AU2006246374B2 - Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids - Google Patents

Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids Download PDF

Info

Publication number
AU2006246374B2
AU2006246374B2 AU2006246374A AU2006246374A AU2006246374B2 AU 2006246374 B2 AU2006246374 B2 AU 2006246374B2 AU 2006246374 A AU2006246374 A AU 2006246374A AU 2006246374 A AU2006246374 A AU 2006246374A AU 2006246374 B2 AU2006246374 B2 AU 2006246374B2
Authority
AU
Australia
Prior art keywords
formula
compound
acid
optionally substituted
water
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
AU2006246374A
Other languages
English (en)
Other versions
AU2006246374A1 (en
Inventor
Rafael Shapiro
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Corteva Agriscience LLC
Original Assignee
Corteva Agriscience LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Corteva Agriscience LLC filed Critical Corteva Agriscience LLC
Publication of AU2006246374A1 publication Critical patent/AU2006246374A1/en
Application granted granted Critical
Publication of AU2006246374B2 publication Critical patent/AU2006246374B2/en
Assigned to CORTEVA AGRISCIENCE LLC reassignment CORTEVA AGRISCIENCE LLC Request for Assignment Assignors: E. I. DU PONT DE NEMOURS AND COMPANY
Anticipated expiration legal-status Critical
Active legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AU2006246374A 2005-05-06 2006-04-28 Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids Active AU2006246374B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US67826405P 2005-05-06 2005-05-06
US60/678,264 2005-05-06
PCT/US2006/016340 WO2006121648A2 (en) 2005-05-06 2006-04-28 Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids

Publications (2)

Publication Number Publication Date
AU2006246374A1 AU2006246374A1 (en) 2006-11-16
AU2006246374B2 true AU2006246374B2 (en) 2012-03-29

Family

ID=36952291

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2006246374A Active AU2006246374B2 (en) 2005-05-06 2006-04-28 Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids

Country Status (25)

Country Link
US (2) US8198442B2 (https=)
EP (1) EP1877384B1 (https=)
JP (1) JP5161764B2 (https=)
KR (1) KR101379967B1 (https=)
CN (2) CN101171237B (https=)
AT (1) ATE506352T1 (https=)
AU (1) AU2006246374B2 (https=)
BR (1) BRPI0612475B8 (https=)
CA (1) CA2607934C (https=)
DE (1) DE602006021411D1 (https=)
DK (1) DK1877384T3 (https=)
EG (1) EG25480A (https=)
ES (1) ES2362005T3 (https=)
GE (1) GEP20105099B (https=)
IL (2) IL185885A (https=)
MA (1) MA29464B1 (https=)
ME (1) ME00498B (https=)
MX (1) MX2007013424A (https=)
NZ (1) NZ561399A (https=)
PL (1) PL1877384T3 (https=)
RS (2) RS51804B (https=)
TN (1) TNSN07403A1 (https=)
UA (1) UA92171C2 (https=)
WO (1) WO2006121648A2 (https=)
ZA (1) ZA200707975B (https=)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5069677B2 (ja) * 2005-05-16 2012-11-07 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー 置換ピリミジンの製造方法
CN101277927A (zh) * 2005-09-29 2008-10-01 帝斯曼知识产权资产管理有限公司 用于酯化有机酸的方法
ES2400405T3 (es) * 2007-08-13 2013-04-09 Dow Agrosciences Llc 2-(Fenil 2-fluoro-substituido)-6-amino-5-cloro-4-pirimidinacarboxilatos y su uso como herbicidas
CA2699598C (en) 2007-10-02 2013-05-21 Dow Agrosciences Llc 2-substituted-6-amino-5-alkyl, alkenyl or alkynyl-4-pyrimidinecarboxylic acids and 6-substituted-4-amino-3-alkyl, alkenyl or alkynyl picolinic acids and their use as herbicides
EP2279178B1 (en) * 2008-04-18 2015-05-20 Dow AgroSciences LLC 2-(substituted phenyl)-6-hydroxy- or alkoxy-5-substituted-4-pyrimidinecarboxylates and their use as herbicides
TWI596088B (zh) * 2011-01-25 2017-08-21 陶氏農業科學公司 4-胺基-6-(經取代的苯基)吡啶甲酸酯及6-胺基-2-(經取代的苯基)-4-嘧啶羧酸酯之芳烷酯以及其等作為除草劑之用途
ES2561887T3 (es) * 2011-07-27 2016-03-01 Bayer Intellectual Property Gmbh Ácidos picolínicos y piridimin-4-carboxílicos sustituidos, procedimiento para su preparación y su uso como herbicidas y reguladores del crecimiento de plantas
US9113629B2 (en) * 2013-03-15 2015-08-25 Dow Agrosciences Llc 4-amino-6-(4-substituted-phenyl)-picolinates and 6-amino-2-(4-substituted-phenyl)-pyrimidine-4-carboxylates and their use as herbicides
CN110583663A (zh) * 2013-03-15 2019-12-20 美国陶氏益农公司 式(i)化合物及其作为除草剂的用途
US9637505B2 (en) 2013-03-15 2017-05-02 Dow Agrosciences Llc 4-amino-6-(heterocyclic)picolinates and 6-amino-2-(heterocyclic)pyrimidine-4-carboxylates and their use as herbicides
TWI685302B (zh) 2014-09-15 2020-02-21 美商陶氏農業科學公司 包含吡啶羧酸除草劑之安全的除草組成物
TWI689251B (zh) 2014-09-15 2020-04-01 美商陶氏農業科學公司 源自於施用吡啶羧酸除草劑與合成生長素除草劑及/或生長素轉運抑制劑的協同性雜草控制
US10455836B2 (en) 2014-09-15 2019-10-29 Dow Agrosciences Llc Synergistic weed control from applications of pyridine carboxylic acid herbicides and photosystem II inhibitors
TWI694770B (zh) 2014-09-15 2020-06-01 美商陶氏農業科學公司 包含吡啶羧酸除草劑之安全的除草組成物(二)
TWI689252B (zh) 2014-09-15 2020-04-01 美商陶氏農業科學公司 源自於施用吡啶羧酸除草劑與乙醯乳酸合成酶(als)抑制劑的協同性雜草控制
WO2026028053A2 (en) 2024-07-27 2026-02-05 Assia Chemical Industries Ltd. Process for the preparation of tovorafenib

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA207185A (en) 1921-01-04 C. Wagner Virgil Warming plate
JPS60100559A (ja) * 1983-11-05 1985-06-04 Morishita Seiyaku Kk 2−アニリノ−1,6−ジヒドロ−6−オキソ−5−ピリミジンカルボン酸誘導体,その製法及び該化合物を含有する抗アレルギ−剤
JPH0331267A (ja) 1989-06-28 1991-02-12 Morishita Pharmaceut Co Ltd 2―アニリノ―1,6―ジヒドロ―6―オキソ―4―ピリミジンカルボン酸誘導体
JPH0341071A (ja) 1989-07-06 1991-02-21 Morishita Pharmaceut Co Ltd 1,6―ジヒドロ―6―オキソ―2―フェノキシアルキルチオ―5―ピリミジンカルボン酸類
DE3935277A1 (de) * 1989-10-24 1991-05-02 Hoechst Ag Sulfonierte heterocyclische carboxamide, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als herbizide oder wachstumsregulatoren
US5637618A (en) * 1990-06-01 1997-06-10 Bioresearch, Inc. Specific eatable taste modifiers
DE4029654A1 (de) 1990-09-19 1992-04-02 Hoechst Ag 2-phenyl-pyrimidine, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als fungizide
DE4131924A1 (de) * 1991-09-25 1993-07-08 Hoechst Ag Substituierte 4-alkoxypyrimidine, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
DE4408404A1 (de) * 1994-03-12 1995-09-14 Huels Chemische Werke Ag Verfahren zur Herstellung von Chlorpyrimidinen
BR9908004A (pt) 1998-02-17 2001-12-18 Tularik Inc Composto, composição e método para prevençãoou supressão de uma infecção viral
US6281358B1 (en) 1999-04-15 2001-08-28 American Cyanamid Company Process for the preparation of substituted pyrimidines
ES2240093T3 (es) 1999-04-15 2005-10-16 Basf Aktiengesellschaft Procedimiento para la preparacion de pirimidinas substituidas.
AU2002258400A1 (en) 2001-02-16 2002-08-28 Tularik Inc. Methods of using pyrimidine-based antiviral agents
DE602004022819D1 (de) 2003-06-06 2009-10-08 Vertex Pharma Von atp-bindende kassette transportern
TWI355894B (en) * 2003-12-19 2012-01-11 Du Pont Herbicidal pyrimidines
EP1849765A4 (en) 2005-02-02 2010-05-05 Ajinomoto Kk PROCESS FOR PREPARING A PYRIMIDINE COMPOUND
DE102005027150A1 (de) 2005-03-12 2006-09-28 Bayer Healthcare Ag Pyrimidincarbonsäure-Derivate und ihre Verwendung
JP5069677B2 (ja) * 2005-05-16 2012-11-07 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー 置換ピリミジンの製造方法

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
J. Org. Chem., vol 26, 1961, p2755-2763 *

Also Published As

Publication number Publication date
TNSN07403A1 (en) 2009-03-17
EP1877384B1 (en) 2011-04-20
IL222041A (en) 2016-10-31
BRPI0612475A2 (pt) 2010-11-23
DE602006021411D1 (de) 2011-06-01
EG25480A (en) 2012-01-15
MA29464B1 (fr) 2008-05-02
GEP20105099B (en) 2010-10-25
US8198442B2 (en) 2012-06-12
CN102153516B (zh) 2013-02-06
BRPI0612475B8 (pt) 2022-12-06
BRPI0612475B1 (pt) 2020-03-10
CA2607934A1 (en) 2006-11-16
WO2006121648A3 (en) 2006-12-28
JP5161764B2 (ja) 2013-03-13
NZ561399A (en) 2009-11-27
ES2362005T3 (es) 2011-06-27
ME00498B (me) 2011-10-10
ATE506352T1 (de) 2011-05-15
ZA200707975B (en) 2008-11-26
JP2008540414A (ja) 2008-11-20
PL1877384T3 (pl) 2011-09-30
RS51804B (sr) 2011-12-31
UA92171C2 (ru) 2010-10-11
US20120232271A1 (en) 2012-09-13
AU2006246374A1 (en) 2006-11-16
KR20080006576A (ko) 2008-01-16
WO2006121648A2 (en) 2006-11-16
MX2007013424A (es) 2008-01-16
CA2607934C (en) 2013-10-01
US20090043098A1 (en) 2009-02-12
DK1877384T3 (da) 2011-08-15
KR101379967B1 (ko) 2014-04-01
IL185885A (en) 2012-10-31
EP1877384A2 (en) 2008-01-16
RS20070434A (sr) 2009-01-22
IL185885A0 (en) 2008-01-06
CN101171237A (zh) 2008-04-30
CN101171237B (zh) 2011-04-20
CN102153516A (zh) 2011-08-17

Similar Documents

Publication Publication Date Title
US20120232271A1 (en) Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids
EP2334645B1 (en) Process for the synthesis of fluorinated cyclic compounds
WO1997048684A1 (en) Preparation of fungicidal quinazolinones and useful intermediates
WO2005063780A1 (en) Process for the preparation of pyridine derivatives
KR100585407B1 (ko) 피리딘-2,3-디카복실레이트 화합물의 제조를 위한 방법 및중간체
KR20190006960A (ko) 제초성 화합물의 제조 방법
EP1215206A1 (en) Processes for the preparation of 4(5)-amino-5(4)-carboxamidoimidazoles and intermediates thereof
EP0819114B1 (en) An arthropodicidal oxadiazine intermediate
JP2024503801A (ja) N-(3-クロロ-1-(ピリジン-3-イル)-1h-ピラゾール-4-イル)-2-(メチルスルホニル)プロパンアミドの形成に関連する方法
KR100361825B1 (ko) 치환된 5-(4,6-디메톡시피리미딘-2-일)옥시-4h-(1,3)-벤조디옥신-4-온 유도체를 이용한 제초성 피리미딜옥시 벤조산 옥심에스테 르 유도체의 제조방법
SK55497A3 (en) Effective and enantiomerically high-selective method for producing enantiomerically pure cyclopentane-beta-amino acids
MXPA06007401A (es) Proceso para la preparacion de derivados de piridina
PL209522B1 (pl) Sposób wytwarzania związku pirydonowego

Legal Events

Date Code Title Description
FGA Letters patent sealed or granted (standard patent)
PC Assignment registered

Owner name: CORTEVA AGRISCIENCE LLC

Free format text: FORMER OWNER(S): E. I. DU PONT DE NEMOURS AND COMPANY