AU2020236225B2 - Salts of a isochromanyl compound and crystalline forms, processes for preparing, therapeutic uses, and pharmaceutical compositions thereof - Google Patents

Salts of a isochromanyl compound and crystalline forms, processes for preparing, therapeutic uses, and pharmaceutical compositions thereof

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Publication number
AU2020236225B2
AU2020236225B2 AU2020236225A AU2020236225A AU2020236225B2 AU 2020236225 B2 AU2020236225 B2 AU 2020236225B2 AU 2020236225 A AU2020236225 A AU 2020236225A AU 2020236225 A AU2020236225 A AU 2020236225A AU 2020236225 B2 AU2020236225 B2 AU 2020236225B2
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AU
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Prior art keywords
compound
salt
disorder
terms
disease
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AU2020236225A
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English (en)
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AU2020236225A1 (en
Inventor
Nandkumar Nivritti BHOGLE
Takahiko Hashizuka
Robert Joseph PRYTKO
John R. Snoonian
Harold Scott Wilkinson
Haitao Zhang
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sumitomo Pharma America Inc
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Sumitomo Pharma America Inc
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Publication of AU2020236225A1 publication Critical patent/AU2020236225A1/en
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Priority to AU2026200097A priority Critical patent/AU2026200097A1/en
Assigned to SUMITOMO PHARMA AMERICA, INC. reassignment SUMITOMO PHARMA AMERICA, INC. Request for Assignment Assignors: SUNOVION PHARMACEUTICALS INC.
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Anticipated expiration legal-status Critical

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/76—Benzo[c]pyrans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hospice & Palliative Care (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2020236225A 2019-03-14 2020-03-13 Salts of a isochromanyl compound and crystalline forms, processes for preparing, therapeutic uses, and pharmaceutical compositions thereof Active AU2020236225B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2026200097A AU2026200097A1 (en) 2019-03-14 2026-01-08 Salts of a isochromanyl compound and crystalline forms, processes for preparing, therapeutic uses, and pharmaceutical compositions thereof

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962818256P 2019-03-14 2019-03-14
US62/818,256 2019-03-14
PCT/US2020/022642 WO2020186165A1 (en) 2019-03-14 2020-03-13 Salts of a isochromanyl compound and crystalline forms, processes for preparing, therapeutic uses, and pharmaceutical compositions thereof

Related Child Applications (1)

Application Number Title Priority Date Filing Date
AU2026200097A Division AU2026200097A1 (en) 2019-03-14 2026-01-08 Salts of a isochromanyl compound and crystalline forms, processes for preparing, therapeutic uses, and pharmaceutical compositions thereof

Publications (2)

Publication Number Publication Date
AU2020236225A1 AU2020236225A1 (en) 2021-09-16
AU2020236225B2 true AU2020236225B2 (en) 2025-12-18

Family

ID=70277473

Family Applications (2)

Application Number Title Priority Date Filing Date
AU2020236225A Active AU2020236225B2 (en) 2019-03-14 2020-03-13 Salts of a isochromanyl compound and crystalline forms, processes for preparing, therapeutic uses, and pharmaceutical compositions thereof
AU2026200097A Pending AU2026200097A1 (en) 2019-03-14 2026-01-08 Salts of a isochromanyl compound and crystalline forms, processes for preparing, therapeutic uses, and pharmaceutical compositions thereof

Family Applications After (1)

Application Number Title Priority Date Filing Date
AU2026200097A Pending AU2026200097A1 (en) 2019-03-14 2026-01-08 Salts of a isochromanyl compound and crystalline forms, processes for preparing, therapeutic uses, and pharmaceutical compositions thereof

Country Status (9)

Country Link
US (3) US11136304B2 (https=)
EP (1) EP3938045A1 (https=)
JP (2) JP7703449B2 (https=)
KR (1) KR20210139376A (https=)
CN (1) CN113784755B (https=)
AU (2) AU2020236225B2 (https=)
CA (1) CA3130849A1 (https=)
MX (2) MX2021010880A (https=)
WO (1) WO2020186165A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA125519C2 (uk) 2016-07-29 2022-04-13 Суновіон Фармасьютікалз Інк. Сполуки і композиції і їх застосування

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2018023072A2 (en) * 2016-07-29 2018-02-01 Sunovion Pharmaceuticals, Inc. Compounds and compositions and uses thereof

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