沃泰克斯药物股份有限公司 可用作激酶抑制剂的氨基嘧啶类化合物
EP2152696B1 (en) 2007-05-02 2014-09-24 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
CA2688584A1 (en) * 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
EP2152694A2 (en) 2007-05-02 2010-02-17 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
CN101687852A (zh) * 2007-05-24 2010-03-31 沃泰克斯药物股份有限公司 可用作激酶抑制剂的噻唑类和吡唑类化合物
ES2400104T3 (es) * 2007-07-31 2013-04-05 Vertex Pharmaceuticals Incorporated Proceso para preparación de 5-fluoro-1H-pirazolo[3,4-b]piridin-3-amina y derivados de la misma
WO2010027921A1 (en) * 2008-09-03 2010-03-11 Vertex Pharmaceuticals Incorporated Co-crystals and pharmaceutical formulations comprising the same
DE102009004245A1 (de) 2009-01-09 2010-07-15 Bayer Schering Pharma Aktiengesellschaft Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung
PT2890684T (pt) 2012-07-24 2018-05-07 Bial Portela & Ca Sa Compostos de ureia e sua utilização como inibidores de enzima
WO2014017938A2 (en) * 2012-07-27 2014-01-30 BIAL - PORTELA & Cª, S.A. Process for the synthesis of substituted urea compounds
CA2918993C (en) 2013-07-24 2021-08-24 Bial - Portela & Ca, S.A. Imidazolecarboxamides and their use as faah inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3133081A (en) * 1964-05-12 J-aminoindazole derivatives
CH397698A (de) * 1961-09-08 1965-08-31 Siegfried Ag Verfahren zur Herstellung neuer 1-Carbamyl-indazole
US3277100A (en) * 1963-05-31 1966-10-04 Du Pont Novel substituted pyrazoles
NL6707299A (sv) * 1966-07-16 1968-01-17
DE1770649A1 (de) * 1968-06-15 1971-11-11 Bayer Ag Substituierte 3-Amino-indazole

Also Published As

Publication number Publication date
IE42208L (en) 1976-06-13
KE3078A (en) 1980-10-03
ES443429A1 (es) 1977-04-16
SU604487A3 (ru) 1978-04-25
US4051252A (en) 1977-09-27
PL99858B1 (pl) 1978-08-31
NO145382C (no) 1982-03-10
ZA757777B (en) 1976-11-24
IE42208B1 (en) 1980-06-18
DK137082B (da) 1978-01-16
LU73993A1 (sv) 1976-11-11
HU173557B (hu) 1979-06-28
CH622250A5 (sv) 1981-03-31
NO145382B (no) 1981-11-30
NL7514521A (nl) 1976-06-15
DD125484A5 (sv) 1977-04-20
NO754024L (sv) 1976-06-15
FI753493A (sv) 1976-06-14
CS189731B2 (en) 1979-04-30
YU315275A (en) 1982-02-28
SE419645B (sv) 1981-08-17
DK137082C (da) 1978-06-19
GB1490306A (en) 1977-11-02
CA1059523A (en) 1979-07-31
AT343653B (de) 1978-06-12
FR2293928A1 (fr) 1976-07-09
ATA939775A (de) 1977-10-15
HK52580A (en) 1980-09-26
IL48642A (en) 1979-12-30
DE2458965A1 (de) 1976-06-16
FR2293928B1 (sv) 1979-09-21
DK567275A (da) 1976-06-14
AU8717075A (en) 1977-06-09
JPS5182266A (en) 1976-07-19
DE2458965B2 (de) 1979-02-22
IL48642A0 (en) 1976-02-29
SE7513990L (sv) 1976-06-14
DE2458965C3 (de) 1979-10-11

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