AU2014272924B2 - Dihydroetorphine for the provision of pain relief and anaesthesia - Google Patents
Dihydroetorphine for the provision of pain relief and anaesthesia Download PDFInfo
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- AU2014272924B2 AU2014272924B2 AU2014272924A AU2014272924A AU2014272924B2 AU 2014272924 B2 AU2014272924 B2 AU 2014272924B2 AU 2014272924 A AU2014272924 A AU 2014272924A AU 2014272924 A AU2014272924 A AU 2014272924A AU 2014272924 B2 AU2014272924 B2 AU 2014272924B2
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- dihydroetorphine
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- medicament
- human subject
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P23/00—Anaesthetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D489/00—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
- C07D489/09—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems
- C07D489/10—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems with a bridge between positions 6 and 14
- C07D489/12—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems with a bridge between positions 6 and 14 the bridge containing only two carbon atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
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- Emergency Medicine (AREA)
- General Chemical & Material Sciences (AREA)
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- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
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- Pain & Pain Management (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Physics & Mathematics (AREA)
- Biophysics (AREA)
- Pathology (AREA)
- Heart & Thoracic Surgery (AREA)
- Medical Informatics (AREA)
- Molecular Biology (AREA)
- Surgery (AREA)
- Dermatology (AREA)
Applications Claiming Priority (3)
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|---|---|---|---|
| GB1309654.0 | 2013-05-30 | ||
| GBGB1309654.0A GB201309654D0 (en) | 2013-05-30 | 2013-05-30 | Method |
| PCT/GB2014/000206 WO2014191710A1 (en) | 2013-05-30 | 2014-05-30 | Dihydroetorphine for the provision of pain relief and anaesthesia |
Publications (2)
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| AU2014272924A1 AU2014272924A1 (en) | 2016-01-28 |
| AU2014272924B2 true AU2014272924B2 (en) | 2019-05-02 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2014272924A Ceased AU2014272924B2 (en) | 2013-05-30 | 2014-05-30 | Dihydroetorphine for the provision of pain relief and anaesthesia |
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| Country | Link |
|---|---|
| US (2) | US10898479B2 (enExample) |
| EP (1) | EP3003310A1 (enExample) |
| JP (3) | JP2016520114A (enExample) |
| KR (1) | KR20160013977A (enExample) |
| CN (1) | CN105555274A (enExample) |
| AU (1) | AU2014272924B2 (enExample) |
| BR (1) | BR112015029709A2 (enExample) |
| CA (1) | CA2913849A1 (enExample) |
| GB (1) | GB201309654D0 (enExample) |
| HK (1) | HK1222585A1 (enExample) |
| MX (1) | MX2015016418A (enExample) |
| PH (1) | PH12015502655A1 (enExample) |
| WO (1) | WO2014191710A1 (enExample) |
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| CN107847471A (zh) | 2015-03-27 | 2018-03-27 | 格吕伦塔尔有限公司 | 他喷他多肠胃外给药的稳定制剂 |
| GB201513442D0 (en) * | 2015-07-30 | 2015-09-16 | Euro Celtique Sa | Transdermal patch |
| PE20190908A1 (es) | 2016-09-23 | 2019-06-26 | Gruenenthal Chemie | Formulacion estable para la administracion parenteral de tapentadol |
| EP3585370A1 (en) | 2017-02-23 | 2020-01-01 | Grünenthal GmbH | Tapentadol as local anesthetic |
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| GB925723A (en) | 1960-09-05 | 1963-05-08 | J F Macfarlan & Company Ltd | Novel thebaine derivatives |
| GB937214A (en) | 1961-06-02 | 1963-09-18 | J F Macfarlan & Company Ltd | Oripavine derivatives |
| JPS59184182A (ja) | 1983-04-02 | 1984-10-19 | Res Inst For Prod Dev | ３−ベンゾイルチオ−４、５α−エポキシ−７α−〔１（Ｒ）−ヒドロキシ−１−メチルベンチル〕−６−メトキシ−１７−メチル−６、１４−エンド−エタノモルヒナン |
| JPS62153214A (ja) | 1985-12-26 | 1987-07-08 | Nitto Electric Ind Co Ltd | 医薬製剤 |
| JPS62281815A (ja) | 1986-05-27 | 1987-12-07 | Teisan Seiyaku Kk | 貼付剤及びその製造法 |
| JPS63201119A (ja) | 1987-02-17 | 1988-08-19 | Kao Corp | 貼付剤組成物 |
| US4891377A (en) | 1988-12-02 | 1990-01-02 | Board Of Regents Acting For And On Behalf Of University Of Michigan | Transdermal delivery of the narcotic analgesics etorphine and analogs |
| PT95069B (pt) | 1989-08-24 | 1997-10-31 | Searle & Co | Processo para a preparacao de (+)-isomeros de derivados de endoetano/endoetanoepoximofinano, uteis como agentes anti-tussicos |
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| WO1994006426A1 (en) | 1992-09-21 | 1994-03-31 | Qin Bo Yi | Methods for identifying and using low/non-addictive opioid analgesics |
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| JP2819236B2 (ja) | 1994-05-06 | 1998-10-30 | 日東電工株式会社 | 経皮吸収製剤 |
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| AUPN603895A0 (en) | 1995-10-19 | 1995-11-09 | University Of Queensland, The | Production of analgesic synergy by co-administration of sub-analgesic doses of two strong opioids |
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- 2013-05-30 GB GBGB1309654.0A patent/GB201309654D0/en not_active Ceased
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2014
- 2014-05-30 MX MX2015016418A patent/MX2015016418A/es unknown
- 2014-05-30 KR KR1020157036442A patent/KR20160013977A/ko not_active Ceased
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- 2014-05-30 CN CN201480042250.XA patent/CN105555274A/zh active Pending
- 2014-05-30 BR BR112015029709A patent/BR112015029709A2/pt not_active IP Right Cessation
- 2014-05-30 JP JP2016516232A patent/JP2016520114A/ja active Pending
- 2014-05-30 AU AU2014272924A patent/AU2014272924B2/en not_active Ceased
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2015
- 2015-11-27 PH PH12015502655A patent/PH12015502655A1/en unknown
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2019
- 2019-03-19 JP JP2019051613A patent/JP2019123730A/ja active Pending
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2020
- 2020-09-17 JP JP2020156242A patent/JP2020200345A/ja active Pending
- 2020-09-30 US US17/038,651 patent/US20210085673A1/en not_active Abandoned
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| JP2016520114A (ja) | 2016-07-11 |
| US10898479B2 (en) | 2021-01-26 |
| US20160106736A1 (en) | 2016-04-21 |
| JP2020200345A (ja) | 2020-12-17 |
| MX2015016418A (es) | 2016-11-08 |
| PH12015502655A1 (en) | 2016-03-07 |
| EP3003310A1 (en) | 2016-04-13 |
| BR112015029709A2 (pt) | 2017-07-25 |
| GB201309654D0 (en) | 2013-07-17 |
| AU2014272924A1 (en) | 2016-01-28 |
| KR20160013977A (ko) | 2016-02-05 |
| HK1222585A1 (zh) | 2017-07-07 |
| CA2913849A1 (en) | 2014-12-04 |
| US20210085673A1 (en) | 2021-03-25 |
| CN105555274A (zh) | 2016-05-04 |
| JP2019123730A (ja) | 2019-07-25 |
| WO2014191710A1 (en) | 2014-12-04 |
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