AU774385B2 - Spherical telithromycin clusters, method for the production and use thereof in the preparation of pharmaceutical forms - Google Patents

Spherical telithromycin clusters, method for the production and use thereof in the preparation of pharmaceutical forms Download PDF

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Publication number
AU774385B2
AU774385B2 AU70181/00A AU7018100A AU774385B2 AU 774385 B2 AU774385 B2 AU 774385B2 AU 70181/00 A AU70181/00 A AU 70181/00A AU 7018100 A AU7018100 A AU 7018100A AU 774385 B2 AU774385 B2 AU 774385B2
Authority
AU
Australia
Prior art keywords
telithromycin
spherical agglomerates
preparation
spherical
microns
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU70181/00A
Other languages
English (en)
Other versions
AU7018100A (en
Inventor
Jean-Yves Godard
Valerie Rognon
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharma SA
Original Assignee
Aventis Pharma SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9549351&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU774385(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Aventis Pharma SA filed Critical Aventis Pharma SA
Publication of AU7018100A publication Critical patent/AU7018100A/en
Application granted granted Critical
Publication of AU774385B2 publication Critical patent/AU774385B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682—Processes
    • A61K9/1688—Processes resulting in pure drug agglomerate optionally containing up to 5% of excipient
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AU70181/00A 1999-08-26 2000-08-28 Spherical telithromycin clusters, method for the production and use thereof in the preparation of pharmaceutical forms Ceased AU774385B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR9910810A FR2797875B1 (fr) 1999-08-26 1999-08-26 Agglomerats spheriques de telithromycine, leur procede de preparation et leur application dans la preparation de formes pharmaceutiques
FR9910810 1999-08-26
PCT/FR2000/002393 WO2001014393A2 (fr) 1999-08-26 2000-08-28 Agglomerats spheriques de telithromycine, leur procede de preparation et leur application dans la preparation de formes pharmaceutiques

Publications (2)

Publication Number Publication Date
AU7018100A AU7018100A (en) 2001-03-19
AU774385B2 true AU774385B2 (en) 2004-06-24

Family

ID=9549351

Family Applications (1)

Application Number Title Priority Date Filing Date
AU70181/00A Ceased AU774385B2 (en) 1999-08-26 2000-08-28 Spherical telithromycin clusters, method for the production and use thereof in the preparation of pharmaceutical forms

Country Status (34)

Country Link
US (1) US6825218B1 (enExample)
EP (1) EP1212336B1 (enExample)
JP (1) JP4871467B2 (enExample)
KR (1) KR100718222B1 (enExample)
CN (1) CN1183151C (enExample)
AR (1) AR025398A1 (enExample)
AT (1) ATE255590T1 (enExample)
AU (1) AU774385B2 (enExample)
BR (1) BR0013569B1 (enExample)
CA (1) CA2382497C (enExample)
CO (1) CO5190666A1 (enExample)
CZ (1) CZ2002594A3 (enExample)
DE (1) DE60006976T2 (enExample)
DK (1) DK1212336T3 (enExample)
EA (1) EA005080B1 (enExample)
ES (1) ES2209970T3 (enExample)
FR (1) FR2797875B1 (enExample)
HK (1) HK1049167B (enExample)
HR (1) HRP20020167B1 (enExample)
HU (1) HU229075B1 (enExample)
IL (2) IL148128A0 (enExample)
ME (2) MEP20108A (enExample)
MX (1) MXPA02001988A (enExample)
NO (1) NO322622B1 (enExample)
PL (1) PL204100B1 (enExample)
PT (1) PT1212336E (enExample)
RS (1) RS50433B (enExample)
SI (1) SI1212336T1 (enExample)
SK (1) SK287588B6 (enExample)
TR (1) TR200200506T2 (enExample)
TW (1) TWI272949B (enExample)
UA (1) UA73523C2 (enExample)
WO (1) WO2001014393A2 (enExample)
ZA (1) ZA200201599B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2002321289B2 (en) * 2002-07-19 2009-07-16 Aventis Pharma S.A. Taste masked oral composition of telithromycin

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9902202D0 (sv) * 1999-06-10 1999-06-10 Astra Ab Production of aggregates
FR2821747B1 (fr) * 2001-03-09 2004-07-02 Ethypharm Lab Prod Ethiques Suspension de telithromycine a gout masque
WO2004009059A1 (en) * 2002-07-19 2004-01-29 Aventis Pharma S.A. Taste masked oral composition of telithromycin
US20040013737A1 (en) * 2002-07-19 2004-01-22 Philippe Becourt Taste masked oral composition of telithromycin
EP1610878B1 (en) * 2003-02-21 2014-09-03 University Of Bath Process for the production of particles
WO2005007143A2 (en) * 2003-07-14 2005-01-27 The Board Of Trustees Of The University Of Illinois Use of makrolides and ketolides for the treatment of tuberculosis
WO2007039914A2 (en) * 2005-10-06 2007-04-12 Alembic Limited Novel polymorphs of telithromycin
US20090075917A1 (en) * 2007-09-19 2009-03-19 Protia, Llc Deuterium-enriched telithromycin
KR101324862B1 (ko) * 2011-07-12 2013-11-01 (주)에이에스텍 클로피도그렐 황산수소염의 구형 입자, 이를 포함하는 약학적 조성물 및 이의 제조방법

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0680967A1 (fr) * 1994-05-03 1995-11-08 Roussel-Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3468336D1 (en) * 1983-06-22 1988-02-11 Univ Ohio State Res Found Small particle formation
JPH02227130A (ja) * 1989-02-28 1990-09-10 Taisho Pharmaceut Co Ltd 球形微小凍結粒子の製造法

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0680967A1 (fr) * 1994-05-03 1995-11-08 Roussel-Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
DRUGS FUTURE 23:591-597 (GRAUL ET AL.) *

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2002321289B2 (en) * 2002-07-19 2009-07-16 Aventis Pharma S.A. Taste masked oral composition of telithromycin
AU2002321289B8 (en) * 2002-07-19 2009-08-06 Aventis Pharma S.A. Taste masked oral composition of telithromycin

Also Published As

Publication number Publication date
AU7018100A (en) 2001-03-19
CA2382497C (fr) 2011-06-28
CZ2002594A3 (cs) 2002-09-11
SK287588B6 (sk) 2011-03-04
SK2532002A3 (en) 2002-09-10
HK1049167B (zh) 2005-08-19
US6825218B1 (en) 2004-11-30
FR2797875B1 (fr) 2001-10-19
IL148128A (en) 2006-10-31
ATE255590T1 (de) 2003-12-15
UA73523C2 (uk) 2005-08-15
HUP0202842A3 (en) 2003-03-28
WO2001014393A3 (fr) 2001-06-21
KR100718222B1 (ko) 2007-05-15
NO20020926L (no) 2002-02-26
DK1212336T3 (da) 2004-03-15
CN1183151C (zh) 2005-01-05
DE60006976T2 (de) 2004-10-21
PL353137A1 (en) 2003-10-20
KR20020033771A (ko) 2002-05-07
HUP0202842A2 (hu) 2003-01-28
JP4871467B2 (ja) 2012-02-08
YU13202A (sh) 2004-09-03
CO5190666A1 (es) 2002-08-29
CA2382497A1 (fr) 2001-03-01
MEP20108A (en) 2010-06-10
CN1371386A (zh) 2002-09-25
BR0013569A (pt) 2002-05-14
ME00112B (me) 2010-10-10
RS50433B (sr) 2009-12-31
ES2209970T3 (es) 2004-07-01
AR025398A1 (es) 2002-11-27
TR200200506T2 (tr) 2002-08-21
EA005080B1 (ru) 2004-10-28
MXPA02001988A (es) 2002-08-20
PT1212336E (pt) 2004-04-30
HK1049167A1 (en) 2003-05-02
ZA200201599B (en) 2003-04-30
HRP20020167B1 (en) 2006-06-30
DE60006976D1 (de) 2004-01-15
WO2001014393A2 (fr) 2001-03-01
TWI272949B (en) 2007-02-11
FR2797875A1 (fr) 2001-03-02
PL204100B1 (pl) 2009-12-31
IL148128A0 (en) 2002-09-12
EP1212336A2 (fr) 2002-06-12
HU229075B1 (hu) 2013-07-29
BR0013569B1 (pt) 2014-02-25
NO20020926D0 (no) 2002-02-26
HRP20020167A2 (en) 2003-06-30
SI1212336T1 (en) 2004-04-30
EP1212336B1 (fr) 2003-12-03
NO322622B1 (no) 2006-11-06
JP2003507484A (ja) 2003-02-25
EA200200294A1 (ru) 2002-08-29

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Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase
TH Corrigenda

Free format text: IN VOL 15, NO 25, PAGE(S) 5185-5188 UNDER THE HEADING APPLICATIONS LAPSED, REFUSED OR WITHDRAWN PLEASE DELETE ALL REFERENCE TO APPLICATION NO. 70181/00 AND 74147/00

FGA Letters patent sealed or granted (standard patent)