AU2009330821B2 - Pharmaceutical compounds - Google Patents

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Publication number
AU2009330821B2
AU2009330821B2 AU2009330821A AU2009330821A AU2009330821B2 AU 2009330821 B2 AU2009330821 B2 AU 2009330821B2 AU 2009330821 A AU2009330821 A AU 2009330821A AU 2009330821 A AU2009330821 A AU 2009330821A AU 2009330821 B2 AU2009330821 B2 AU 2009330821B2
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Australia
Prior art keywords
alkyl
heterocyclyl
aryl
heteroaryl
substituted
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Ceased
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AU2009330821A
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AU2009330821A1 (en
Inventor
Alexander Beliaev
Rita Gusmao De Noronha
Laszlo Erno Kiss
David Alexander Learmonth
Pedro Nuno Leal Palma
Carla Patricia Da Costa Pereira Rosa
Patricio Manuel Vieira Araujo Soares Da Silva
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Bial Portela and Cia SA
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Bial Portela and Cia SA
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Application filed by Bial Portela and Cia SA filed Critical Bial Portela and Cia SA
Publication of AU2009330821A1 publication Critical patent/AU2009330821A1/en
Application granted granted Critical
Publication of AU2009330821B2 publication Critical patent/AU2009330821B2/en
Priority to AU2015224424A priority Critical patent/AU2015224424A1/en
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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