AU536854B2 - 1 1-dioxopenicillanoyl methyl penicillanate esters - Google Patents

1 1-dioxopenicillanoyl methyl penicillanate esters

Info

Publication number
AU536854B2
AU536854B2 AU13871/83A AU1387183A AU536854B2 AU 536854 B2 AU536854 B2 AU 536854B2 AU 13871/83 A AU13871/83 A AU 13871/83A AU 1387183 A AU1387183 A AU 1387183A AU 536854 B2 AU536854 B2 AU 536854B2
Authority
AU
Australia
Prior art keywords
dioxopenicillanoyl
esters
methyl penicillanate
penicillanate
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
AU13871/83A
Other languages
English (en)
Other versions
AU1387183A (en
Inventor
Wayne Ernest Barth
Vytautas John Jasys
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp SRL
Original Assignee
Pfizer Corp Belgium
Pfizer Corp SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp Belgium, Pfizer Corp SRL filed Critical Pfizer Corp Belgium
Publication of AU1387183A publication Critical patent/AU1387183A/en
Application granted granted Critical
Publication of AU536854B2 publication Critical patent/AU536854B2/en
Anticipated expiration legal-status Critical
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32—Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
AU13871/83A 1982-04-23 1983-04-22 1 1-dioxopenicillanoyl methyl penicillanate esters Expired AU536854B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/371,156 US4432987A (en) 1982-04-23 1982-04-23 Crystalline benzenesulfonate salts of sultamicillin
US371156 1999-08-09

Publications (2)

Publication Number Publication Date
AU1387183A AU1387183A (en) 1983-11-17
AU536854B2 true AU536854B2 (en) 1984-05-24

Family

ID=23462725

Family Applications (1)

Application Number Title Priority Date Filing Date
AU13871/83A Expired AU536854B2 (en) 1982-04-23 1983-04-22 1 1-dioxopenicillanoyl methyl penicillanate esters

Country Status (27)

Country Link
US (1) US4432987A (OSRAM)
EP (1) EP0092968B1 (OSRAM)
JP (1) JPS58201792A (OSRAM)
KR (1) KR860001279B1 (OSRAM)
AU (1) AU536854B2 (OSRAM)
CA (1) CA1187484A (OSRAM)
CS (1) CS235320B2 (OSRAM)
DD (1) DD209632A5 (OSRAM)
DE (1) DE3362502D1 (OSRAM)
DK (1) DK162168C (OSRAM)
EG (1) EG16412A (OSRAM)
ES (1) ES8406075A1 (OSRAM)
FI (1) FI76092C (OSRAM)
GR (1) GR78582B (OSRAM)
HK (1) HK20588A (OSRAM)
HU (1) HU187068B (OSRAM)
IE (1) IE54628B1 (OSRAM)
IL (1) IL68453A (OSRAM)
NO (1) NO156202C (OSRAM)
NZ (1) NZ203988A (OSRAM)
PH (1) PH18035A (OSRAM)
PL (1) PL134978B1 (OSRAM)
PT (1) PT76587B (OSRAM)
SG (1) SG104087G (OSRAM)
SU (1) SU1138030A3 (OSRAM)
YU (1) YU43170B (OSRAM)
ZA (1) ZA832845B (OSRAM)

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CN1048248C (zh) * 1994-05-02 2000-01-12 盐野义制药株式会社 吡咯烷基硫基碳代青霉烯衍生物的结晶、含该结晶的冷冻干燥制剂及其制造方法
JP3382159B2 (ja) * 1998-08-05 2003-03-04 株式会社東芝 情報記録媒体とその再生方法及び記録方法
UA78104C2 (en) 2002-08-29 2007-02-15 Taisho Pharmaceutical Co Ltd Benzenesulfonate salts of 4-fluoro-2-cyanopyrrolidine derivatives
DE602004022643D1 (de) * 2003-03-27 2009-10-01 Basilea Pharmaceutica Ag Cephalosporin in kristalliner form
US20050163849A1 (en) * 2003-10-31 2005-07-28 Wong Patrick S. Compositions and dosage forms for enhanced absorption of iron
FR2877696B1 (fr) 2004-11-09 2009-09-18 Renault Sas Dispositif et procede d'estimation en temps reel de l'angle de debut de combustion d'un moteur a combustion interne
ES2442926T3 (es) 2007-08-22 2014-02-14 Astrazeneca Ab Derivados de ciclopropilamida `978
US8680291B2 (en) 2007-10-26 2014-03-25 The Regents Of The University Of California Diarylhydantoin compounds
UA106740C2 (uk) * 2009-01-30 2014-10-10 Глаксосмітклайн Ллс Кристалічний гідрохлорид n-{(1s)-2-аміно-1-[(3-фторфеніл)метил]етил}-5-хлор-4-(4-хлор-1-метил-1h-піразол-5-іл)-2-тіофенкарбоксаміду
TW201039825A (en) 2009-02-20 2010-11-16 Astrazeneca Ab Cyclopropyl amide derivatives 983
KR20120079054A (ko) * 2009-07-10 2012-07-11 에볼바 아게 디인 조성물
AR080203A1 (es) * 2010-02-18 2012-03-21 Astrazeneca Ab Formas solidas que comprenden una ciclopropilamida
NZ602110A (en) * 2010-02-18 2014-09-26 Astrazeneca Ab Processes for making cyclopropyl amide derivatives and intermediates associated therewith
CN104903289B (zh) * 2012-12-03 2017-06-09 株式会社钟化 还元型辅酶q10衍生物及其制造方法
EP3042893B1 (en) * 2013-09-05 2018-10-31 Mitsubishi Tanabe Pharma Corporation Novel crystalline arylalkylamine compound and method for producing same
SG11201702980QA (en) 2014-10-21 2017-05-30 Ariad Pharma Inc Crystalline forms of 5-chloro-n4-[-2-(dimethylphosphoryl) phenyl]-n2-{2-methoxy-4-[4-(4-methylpiperazin-1-yl) piperidin-1-yl] pyrimidine-2,4-diamine
CN104958318A (zh) * 2015-08-04 2015-10-07 青岛蓝盛洋医药生物科技有限责任公司 一种治疗感染性疾病的药物舒巴坦钠组合物
WO2017125557A1 (en) * 2016-01-22 2017-07-27 Sandoz Ag Crystalline eravacycline bis-hydrochloride
EP3481820B1 (en) 2016-07-07 2023-10-18 Cyclerion Therapeutics, Inc. Solid forms of an sgc stimulator
EP3703686A4 (en) * 2017-10-30 2021-11-17 Theracaine LLC HYDROPHOBIC ARENE SULFONATE SALTS
US11186556B1 (en) * 2018-10-16 2021-11-30 Celgene Corporation Salts of a thiazolidinone compound, solid forms, compositions and methods of use thereof
UA119735C2 (uk) 2018-12-20 2019-07-25 Анатолій Семенович Редер Фармацевтична сполука, спосіб її отримання та застосування як лікарського засобу
USD1077123S1 (en) 2019-02-13 2025-05-27 Hs Produkt D.O.O. Firearm sight
USD998740S1 (en) 2019-02-13 2023-09-12 Hs Produkt D.O.O. Firearm
USD1071069S1 (en) 2019-02-13 2025-04-15 Hs Produkt D.O.O. Stippled textured body for a firearm or the like
USD994821S1 (en) 2019-02-13 2023-08-08 Hs Produkt D.O.O. Pistol
USD1057880S1 (en) 2019-08-09 2025-01-14 Hs Produkt D.O.O. Pistol
JP2024506382A (ja) * 2021-02-15 2024-02-13 プロペラ セラピューティクス インコーポレイテッド アビラテロンプロドラッグ
USD1049292S1 (en) * 2021-04-06 2024-10-29 Springfield, Inc. Pistol
MX2023012156A (es) * 2021-05-14 2023-10-26 Global Blood Therapeutics Inc Formas solidas de un modulador de hemoglobina.
USD1069964S1 (en) 2021-11-03 2025-04-08 Hs Produkt D.O.O. Pistol slide
US12410155B2 (en) * 2021-12-28 2025-09-09 Zhejiang Yangli Pharmaceutical Technology Co., Ltd. Salt form and crystal form of tetrahydrocyclohepta indazole compound
USD1057882S1 (en) 2022-08-29 2025-01-14 Springfield, Inc. Combined serrations for a firearm slide
USD1072997S1 (en) 2022-08-29 2025-04-29 Springfield, Inc. Firearm
USD1061781S1 (en) 2022-11-30 2025-02-11 Hs Produkt D.O.O. Pistol
ZAA202301175S (en) 2023-04-28 2024-06-26 Hs Produkt D O O Firearm
TW202517651A (zh) * 2023-07-17 2025-05-01 美商庫拉腫瘤技術股份有限公司 Menin抑制劑之晶型

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US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
ZA80796B (en) * 1979-02-13 1981-02-25 Leo Pharm Prod Ltd Chemical compounds
IE49881B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
IE51516B1 (en) * 1980-10-06 1987-01-07 Leo Pharm Prod Ltd 1,1-dioxapenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate napsylate
GB2084572B (en) * 1980-10-06 1984-07-11 Leo Pharm Prod Ltd 1,1-dioxopenicillanoyloxymethyl 6-(d-aphenylacetamido)penicillanate napsylate
IL64009A (en) * 1980-10-31 1984-09-30 Rech Applications Therap Crystalline 1,1-dioxopenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate tosylate hydrates,their production and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
SG104087G (en) 1988-07-15
YU43170B (en) 1989-04-30
FI76092C (fi) 1988-09-09
US4432987A (en) 1984-02-21
HK20588A (en) 1988-03-25
NO831430L (no) 1983-10-24
NZ203988A (en) 1986-01-24
DK101783A (da) 1983-10-24
HU187068B (en) 1985-11-28
NO156202C (no) 1987-08-19
JPH0119395B2 (OSRAM) 1989-04-11
FI831392L (fi) 1983-10-24
DK162168B (da) 1991-09-23
IL68453A0 (en) 1983-07-31
EP0092968A1 (en) 1983-11-02
IL68453A (en) 1986-08-31
FI76092B (fi) 1988-05-31
CA1187484A (en) 1985-05-21
SU1138030A3 (ru) 1985-01-30
ES521728A0 (es) 1984-07-01
PL134978B1 (en) 1985-09-30
DK101783D0 (da) 1983-02-28
AU1387183A (en) 1983-11-17
EG16412A (en) 1989-03-30
YU90483A (en) 1986-04-30
PL241553A1 (en) 1983-11-21
CS235320B2 (en) 1985-05-15
PH18035A (en) 1985-03-06
IE54628B1 (en) 1989-12-20
DK162168C (da) 1992-03-02
IE830926L (en) 1983-10-23
NO156202B (no) 1987-05-04
PT76587A (en) 1983-05-01
ES8406075A1 (es) 1984-07-01
PT76587B (en) 1986-02-27
KR840004437A (ko) 1984-10-15
FI831392A0 (fi) 1983-04-22
KR860001279B1 (ko) 1986-09-05
DE3362502D1 (en) 1986-04-17
EP0092968B1 (en) 1986-03-12
DD209632A5 (de) 1984-05-16
ZA832845B (en) 1984-11-28
GR78582B (OSRAM) 1984-09-27
JPS58201792A (ja) 1983-11-24

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Legal Events

Date Code Title Description
MK14 Patent ceased section 143(a) (annual fees not paid) or expired