AU536854B2 - 1 1-dioxopenicillanoyl methyl penicillanate esters - Google Patents

1 1-dioxopenicillanoyl methyl penicillanate esters

Info

Publication number
AU536854B2
AU536854B2 AU13871/83A AU1387183A AU536854B2 AU 536854 B2 AU536854 B2 AU 536854B2 AU 13871/83 A AU13871/83 A AU 13871/83A AU 1387183 A AU1387183 A AU 1387183A AU 536854 B2 AU536854 B2 AU 536854B2
Authority
AU
Australia
Prior art keywords
dioxopenicillanoyl
esters
methyl penicillanate
penicillanate
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
AU13871/83A
Other languages
English (en)
Other versions
AU1387183A (en
Inventor
Wayne Ernest Barth
Vytautas John Jasys
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
PFIZER
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by PFIZER, Pfizer Inc filed Critical PFIZER
Publication of AU1387183A publication Critical patent/AU1387183A/en
Application granted granted Critical
Publication of AU536854B2 publication Critical patent/AU536854B2/en
Anticipated expiration legal-status Critical
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32—Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Cephalosporin Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU13871/83A 1982-04-23 1983-04-22 1 1-dioxopenicillanoyl methyl penicillanate esters Expired AU536854B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/371,156 US4432987A (en) 1982-04-23 1982-04-23 Crystalline benzenesulfonate salts of sultamicillin
US371156 1999-08-09

Publications (2)

Publication Number Publication Date
AU1387183A AU1387183A (en) 1983-11-17
AU536854B2 true AU536854B2 (en) 1984-05-24

Family

ID=23462725

Family Applications (1)

Application Number Title Priority Date Filing Date
AU13871/83A Expired AU536854B2 (en) 1982-04-23 1983-04-22 1 1-dioxopenicillanoyl methyl penicillanate esters

Country Status (27)

Country Link
US (1) US4432987A (https=)
EP (1) EP0092968B1 (https=)
JP (1) JPS58201792A (https=)
KR (1) KR860001279B1 (https=)
AU (1) AU536854B2 (https=)
CA (1) CA1187484A (https=)
CS (1) CS235320B2 (https=)
DD (1) DD209632A5 (https=)
DE (1) DE3362502D1 (https=)
DK (1) DK162168C (https=)
EG (1) EG16412A (https=)
ES (1) ES8406075A1 (https=)
FI (1) FI76092C (https=)
GR (1) GR78582B (https=)
HK (1) HK20588A (https=)
HU (1) HU187068B (https=)
IE (1) IE54628B1 (https=)
IL (1) IL68453A (https=)
NO (1) NO156202C (https=)
NZ (1) NZ203988A (https=)
PH (1) PH18035A (https=)
PL (1) PL134978B1 (https=)
PT (1) PT76587B (https=)
SG (1) SG104087G (https=)
SU (1) SU1138030A3 (https=)
YU (1) YU43170B (https=)
ZA (1) ZA832845B (https=)

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JP3382159B2 (ja) * 1998-08-05 2003-03-04 株式会社東芝 情報記録媒体とその再生方法及び記録方法
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KR20060108692A (ko) * 2003-10-31 2006-10-18 알자 코포레이션 메트포르민의 개선된 흡수를 위한 조성물 및 제형
FR2877696B1 (fr) 2004-11-09 2009-09-18 Renault Sas Dispositif et procede d'estimation en temps reel de l'angle de debut de combustion d'un moteur a combustion interne
DK2195293T3 (da) 2007-08-22 2014-02-03 Astrazeneca Ab Cyclopropylamidderivater
EP2620432A3 (en) 2007-10-26 2013-12-18 The Regents Of the University of California Diarylhydantoin compounds
CN102405047B (zh) * 2009-01-30 2014-07-09 葛兰素史密斯克莱有限责任公司 结晶型的n-{(1s)-2-氨基-1-[(3-氟苯基)甲基]乙基}-5-氯-4-(4-氯-1-甲基-1h-吡唑-5-基)-2-噻吩甲酰胺盐酸盐
TW201039825A (en) 2009-02-20 2010-11-16 Astrazeneca Ab Cyclopropyl amide derivatives 983
JP2012532886A (ja) * 2009-07-10 2012-12-20 エボルバ アクチェンゲゼルシャフト ジイン組成物
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US20110201622A1 (en) * 2010-02-18 2011-08-18 Collins Craig D Solid Forms Comprising A Cyclopropyl Amide Derivative
WO2014087972A1 (ja) * 2012-12-03 2014-06-12 株式会社カネカ 還元型補酵素ｑ10誘導体およびその製造方法
CN105517992B (zh) * 2013-09-05 2018-06-22 田边三菱制药株式会社 新型结晶性芳烷基胺化合物及其制造方法
UA119794C2 (uk) * 2014-10-21 2019-08-12 Аріад Фармасьютикалз, Інк. Кристалічна форма 5-хлор-n4-[2-(диметилфосфорил)феніл]-n2-{2-метокси-4-[4-(4-метилпіперазин-1-іл)піперидин-1-іл]}піримідин-2,4-діаміну
CN104958318A (zh) * 2015-08-04 2015-10-07 青岛蓝盛洋医药生物科技有限责任公司 一种治疗感染性疾病的药物舒巴坦钠组合物
EP3778567A1 (en) * 2016-01-22 2021-02-17 Sandoz Ag Crystalline eravacycline bis-hydrochloride
CN109563087A (zh) * 2016-07-07 2019-04-02 铁木医药有限公司 sGC刺激剂的固体形式
EP3703686A4 (en) * 2017-10-30 2021-11-17 Theracaine LLC HYDROPHOBIC ARENE SULFONATE SALTS
US11186556B1 (en) * 2018-10-16 2021-11-30 Celgene Corporation Salts of a thiazolidinone compound, solid forms, compositions and methods of use thereof
UA119735C2 (uk) 2018-12-20 2019-07-25 Анатолій Семенович Редер Фармацевтична сполука, спосіб її отримання та застосування як лікарського засобу
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JP7805677B2 (ja) * 2021-12-28 2026-01-26 浙江揚歴医薬技術有限公司 テトラヒドロシクロヘプタインダゾール化合物の結晶
EP4525860A2 (en) * 2022-05-20 2025-03-26 Caamtech, Inc. Tryptamine derivatives
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USD1057882S1 (en) 2022-08-29 2025-01-14 Springfield, Inc. Combined serrations for a firearm slide
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IL325861A (en) * 2023-07-17 2026-03-01 Kura Oncology Inc Crystalline forms of menin inhibitor
TW202517650A (zh) * 2023-07-17 2025-05-01 美商庫拉腫瘤技術股份有限公司 包含ｍｅｎｉｎ抑制劑之醫藥組合物

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US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
IE49881B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates
KR830001903B1 (ko) * 1979-02-13 1983-09-19 레오 파마슈티칼 프로덕츠 리미티드 페니실란산유도체의 제조방법
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IE51516B1 (en) * 1980-10-06 1987-01-07 Leo Pharm Prod Ltd 1,1-dioxapenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate napsylate
GB2084572B (en) * 1980-10-06 1984-07-11 Leo Pharm Prod Ltd 1,1-dioxopenicillanoyloxymethyl 6-(d-aphenylacetamido)penicillanate napsylate
IL64009A (en) * 1980-10-31 1984-09-30 Rech Applications Therap Crystalline 1,1-dioxopenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate tosylate hydrates,their production and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
SU1138030A3 (ru) 1985-01-30
FI831392L (fi) 1983-10-24
PH18035A (en) 1985-03-06
FI76092C (fi) 1988-09-09
YU90483A (en) 1986-04-30
DD209632A5 (de) 1984-05-16
HU187068B (en) 1985-11-28
EP0092968A1 (en) 1983-11-02
IE54628B1 (en) 1989-12-20
PT76587A (en) 1983-05-01
FI76092B (fi) 1988-05-31
ES521728A0 (es) 1984-07-01
NO156202B (no) 1987-05-04
EP0092968B1 (en) 1986-03-12
AU1387183A (en) 1983-11-17
JPS58201792A (ja) 1983-11-24
ZA832845B (en) 1984-11-28
YU43170B (en) 1989-04-30
IL68453A0 (en) 1983-07-31
NO156202C (no) 1987-08-19
KR840004437A (ko) 1984-10-15
GR78582B (https=) 1984-09-27
DK162168B (da) 1991-09-23
DK162168C (da) 1992-03-02
DE3362502D1 (en) 1986-04-17
NO831430L (no) 1983-10-24
NZ203988A (en) 1986-01-24
CA1187484A (en) 1985-05-21
EG16412A (en) 1989-03-30
PT76587B (en) 1986-02-27
PL241553A1 (en) 1983-11-21
SG104087G (en) 1988-07-15
PL134978B1 (en) 1985-09-30
HK20588A (en) 1988-03-25
FI831392A0 (fi) 1983-04-22
DK101783A (da) 1983-10-24
IL68453A (en) 1986-08-31
KR860001279B1 (ko) 1986-09-05
CS235320B2 (en) 1985-05-15
DK101783D0 (da) 1983-02-28
ES8406075A1 (es) 1984-07-01
IE830926L (en) 1983-10-23
US4432987A (en) 1984-02-21
JPH0119395B2 (https=) 1989-04-11

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Legal Events

Date Code Title Description
MK14 Patent ceased section 143(a) (annual fees not paid) or expired